Synthesis and preliminary biological evaluation of a cyclic somatostatin analog with high affinity to sst1–5

2005 ◽  
Author(s):  
Christos Petrou ◽  
Anastasia Nikolopoulou ◽  
Vassiliki Magafa ◽  
Berthold Nock ◽  
Theodosia Maina ◽  
...  
Keyword(s):  
Biological Evaluation ◽  
Somatostatin Analog ◽  
High Affinity

Synthesis and preliminary biological evaluation of [3H]-MRE 3008-F20: the first high affinity radioligand antagonist for the human A3 adenosine receptors

2000 ◽  
Vol 10 (3) ◽  
pp. 209-211 ◽  
Author(s):  
Pier Giovanni Baraldi ◽  
Barbara Cacciari ◽  
Romeo Romagnoli ◽  
Katia Varani ◽  
Stefania Merighi ◽  
...  
Keyword(s):  
Adenosine Receptors ◽  
Biological Evaluation ◽  
High Affinity

Synthesis of novel multivalent fluorescent inhibitors with high affinity to prostate cancer and their biological evaluation

2018 ◽  
Vol 28 (4) ◽  
pp. 572-576 ◽  
Author(s):  
Young-Do Kwon ◽  
Hea-Jong Chung ◽  
Sun Joo Lee ◽  
Sun-Hwa Lee ◽  
Byung-Hoon Jeong ◽  
...  
Keyword(s):  
Prostate Cancer ◽  
Biological Evaluation ◽  
High Affinity

scholarly journals Synthesis and pre-clinical evaluation of a [18F]fluoromethyl-tanaproget derivative for imaging of progesterone receptor expression

RSC Advances ◽  
2016 ◽  
Vol 6 (62) ◽  
pp. 57569-57579 ◽  
Author(s):  
Shairoz Merchant ◽  
Louis Allott ◽  
Laurence Carroll ◽  
Vickram Tittrea ◽  
Steven Kealey ◽  
...  
Keyword(s):  
Progesterone Receptor ◽  
Clinical Evaluation ◽  
Biological Evaluation ◽  
Receptor Expression ◽  
Progesterone Receptor Expression ◽  
High Affinity ◽  
Synthesis And Biological Evaluation

This work features the synthesis and biological evaluation of a novel fluorinated derivative of tanaproget and a carbon-11 labelled analogue, a high affinity non-steroidal PR ligand, as a possible candidate for imaging PR expressionin vivo.

scholarly journals Design and Synthesis of Potent HIV-1 Protease Inhibitors Incorporating Hexahydrofuropyranol-Derived High Affinity P2Ligands: Structure−Activity Studies and Biological Evaluation

2011 ◽  
Vol 54 (2) ◽  
pp. 622-634 ◽  
Author(s):  
Arun K. Ghosh ◽  
Bruno D. Chapsal ◽  
Abigail Baldridge ◽  
Melinda P. Steffey ◽  
D. Eric Walters ◽  
...  
Keyword(s):  
Protease Inhibitors ◽  
Biological Evaluation ◽  
Design And Synthesis ◽  
High Affinity ◽  
Structure Activity ◽  
Hiv 1
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