scholarly journals Studies on Analgesic Oligopeptides. VII. Solid Phase Synthesis and Biological Properties of Tyr-D-Arg-Phe-.BETA.Ala-NH2 and its Fluorinated Aromatic Amino Acid Derivatives.

1991 ◽  
Vol 39 (9) ◽  
pp. 2316-2318 ◽  
Author(s):  
Yusuke SASAKI ◽  
Akihiro AMBO ◽  
Kenji SUZUKI
Keyword(s):  
Amino Acid ◽  
Aromatic Amino Acid ◽  
Solid Phase Synthesis ◽  
Solid Phase ◽  
Biological Properties ◽  
Amino Acid Derivatives ◽  
Phase Synthesis

Synthesis and biological properties of vasopressin analogues containing 1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid

1990 ◽  
Vol 55 (4) ◽  
pp. 1099-1105 ◽  
Author(s):  
Zdenko Procházka ◽  
Juris E. Ancans ◽  
Jiřina Slaninová ◽  
Alena Machová ◽  
Tomislav Barth ◽  
...  
Keyword(s):  
Amino Acid ◽  
Carboxylic Acid ◽  
Solid Phase Synthesis ◽  
Solid Phase ◽  
Biological Activities ◽  
Biological Properties ◽  
Phase Synthesis ◽  
Aromatic Residues ◽  
Synthesis Methodology ◽  
Vasopressin Analogues

Solid phase synthesis methodology on a benzhydrylamine resin was used for the synthesis of three analogues of vasopressin with the non-coded amino acid, 1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid (Tic), in the position 2 ([Tic2, Lys8]VP (I)) and in the position 3 ([Tic3, Lys8]VP (II)). The analogue containing only one Tic in place of both aromatic residues was also isolated (des-Tyr2-[Tic3, Lys8]VP (III)). The biological activities of all analogues were negligible.

Asymmetric Solid-Phase Synthesis of (R)-α-Amino Acid Derivatives

Synfacts ◽  
2007 ◽  
Vol 2007 (7) ◽  
pp. 0777-0777
Author(s):  
H.-G. Park ◽  
B.-S. Jeong ◽  
M.-J. Kim ◽  
S.-S. Jew
Keyword(s):  
Amino Acid ◽  
Solid Phase Synthesis ◽  
Solid Phase ◽  
Amino Acid Derivatives ◽  
Phase Synthesis

Enantioselective solid-phase synthesis of α-amino acid derivatives

Tetrahedron ◽  
1999 ◽  
Vol 55 (20) ◽  
pp. 6347-6362 ◽  
Author(s):  
Martin J. O'Donnell ◽  
Francisca Delgado ◽  
Richard S. Pottorf
Keyword(s):  
Amino Acid ◽  
Solid Phase Synthesis ◽  
Solid Phase ◽  
Amino Acid Derivatives ◽  
Phase Synthesis
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