Synthesis and In Vitro Evaluation of Novel 2-oxo-1,2-dihydroquinoline CB2 Receptor Inverse Agonists

2006 ◽  
Vol 68 (6) ◽  
pp. 334-340 ◽  
Author(s):  
Katri H. Raitio ◽  
Juha R. Savinainen ◽  
Tapio Nevalainen ◽  
Tomi Järvinen ◽  
Jouko Vepsäläinen
Keyword(s):  
Cb2 Receptor ◽  
In Vitro Evaluation ◽  
Inverse Agonists

Synthesis and in vitro evaluation of fluorine-18 benzimidazole sulfones as CB2 PET-radioligands

2019 ◽  
Vol 17 (20) ◽  
pp. 5086-5098 ◽  
Author(s):  
Annukka Kallinen ◽  
Rochelle Boyd ◽  
Samuel Lane ◽  
Rajiv Bhalla ◽  
Karine Mardon ◽  
...  
Keyword(s):  
Binding Affinity ◽  
Cb2 Receptor ◽  
In Vitro Evaluation

New 18F-fluorinated benzimidazole 5-sulfones with low nanomolar binding affinity were synthesised as PET-radioligand candidates for the CB2 receptor.

In vitro and in vivo pharmacological characterization of two novel selective cannabinoid CB2 receptor inverse agonists

2010 ◽  
Vol 61 (4) ◽  
pp. 349-354 ◽  
Author(s):  
Maria Grazia Cascio ◽  
Daniele Bolognini ◽  
Roger G. Pertwee ◽  
Enza Palazzo ◽  
Federico Corelli ◽  
...  
Keyword(s):  
Cb2 Receptor ◽  
Pharmacological Characterization ◽  
Inverse Agonists

In vitro evaluation of IL-18 effects in Crohn's disease

2001 ◽  
Vol 120 (5) ◽  
pp. A316-A317
Author(s):  
P MAERTEN ◽  
S COLPAERT ◽  
Z LIU ◽  
K GEBOES ◽  
J CEUPPENS ◽  
...  
Keyword(s):  
Crohn’S Disease ◽  
Crohn's Disease ◽  
In Vitro Evaluation

52: In Vitro Evaluation of Ureteral Stent Compression

2006 ◽  
Vol 175 (4S) ◽  
pp. 18-18
Author(s):  
Kari Hendlin ◽  
Krishna Vedula ◽  
Christina Horn ◽  
Manoj Monga
Keyword(s):  
Ureteral Stent ◽  
In Vitro Evaluation

Purification hemisynthesis of xanthatin derivates and in vitro evaluation of their activity towards farnesyltransferase (PFTase)

Planta Medica ◽  
2008 ◽  
Vol 74 (09) ◽  
Author(s):  
B Pinel ◽  
A Landreau ◽  
J Dubois ◽  
G Au do ◽  
F De la Poype ◽  
...  
Keyword(s):  
In Vitro Evaluation

In vitro evaluation of the effect of selected herbal extracts on drug transport across porcine jejunal tissue

Planta Medica ◽  
2010 ◽  
Vol 76 (12) ◽  
Author(s):  
C Tarirai ◽  
A Viljoen ◽  
P Chinyemba ◽  
A Khatib ◽  
P Jiyane ◽  
...  
Keyword(s):  
Drug Transport ◽  
Herbal Extracts ◽  
In Vitro Evaluation

In vitro evaluation of the synergetic interaction between antibiotics tetracyclin and penicillin with (+)-usnic acid isolated from Usnea steineri against multiresistant bacteria

Planta Medica ◽  
2014 ◽  
Vol 80 (16) ◽  
Author(s):  
M Gomide Tozatti ◽  
D da Silva Ferreira ◽  
G Morette Mazza ◽  
T da Silva Moraes ◽  
CH Gomes Martins ◽  
...  
Keyword(s):  
Usnic Acid ◽  
In Vitro Evaluation ◽  
Multiresistant Bacteria
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