A Combined Quantitative Structure-Activity Relationship Research of Quinolinone Derivatives as Androgen Receptor Antagonists

Combinatorial Chemistry & High Throughput Screening ◽

10.2174/1386207318666150831125750 ◽

2015 ◽

Vol 18 (9) ◽

pp. 834-845 ◽

Author(s):

Yuwei Wang ◽

Fang Bai ◽

Hong Cao ◽

Jiazhong Li ◽

Huanxiang Liu ◽

...

Keyword(s):

Androgen Receptor ◽

Quantitative Structure Activity Relationship ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Quantitative Structure ◽

Receptor Antagonists ◽

Structure Activity ◽

Androgen Receptor Antagonists

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Quantitative Structure—Activity Relationship (QSAR) Studies on Sulfide Analogues as Potent M2 Muscarinic Receptor Antagonists.

10.1002/chin.200622145 ◽

2006 ◽

Vol 37 (22) ◽

Author(s):

A. K. Srivastava ◽

A. A. Khan ◽

Abha Tripathi ◽

Archana Archana

Keyword(s):

Muscarinic Receptor ◽

Quantitative Structure Activity Relationship ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Quantitative Structure ◽

Receptor Antagonists ◽

Qsar Studies ◽

Structure Activity ◽

Muscarinic Receptor Antagonists ◽

M2 Muscarinic Receptor

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Structure–activity relationship analysis of carbobicyclo and oxabicyclo succinimide analogs as potential androgen receptor antagonists

Journal of Biomolecular Structure and Dynamics ◽

10.1080/07391102.2017.1371643 ◽

2017 ◽

Vol 36 (11) ◽

pp. 2876-2892 ◽

Author(s):

Lingyan Wang ◽

Jiazhong Li

Keyword(s):

Androgen Receptor ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Receptor Antagonists ◽

Relationship Analysis ◽

Structure Activity ◽

Androgen Receptor Antagonists

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Quantitative structure activity relationship (QSAR) studies on a series of imidazole derivatives as novel ORL1 receptor antagonists

Journal of Saudi Chemical Society ◽

10.1016/j.jscs.2011.04.014 ◽

2013 ◽

Vol 17 (3) ◽

pp. 321-328 ◽

Author(s):

A.K. Srivastava ◽

Neerja Shukla

Keyword(s):

Quantitative Structure Activity Relationship ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Quantitative Structure ◽

Receptor Antagonists ◽

Qsar Studies ◽

Imidazole Derivatives ◽

Orl1 Receptor ◽

Structure Activity

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Relevance of theoretical molecular descriptors in quantitative structure–activity relationship analysis of α1-adrenergic receptor antagonists

Bioorganic & Medicinal Chemistry ◽

10.1016/s0968-0896(99)00194-7 ◽

1999 ◽

Vol 7 (11) ◽

pp. 2437-2451 ◽

Author(s):

M.C. Menziani ◽

M. Montorsi ◽

P.G. De Benedetti ◽

M. Karelson

Keyword(s):

Adrenergic Receptor ◽

Molecular Descriptors ◽

Quantitative Structure Activity Relationship ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Quantitative Structure ◽

Receptor Antagonists ◽

Relationship Analysis ◽

Structure Activity

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Quantitative structure activity relationship analysis of angiotensin II AT1 receptor antagonists

Medicinal Chemistry Research ◽

10.1007/s00044-009-9205-9 ◽

2009 ◽

Vol 19 (5) ◽

pp. 475-489 ◽

Author(s):

Sarvesh Kumar Paliwal ◽

Mahima Pal ◽

Anees A. Siddiqui

Keyword(s):

Angiotensin Ii ◽

Quantitative Structure Activity Relationship ◽

Structure Activity Relationship ◽

At1 Receptor ◽

Activity Relationship ◽

Quantitative Structure ◽

Receptor Antagonists ◽

Relationship Analysis ◽

Structure Activity ◽

At1 Receptor Antagonists

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Quantitative structure–Activity relationship studies on 5-phenyl-3-ureido-1,5-benzodiazepine as cholecystokinin-A receptor antagonists

Bioorganic & Medicinal Chemistry ◽

10.1016/s0968-0896(02)00167-0 ◽

2002 ◽

Vol 10 (11) ◽

pp. 3571-3581 ◽

Author(s):

Vijay K. Agrawal ◽

Ruchi Sharma ◽

Padmakar V. Khadikar

Keyword(s):

Quantitative Structure Activity Relationship ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Quantitative Structure ◽

Receptor Antagonists ◽

Structure Activity

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Synthesis and Three-Dimensional Quantitative Structure-Activity Relationship Analysis of H3 Receptor Antagonists Containing a Neutral Heterocyclic Polar Group

Drug Design and Discovery ◽

10.3109/10559610290249539 ◽

2003 ◽

Vol 18 (2-3) ◽

pp. 65-79 ◽

Author(s):

Silvia Rivara ◽

Marco Mor ◽

Fabrizio Bordi ◽

Claudia Silva ◽

Valentina Zuliani ◽

...

Keyword(s):

Three Dimensional ◽

Quantitative Structure Activity Relationship ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Polar Group ◽

Quantitative Structure ◽

Receptor Antagonists ◽

Relationship Analysis ◽

Structure Activity ◽

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Quantitative structure activity relationship of benzoxazinone derivatives as neuropeptide Y Y5 receptor antagonists

European Journal of Medicinal Chemistry ◽

10.1016/j.ejmech.2006.01.012 ◽

2006 ◽

Vol 41 (4) ◽

pp. 552-557 ◽

Author(s):

S. Deswal ◽

N. Roy

Keyword(s):

Neuropeptide Y ◽

Quantitative Structure Activity Relationship ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Quantitative Structure ◽

Receptor Antagonists ◽

Structure Activity ◽

Relationship Of

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Structure-activity relationship analysis of 3-phenylpyrazole derivatives as androgen receptor antagonists

Journal of Biomolecular Structure and Dynamics ◽

10.1080/07391102.2019.1635913 ◽

2019 ◽

Vol 38 (9) ◽

pp. 2582-2591 ◽

Author(s):

Wenya Han ◽

Jiazhong Li

Keyword(s):

Androgen Receptor ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Receptor Antagonists ◽

Relationship Analysis ◽

Structure Activity ◽

Androgen Receptor Antagonists

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Screening of 397 Chemicals and Development of a Quantitative Structure−Activity Relationship Model for Androgen Receptor Antagonism

Chemical Research in Toxicology ◽

10.1021/tx7002382 ◽

2008 ◽

Vol 21 (4) ◽

pp. 813-823 ◽

Author(s):

Anne Marie Vinggaard ◽

Jay Niemelä ◽

Eva Bay Wedebye ◽

Gunde Egeskov Jensen

Keyword(s):

Androgen Receptor ◽

Quantitative Structure Activity Relationship ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Quantitative Structure ◽

Receptor Antagonism ◽

Structure Activity ◽

Relationship Model

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