Progress in the development of histamine H3 receptor antagonists/inverse agonists: a patent review (2013-2017)

2018 ◽  
Vol 28 (3) ◽  
pp. 175-196 ◽  
Author(s):  
Dorota Łażewska ◽  
Katarzyna Kieć-Kononowicz
Keyword(s):  
Receptor Antagonists ◽  
Histamine H3 Receptor ◽  
Inverse Agonists ◽  
H3 Receptor ◽  
Patent Review ◽  
Histamine H3

Histamine H3 receptor antagonists/inverse agonists: Where do they go?

2019 ◽  
Vol 200 ◽  
pp. 69-84 ◽  
Author(s):  
Nakisa Ghamari ◽  
Omid Zarei ◽  
José-Antonio Arias-Montaño ◽  
David Reiner ◽  
Siavoush Dastmalchi ◽  
...  
Keyword(s):  
Receptor Antagonists ◽  
Histamine H3 Receptor ◽  
Inverse Agonists ◽  
H3 Receptor ◽  
Histamine H3

Discovery of novel steroidal histamine H3 receptor antagonists/inverse agonists. Part 2. Versatile steroidal carboxamide derivatives

2019 ◽  
Vol 29 (20) ◽  
pp. 126643
Author(s):  
István Ledneczki ◽  
Zsolt Némethy ◽  
Pál Tapolcsányi ◽  
János Éles ◽  
István Greiner ◽  
...  
Keyword(s):  
Receptor Antagonists ◽  
Histamine H3 Receptor ◽  
Inverse Agonists ◽  
H3 Receptor ◽  
Histamine H3

ChemInform Abstract: 4-Chlorobenzyl Sulfonamide and Sulfamide Derivatives of Histamine Homologues: The Design of Potent Histamine H3 Receptor Antagonists.

ChemInform ◽  
2010 ◽  
Vol 31 (8) ◽  
pp. no-no
Author(s):  
Matthew J. Tozer ◽  
Ildiko M. Buck ◽  
Tracey Cooke ◽  
S. Barret Kalindjian ◽  
Iain M. McDonald ◽  
...  
Keyword(s):  
Receptor Antagonists ◽  
Histamine H3 Receptor ◽  
H3 Receptor ◽  
Derivatives Of ◽  
Histamine H3

Development of novel 2-[4-(aminoalkoxy)phenyl]-4(3H)-quinazolinone derivatives as potent and selective histamine H3 receptor inverse agonists

2008 ◽  
Vol 18 (23) ◽  
pp. 6041-6045 ◽  
Author(s):  
Takashi Mizutani ◽  
Tsuyoshi Nagase ◽  
Sayaka Ito ◽  
Yasuhisa Miyamoto ◽  
Takeshi Tanaka ◽  
...  
Keyword(s):  
Histamine H3 Receptor ◽  
Inverse Agonists ◽  
H3 Receptor ◽  
Quinazolinone Derivatives ◽  
Histamine H3

ChemInform Abstract: Substituted N-Phenylcarbamates as Histamine H3 Receptor Antagonists with Improved in vivo Potency.

ChemInform ◽  
2010 ◽  
Vol 31 (24) ◽  
pp. no-no
Author(s):  
S. Reidemeister ◽  
H. Stark ◽  
X. Ligneau ◽  
C. R. Ganellin ◽  
J.-C. Schwartz ◽  
...  
Keyword(s):  
Receptor Antagonists ◽  
Histamine H3 Receptor ◽  
H3 Receptor ◽  
Histamine H3

scholarly journals Development of a Conformational Histamine H3 Receptor Biosensor for the Synchronous Screening of Agonists and Inverse Agonists

ACS Sensors ◽  
2020 ◽  
Vol 5 (6) ◽  
pp. 1734-1742 ◽  
Author(s):  
Hannes Schihada ◽  
Xiaoyuan Ma ◽  
Ulrike Zabel ◽  
Henry F. Vischer ◽  
Gunnar Schulte ◽  
...  
Keyword(s):  
Histamine H3 Receptor ◽  
Inverse Agonists ◽  
H3 Receptor ◽  
Histamine H3

Piperidine-Containing Histamine H3 Receptor Antagonists of the Carbamate Series: The Influence of the Additional Ether Functionality

ChemInform ◽  
2003 ◽  
Vol 34 (16) ◽  
Author(s):  
D. Lazewska ◽  
K. Kiec-Kononowicz ◽  
H. H. Pertz ◽  
S. Elz ◽  
H. Stark ◽  
...  
Keyword(s):  
Receptor Antagonists ◽  
Histamine H3 Receptor ◽  
H3 Receptor ◽  
Histamine H3
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