4-Thiazolidinone coumarin derivatives as two-component NS2B/NS3 DENV flavivirus serine protease inhibitors: synthesis, molecular docking, biological evaluation and structure–activity relationship studies

Biological Evaluation ◽

Activity Relationship ◽

Coumarin Derivatives ◽

Serine Protease Inhibitors ◽

Structure Activity ◽

Two Component

Symmetrical anhydride-type serine protease inhibitors: Structure-activity relationship studies of human chymase inhibitors

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/s0960-894x(99)00012-8 ◽

1999 ◽

Vol 9 (3) ◽

pp. 413-418 ◽

Cited By ~ 19

Author(s):

Kiyoko Iijima ◽

Jun Katada ◽

Yoshio Hayashi

Keyword(s):

Serine Protease ◽

Protease Inhibitors ◽

Activity Relationship ◽

Serine Protease Inhibitors ◽

Structure-Activity Relationship Within the Serine Protease Inhibitors of the Pacifastin Family

Protein and Peptide Letters ◽

10.2174/0929866054395239 ◽

2005 ◽

Vol 12 (5) ◽

pp. 409-414 ◽

Cited By ~ 15

Author(s):

Christine Kellenberger ◽

Alain Roussel

Keyword(s):

Serine Protease ◽

Protease Inhibitors ◽

Activity Relationship ◽

Serine Protease Inhibitors ◽

Molecular docking, structure–activity relationship and biological evaluation of the anticancer drug monastrol as a pteridine reductase inhibitor in a clinical isolate of Leishmania donovani

Journal of Antimicrobial Chemotherapy ◽

10.1093/jac/dkq189 ◽

2010 ◽

Vol 65 (8) ◽

pp. 1742-1748 ◽

Cited By ~ 24

Author(s):

Jaspreet Kaur ◽

Shyam Sundar ◽

Neeloo Singh

Keyword(s):

Molecular Docking ◽

Clinical Isolate ◽

Anticancer Drug ◽

Reductase Inhibitor ◽

Leishmania Donovani ◽

Biological Evaluation ◽

Activity Relationship ◽

Chromanyl-isoxazolidines as Antibacterial agents: Synthesis, Biological Evaluation, Quantitative Structure Activity Relationship, and Molecular Docking Studies

Chemical Biology & Drug Design ◽

10.1111/cbdd.12653 ◽

2015 ◽

Vol 87 (2) ◽

pp. 213-223 ◽

Cited By ~ 17

Author(s):

Gagandeep Singh ◽

Anuradha Sharma ◽

Harpreet Kaur ◽

Mohan Paul S. Ishar

Keyword(s):

Molecular Docking ◽

Antibacterial Agents ◽

Quantitative Structure Activity Relationship ◽

Docking Studies ◽

Biological Evaluation ◽

Activity Relationship ◽

Quantitative Structure ◽

Molecular Docking Studies ◽

Design, synthesis, and biological evaluation of novel dipeptide-type SARS-CoV 3CL protease inhibitors: Structure–activity relationship study

European Journal of Medicinal Chemistry ◽

10.1016/j.ejmech.2013.05.005 ◽

2013 ◽

Vol 65 ◽

pp. 436-447 ◽

Cited By ~ 19

Author(s):

Pillaiyar Thanigaimalai ◽

Sho Konno ◽

Takehito Yamamoto ◽

Yuji Koiwai ◽

Akihiro Taguchi ◽

...

Keyword(s):

Protease Inhibitors ◽

Synthesis And Biological Evaluation

Biological Evaluation ◽

Activity Relationship ◽

Design Synthesis ◽

Structure Activity ◽

Relationship Study ◽

3Cl Protease ◽

Synthesis, biological evaluation, molecular docking and structure-activity relationship studies of halogenated quinone and naphthoquinone derivatives

Journal of Molecular Structure ◽

10.1016/j.molstruc.2019.06.002 ◽

2019 ◽

Vol 1195 ◽

pp. 462-469 ◽

Cited By ~ 4

Author(s):

Ghulam Abbas ◽

Zahid Hassan ◽

Ahmed Al-Harrasi ◽

Ajmal khan ◽

Ahmed Al-Adawi ◽

...

Keyword(s):

Molecular Docking ◽

Biological Evaluation ◽

Activity Relationship ◽

Discovery of indolin-2-one derivatives as potent PAK4 inhibitors: Structure-activity relationship analysis, biological evaluation and molecular docking study

Bioorganic & Medicinal Chemistry ◽

10.1016/j.bmc.2017.04.047 ◽

2017 ◽

Vol 25 (13) ◽

pp. 3500-3511 ◽

Cited By ~ 12

Author(s):

Jing Guo ◽

Mingyue Zhu ◽

Tianxiao Wu ◽

Chenzhou Hao ◽

Kai Wang ◽

...

Keyword(s):

Molecular Docking ◽

Docking Study ◽

Biological Evaluation ◽

Activity Relationship ◽

Molecular Docking Study ◽

Relationship Analysis ◽

Enhancing monoamine oxidase B inhibitory activity via chiral fluorination: Structure-activity relationship, biological evaluation, and molecular docking study

European Journal of Medicinal Chemistry ◽

10.1016/j.ejmech.2021.114025 ◽

2021 ◽

pp. 114025

Author(s):

Zhizheng Wang ◽

Chao Yi ◽

Kangzhi Chen ◽

Tao Wang ◽

Kang Deng ◽

...

Keyword(s):

Molecular Docking ◽

Monoamine Oxidase ◽

Inhibitory Activity ◽

Docking Study ◽

Biological Evaluation ◽

Activity Relationship ◽

Monoamine Oxidase B ◽

Molecular Docking Study ◽

In vitro α-Glucosidase Inhibition by Non-sugar based Triazoles of Dibenzoazepine, their Structure-Activity Relationship, and Molecular Docking

Medicinal Chemistry ◽

10.2174/1573406413666170726142949 ◽

2017 ◽

Vol 13 (7) ◽

Author(s):

Maria A. Khan ◽

Kulsoom Javaid ◽

Abdul Wadood ◽

Alam Jamal ◽

Farhana Batool ◽

...

Keyword(s):

Molecular Docking ◽

Activity Relationship ◽

Structure Activity Relationship of Arylidene Pyrrolo and Pyrido [2,1-b] Quinazolones as Cytotoxic Agents: Synthesis, SAR Studies, Biological Evaluation and Docking Studies

Medicinal Chemistry ◽

10.2174/1573406411309050003 ◽

2013 ◽

Vol 9 (5) ◽

pp. 642-650 ◽

Cited By ~ 3

Author(s):

Veenu Mangla ◽

Kunal Nepali ◽

Gagandip Singh ◽

Jagjeet Singh ◽

Santosh Guru ◽

...

Keyword(s):

Docking Studies ◽

Biological Evaluation ◽

Cytotoxic Agents ◽

Activity Relationship ◽

Sar Studies ◽

Structure Activity ◽

Relationship Of