scholarly journals TRV130 partial agonism and capacity to induce anti‐nociceptive tolerance revealed through reducing available μ‐opioid receptor number

2021 ◽  
Vol 178 (8) ◽  
pp. 1855-1868
Author(s):  
Samuel Singleton ◽  
Daniel T. Baptista‐Hon ◽  
Emily Edelsten ◽  
Kirsty S. McCaughey ◽  
Ewan Camplisson ◽  
...  
Keyword(s):  
Opioid Receptor ◽  
Partial Agonism ◽  
Μ Opioid Receptor ◽  
Receptor Number

FUNCTIONAL INTERACTIONS OF PERTUSSIS TOXIN-SENSITIVE G-PROTEINS WITH THE TRANSFECTED μ-OPIOID RECEPTOR IN RAT 1 FIBROBLASTS

Analgesia ◽  
1995 ◽  
Vol 1 (4) ◽  
pp. 438-441
Author(s):  
Zafiroula Georgoussi ◽  
Ian Mullaney ◽  
Alan Wise ◽  
Craig Carr ◽  
Graeme Milligan
Keyword(s):  
G Proteins ◽  
Opioid Receptor ◽  
Pertussis Toxin ◽  
Functional Interactions ◽  
Μ Opioid Receptor

scholarly journals A Promising Chemical Series of Positive Allosteric Modulators of the μ-Opioid Receptor that Enhance the Antinociceptive Efficacy of Opioids but not their Adverse Effects

2021 ◽  
pp. 108673
Author(s):  
Kerri D. Pryce ◽  
Hye Jin Kang ◽  
Farhana Sakloth ◽  
Yongfeng Liu ◽  
Susan Khan ◽  
...  
Keyword(s):  
Adverse Effects ◽  
Opioid Receptor ◽  
Allosteric Modulators ◽  
Μ Opioid Receptor ◽  
Positive Allosteric Modulators

Modulation of μ-opioid receptor desensitization in peripheral sensory neurons by phosphoinositide 3-kinase γ

Neuroscience ◽  
2010 ◽  
Vol 169 (1) ◽  
pp. 449-454 ◽  
Author(s):  
C. König ◽  
O. Gavrilova-Ruch ◽  
G. Segond von Banchet ◽  
R. Bauer ◽  
M. Grün ◽  
...  
Keyword(s):  
Opioid Receptor ◽  
Sensory Neurons ◽  
Receptor Desensitization ◽  
Peripheral Sensory Neurons ◽  
Μ Opioid Receptor ◽  
Phosphoinositide 3 Kinase ◽  
Peripheral Sensory

Alleviating waiting impulsivity and perseverative responding by μ-opioid receptor antagonism in two inbred mouse strains

2014 ◽  
Vol 232 (8) ◽  
pp. 1483-1492 ◽  
Author(s):  
Sandra Sanchez-Roige ◽  
Tamzin L. Ripley ◽  
David N. Stephens
Keyword(s):  
Opioid Receptor ◽  
Inbred Mouse ◽  
Mouse Strains ◽  
Inbred Mouse Strains ◽  
Receptor Antagonism ◽  
Μ Opioid Receptor

Blockade of lipopolysaccharide-induced fever by a μ-opioid receptor-selective antagonist in rats

2000 ◽  
Vol 401 (2) ◽  
pp. 161-165 ◽  
Author(s):  
Khalid Benamar ◽  
Li Xin ◽  
Ellen B Geller ◽  
Martin W Adler
Keyword(s):  
Opioid Receptor ◽  
Selective Antagonist ◽  
Μ Opioid Receptor

Brain regional μ-opioid receptor function in rat lines selected for differences in alcohol preference

2002 ◽  
Vol 448 (2-3) ◽  
pp. 157-163 ◽  
Author(s):  
Sanna L Soini ◽  
Petri Hyytiä ◽  
Esa R Korpi
Keyword(s):  
Opioid Receptor ◽  
Alcohol Preference ◽  
Receptor Function ◽  
Μ Opioid Receptor

scholarly journals The region in the μ opioid receptor conferring selectivity for sufentanil over the δ receptor is different from that over the κ receptor

FEBS Letters ◽  
1996 ◽  
Vol 384 (2) ◽  
pp. 198-202 ◽  
Author(s):  
Jinmin Zhu ◽  
Ji-Chun Xue ◽  
Ping-Yee Law ◽  
Patricia A. Claude ◽  
Lai-Yi Luo ◽  
...  
Keyword(s):  
Opioid Receptor ◽  
Μ Opioid Receptor ◽  
Κ Receptor
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