Calcitonin gene-related peptide receptor antagonist olcegepant acts in the spinal trigeminal nucleus

Trigeminal Nucleus ◽

Peptide Receptor ◽

Related Peptide ◽

The Nonpeptide Calcitonin Gene-Related Peptide Receptor Antagonist BIBN4096BS Lowers the Activity of Neurons with Meningeal Input in the Rat Spinal Trigeminal Nucleus

Journal of Neuroscience ◽

10.1523/jneurosci.0869-05.2005 ◽

2005 ◽

Vol 25 (25) ◽

pp. 5877-5883 ◽

Cited By ~ 102

Author(s):

M. J. M. Fischer

Keyword(s):

Receptor Antagonist ◽

Trigeminal Nucleus ◽

Peptide Receptor ◽

Related Peptide ◽

Faculty Opinions recommendation of Calcitonin gene-related peptide receptor antagonist olcegepant acts in the spinal trigeminal nucleus.

Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature ◽

10.3410/f.2111979.1706078 ◽

2010 ◽

Author(s):

Ana Recober

Keyword(s):

Receptor Antagonist ◽

Trigeminal Nucleus ◽

Peptide Receptor ◽

Related Peptide ◽

Sex differences in the expression of calcitonin gene-related peptide receptor components in the spinal trigeminal nucleus

Neurobiology of Pain ◽

10.1016/j.ynpai.2019.100031 ◽

2019 ◽

Vol 6 ◽

pp. 100031 ◽

Cited By ~ 2

Author(s):

Yadong Ji ◽

Alexandra Rizk ◽

Pamela Voulalas ◽

Hanan Aljohani ◽

Simon Akerman ◽

...

Keyword(s):

Sex Differences ◽

Trigeminal Nucleus ◽

Peptide Receptor ◽

Related Peptide ◽

Pharmacological Properties of MK-3207, a Potent and Orally Active Calcitonin Gene-Related Peptide Receptor Antagonist

Journal of Pharmacology and Experimental Therapeutics ◽

10.1124/jpet.109.163816 ◽

2010 ◽

Vol 333 (1) ◽

pp. 152-160 ◽

Cited By ~ 52

Author(s):

Christopher A. Salvatore ◽

Eric L. Moore ◽

Amy Calamari ◽

Jacquelynn J. Cook ◽

Maria S. Michener ◽

...

Keyword(s):

Receptor Antagonist ◽

Pharmacological Properties ◽

Peptide Receptor ◽

Related Peptide ◽

Calcitonin Gene ◽

Orally Active

Comparison of the Vasoconstrictor Effects of the Calcitonin Gene-related Peptide Receptor Antagonist Telcagepant (MK-0974) and Zolmitriptan in Human Isolated Coronary Arteries

Journal of Cardiovascular Pharmacology ◽

10.1097/fjc.0b013e3181d7665f ◽

2010 ◽

Vol 55 (5) ◽

pp. 518-521 ◽

Cited By ~ 5

Author(s):

Joseph J Lynch ◽

Christopher P Regan ◽

Lars Edvinsson ◽

Richard J Hargreaves ◽

Stefanie A Kane

Keyword(s):

Receptor Antagonist ◽

Coronary Arteries ◽

Peptide Receptor ◽

Related Peptide ◽

An oral calcitonin gene-related peptide receptor antagonist for acute migraine management: Sign of a possible new chapter in headache medicine

Current Neurology and Neuroscience Reports ◽

10.1007/s11910-009-0014-9 ◽

2009 ◽

Vol 9 (2) ◽

pp. 91-93

Author(s):

Ivan Garza

Keyword(s):

Receptor Antagonist ◽

Acute Migraine ◽

Peptide Receptor ◽

Related Peptide ◽

Characterization of the effects of calcitonin gene-related peptide receptor antagonist for Alzheimer's disease

Neuropharmacology ◽

10.1016/j.neuropharm.2020.108017 ◽

2020 ◽

Vol 168 ◽

pp. 108017

Author(s):

Hana Na ◽

Qini Gan ◽

Liam Mcparland ◽

Jack B. Yang ◽

Hongbo Yao ◽

...

Keyword(s):

Alzheimer’S Disease ◽

Alzheimer's Disease ◽

Receptor Antagonist ◽

Peptide Receptor ◽

Related Peptide ◽

Asymmetric Synthesis of the Major Metabolite of a Calcitonin Gene-Related Peptide Receptor Antagonist and Mechanism of Epoxide Hydrogenolysis

The Journal of Organic Chemistry ◽

10.1021/acs.joc.7b00052 ◽

2017 ◽

Vol 82 (7) ◽

pp. 3710-3720 ◽

Cited By ~ 1

Author(s):

Guanglin Luo ◽

Ling Chen ◽

Charles M. Conway ◽

Walter Kostich ◽

Benjamin M. Johnson ◽

...

Keyword(s):

Receptor Antagonist ◽

Asymmetric Synthesis ◽

Major Metabolite ◽

Peptide Receptor ◽

Related Peptide ◽

Effect of a calcitonin gene-related peptide-binding L-RNA aptamer on neuronal activity in the rat spinal trigeminal nucleus

The Journal of Headache and Pain ◽

10.1186/s10194-018-0832-8 ◽

2018 ◽

Vol 19 (1) ◽

Cited By ~ 2

Author(s):

Michael J. M. Fischer ◽

Jakob Schmidt ◽

Stanislav Koulchitsky ◽

Sven Klussmann ◽

Axel Vater ◽

...

Keyword(s):

Neuronal Activity ◽

Peptide Binding ◽

Rna Aptamer ◽

Trigeminal Nucleus ◽

Related Peptide ◽

Characterizing the PK/PD relationship for inhibition of capsaicin-induced dermal vasodilatation by MK-3207, an oral calcitonin gene related peptide receptor antagonist

British Journal of Clinical Pharmacology ◽

10.1111/bcp.12547 ◽

2015 ◽

Vol 79 (5) ◽

pp. 831-837 ◽

Cited By ~ 13

Author(s):

Chi-Chung Li ◽

Steve Vermeersch ◽

William S. Denney ◽

William P. Kennedy ◽

John Palcza ◽

...

Keyword(s):

Receptor Antagonist ◽

Peptide Receptor ◽

Related Peptide ◽