Constitutively Active Mutants of the Histamine H1 Receptor Suggest a Conserved Hydrophobic Asparagine-Cage That Constrains the Activation of Class A G Protein-Coupled Receptors

2007 ◽  
Vol 73 (1) ◽  
pp. 94-103 ◽  
Author(s):  
Remko A. Bakker ◽  
Aldo Jongejan ◽  
Kamonchanok Sansuk ◽  
Uli Hacksell ◽  
Henk Timmerman ◽  
...  
Keyword(s):  
G Protein ◽  
G Protein Coupled Receptors ◽  
H1 Receptor ◽  
Histamine H1 Receptor ◽  
Class A ◽  
Constitutively Active Mutants ◽  
G Protein Coupled ◽  
Constitutively Active

Lessons from constitutively active mutants of G protein-coupled receptors

2002 ◽  
Vol 13 (8) ◽  
pp. 336-343 ◽  
Author(s):  
Charles Parnot ◽  
Stéphanie Miserey-Lenkei ◽  
Sabine Bardin ◽  
Pierre Corvol ◽  
Eric Clauser
Keyword(s):  
G Protein ◽  
G Protein Coupled Receptors ◽  
Constitutively Active Mutants ◽  
G Protein Coupled ◽  
Constitutively Active

scholarly journals Constitutive Activity among Orphan Class-A G Protein Coupled Receptors

PLoS ONE ◽  
2015 ◽  
Vol 10 (9) ◽  
pp. e0138463 ◽  
Author(s):  
Adam L. Martin ◽  
Michael A. Steurer ◽  
Robert S. Aronstam
Keyword(s):  
G Protein ◽  
G Protein Coupled Receptors ◽  
Constitutive Activity ◽  
Class A ◽  
G Protein Coupled

Universality of the Sodium Ion Binding Mechanism in Class A G-Protein-Coupled Receptors

2018 ◽  
Vol 130 (12) ◽  
pp. 3102-3107 ◽  
Author(s):  
Balaji Selvam ◽  
Zahra Shamsi ◽  
Diwakar Shukla
Keyword(s):  
G Protein ◽  
G Protein Coupled Receptors ◽  
Sodium Ion ◽  
Ion Binding ◽  
Binding Mechanism ◽  
Class A ◽  
G Protein Coupled

scholarly journals G protein-coupled receptors of class A harness the energy of membrane potential to increase their sensitivity and selectivity

2019 ◽  
Vol 1861 (12) ◽  
pp. 183051 ◽  
Author(s):  
Daria N. Shalaeva ◽  
Dmitry A. Cherepanov ◽  
Michael Y. Galperin ◽  
Gert Vriend ◽  
Armen Y. Mulkidjanian
Keyword(s):  
Membrane Potential ◽  
G Protein ◽  
G Protein Coupled Receptors ◽  
Class A ◽  
Sensitivity And Selectivity ◽  
G Protein Coupled

Constitutively Active Mutations of G Protein-Coupled Receptors

1999 ◽  
Vol 30 (6) ◽  
pp. 501-509 ◽  
Author(s):  
Verena Nordhoff ◽  
Jörg Gromoll ◽  
Manuela Simoni
Keyword(s):  
G Protein ◽  
G Protein Coupled Receptors ◽  
G Protein Coupled ◽  
Constitutively Active
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