scholarly journals Design, synthesis, and anticonvulsant effects evaluation of nonimidazole histamine H3 receptor antagonists/inverse agonists containing triazole moiety

2020 ◽  
Vol 35 (1) ◽  
pp. 1310-1321 ◽  
Author(s):  
Mingxia Song ◽  
Rui Yan ◽  
Yanhui Zhang ◽  
Dongfu Guo ◽  
Naiming Zhou ◽  
...  
Keyword(s):  
Receptor Antagonists ◽  
Design Synthesis ◽  
Histamine H3 Receptor ◽  
Inverse Agonists ◽  
H3 Receptor ◽  
Anticonvulsant Effects ◽  
Histamine H3

scholarly journals Design, synthesis, and in vitro and in vivo characterization of 1-{4-[4-(substituted)piperazin-1-yl]butyl}guanidines and their piperidine analogues as histamine H3 receptor antagonists

MedChemComm ◽  
2019 ◽  
Vol 10 (2) ◽  
pp. 234-251 ◽  
Author(s):  
Marek Staszewski ◽  
Anna Stasiak ◽  
Tadeusz Karcz ◽  
Daniel McNaught Flores ◽  
Wiesława Agnieszka Fogel ◽  
...  
Keyword(s):  
Receptor Antagonists ◽  
Design Synthesis ◽  
Histamine H3 Receptor ◽  
H3 Receptor ◽  
In Vivo Characterization ◽  
Histamine H3

The prominent members of 1-{4-[4-(substituted)piperazin-1-yl]butyl}guanidines as histamine H3 receptor antagonists.

Histamine H3 receptor antagonists/inverse agonists: Where do they go?

2019 ◽  
Vol 200 ◽  
pp. 69-84 ◽  
Author(s):  
Nakisa Ghamari ◽  
Omid Zarei ◽  
José-Antonio Arias-Montaño ◽  
David Reiner ◽  
Siavoush Dastmalchi ◽  
...  
Keyword(s):  
Receptor Antagonists ◽  
Histamine H3 Receptor ◽  
Inverse Agonists ◽  
H3 Receptor ◽  
Histamine H3

ChemInform Abstract: Design, Synthesis, and Structure-Activity Relationships of Novel Non-Imidazole Histamine H3 Receptor Antagonists.

ChemInform ◽  
2000 ◽  
Vol 31 (40) ◽  
pp. no-no
Author(s):  
Ian D. Linney ◽  
Ildiko M. Buck ◽  
Elaine A. Harper ◽  
S. Barret-Kalindjian ◽  
Michael J. Pether ◽  
...  
Keyword(s):  
Receptor Antagonists ◽  
Design Synthesis ◽  
Histamine H3 Receptor ◽  
Structure Activity Relationships ◽  
Structure Activity ◽  
H3 Receptor ◽  
Histamine H3

Discovery of novel steroidal histamine H3 receptor antagonists/inverse agonists. Part 2. Versatile steroidal carboxamide derivatives

2019 ◽  
Vol 29 (20) ◽  
pp. 126643
Author(s):  
István Ledneczki ◽  
Zsolt Némethy ◽  
Pál Tapolcsányi ◽  
János Éles ◽  
István Greiner ◽  
...  
Keyword(s):  
Receptor Antagonists ◽  
Histamine H3 Receptor ◽  
Inverse Agonists ◽  
H3 Receptor ◽  
Histamine H3

ChemInform Abstract: 4-Chlorobenzyl Sulfonamide and Sulfamide Derivatives of Histamine Homologues: The Design of Potent Histamine H3 Receptor Antagonists.

ChemInform ◽  
2010 ◽  
Vol 31 (8) ◽  
pp. no-no
Author(s):  
Matthew J. Tozer ◽  
Ildiko M. Buck ◽  
Tracey Cooke ◽  
S. Barret Kalindjian ◽  
Iain M. McDonald ◽  
...  
Keyword(s):  
Receptor Antagonists ◽  
Histamine H3 Receptor ◽  
H3 Receptor ◽  
Derivatives Of ◽  
Histamine H3

Development of novel 2-[4-(aminoalkoxy)phenyl]-4(3H)-quinazolinone derivatives as potent and selective histamine H3 receptor inverse agonists

2008 ◽  
Vol 18 (23) ◽  
pp. 6041-6045 ◽  
Author(s):  
Takashi Mizutani ◽  
Tsuyoshi Nagase ◽  
Sayaka Ito ◽  
Yasuhisa Miyamoto ◽  
Takeshi Tanaka ◽  
...  
Keyword(s):  
Histamine H3 Receptor ◽  
Inverse Agonists ◽  
H3 Receptor ◽  
Quinazolinone Derivatives ◽  
Histamine H3

ChemInform Abstract: Substituted N-Phenylcarbamates as Histamine H3 Receptor Antagonists with Improved in vivo Potency.

ChemInform ◽  
2010 ◽  
Vol 31 (24) ◽  
pp. no-no
Author(s):  
S. Reidemeister ◽  
H. Stark ◽  
X. Ligneau ◽  
C. R. Ganellin ◽  
J.-C. Schwartz ◽  
...  
Keyword(s):  
Receptor Antagonists ◽  
Histamine H3 Receptor ◽  
H3 Receptor ◽  
Histamine H3
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