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Advances in the Discovery of Novel Positive Allosteric Modulators of the α7 Nicotinic Acetylcholine Receptor
Recent Patents on CNS Drug Discovery
◽
10.2174/157488907780832751
◽
2007
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Vol 2
(2)
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Cited By ~ 27
Author(s):
Ramin Faghih
◽
Gregory A. Gfesser
◽
Murali Gopalakrishnan
Keyword(s):
Acetylcholine Receptor
◽
Nicotinic Acetylcholine Receptor
◽
Allosteric Modulators
◽
Α7 Nicotinic Acetylcholine Receptor
◽
Nicotinic Acetylcholine
◽
Positive Allosteric Modulators
Download Full-text
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Discovery of novel positive allosteric modulators of the α7 nicotinic acetylcholine receptor: Scaffold hopping approach
European Journal of Medicinal Chemistry
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10.1016/j.ejmech.2021.113189
◽
2021
◽
Vol 214
◽
pp. 113189
Author(s):
István Ledneczki
◽
Pál Tapolcsányi
◽
Eszter Gábor
◽
András Visegrády
◽
Márton Vass
◽
...
Keyword(s):
Acetylcholine Receptor
◽
Nicotinic Acetylcholine Receptor
◽
Allosteric Modulators
◽
Scaffold Hopping
◽
Α7 Nicotinic Acetylcholine Receptor
◽
Nicotinic Acetylcholine
◽
Positive Allosteric Modulators
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3 α7 Nicotinic Acetylcholine Receptor Agonists and Positive Allosteric Modulators
Progress in Medicinal Chemistry - Progress in Medicinal Chemistry Volume 46
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10.1016/s0079-6468(07)00003-3
◽
2008
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pp. 131-171
◽
Cited By ~ 31
Author(s):
Andrew P. Lightfoot
◽
James N.C. Kew
◽
John Skidmore
Keyword(s):
Acetylcholine Receptor
◽
Nicotinic Acetylcholine Receptor
◽
Allosteric Modulators
◽
Α7 Nicotinic Acetylcholine Receptor
◽
Nicotinic Acetylcholine
◽
Receptor Agonists
◽
Positive Allosteric Modulators
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Characterization of the effects of novel positive allosteric modulators on the functionality of the α7 nicotinic acetylcholine receptor (nAChR)
The FASEB Journal
◽
10.1096/fasebj.2018.32.1_supplement.533.80
◽
2018
◽
Vol 32
(S1)
◽
Author(s):
Francis Reilly‐Andujar
◽
José A. Lasalde
◽
José O. Colón
Keyword(s):
Acetylcholine Receptor
◽
Nicotinic Acetylcholine Receptor
◽
Allosteric Modulators
◽
Α7 Nicotinic Acetylcholine Receptor
◽
Nicotinic Acetylcholine
◽
Positive Allosteric Modulators
Download Full-text
Positive allosteric modulators of the α7 nicotinic acetylcholine receptor potentiate glutamate release in the prefrontal cortex of freely-moving rats
Neuropharmacology
◽
10.1016/j.neuropharm.2016.08.033
◽
2016
◽
Vol 111
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pp. 78-91
◽
Cited By ~ 3
Author(s):
D.M. Bortz
◽
B.A. Upton
◽
J.D. Mikkelsen
◽
J.P. Bruno
Keyword(s):
Prefrontal Cortex
◽
Acetylcholine Receptor
◽
Nicotinic Acetylcholine Receptor
◽
Glutamate Release
◽
Allosteric Modulators
◽
Α7 Nicotinic Acetylcholine Receptor
◽
Nicotinic Acetylcholine
◽
Freely Moving Rats
◽
Freely Moving
◽
Positive Allosteric Modulators
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HTS-based discovery and optimization of novel positive allosteric modulators of the α7 nicotinic acetylcholine receptor
European Journal of Medicinal Chemistry
◽
10.1016/j.ejmech.2021.113560
◽
2021
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pp. 113560
Author(s):
István Ledneczki
◽
Anita Horváth
◽
Pál Tapolcsányi
◽
János Éles
◽
Katalin Dudás Molnár
◽
...
Keyword(s):
Acetylcholine Receptor
◽
Nicotinic Acetylcholine Receptor
◽
Allosteric Modulators
◽
Α7 Nicotinic Acetylcholine Receptor
◽
Nicotinic Acetylcholine
◽
Positive Allosteric Modulators
Download Full-text
Repeated administration of α7 nicotinic acetylcholine receptor (nAChR) agonists, but not positive allosteric modulators, increases α7 nAChR levels in the brain
Journal of Neurochemistry
◽
10.1111/j.1471-4159.2010.06845.x
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2010
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pp. no-no
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Cited By ~ 1
Author(s):
Ditte Z. Christensen
◽
Jens D. Mikkelsen
◽
Henrik H. Hansen
◽
Morten S. Thomsen
Keyword(s):
Acetylcholine Receptor
◽
Nicotinic Acetylcholine Receptor
◽
Repeated Administration
◽
Allosteric Modulators
◽
Α7 Nicotinic Acetylcholine Receptor
◽
Nicotinic Acetylcholine
◽
Α7 Nachr
◽
Positive Allosteric Modulators
◽
The Brain
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Novel Positive Allosteric Modulators of the Human α7 Nicotinic Acetylcholine Receptor
Biochemistry
◽
10.1021/bi102001m
◽
2011
◽
Vol 50
(23)
◽
pp. 5263-5278
◽
Cited By ~ 37
Author(s):
Hugo R. Arias
◽
Ruo-Xu Gu
◽
Dominik Feuerbach
◽
Bao-Bao Guo
◽
Yong Ye
◽
...
Keyword(s):
Acetylcholine Receptor
◽
Nicotinic Acetylcholine Receptor
◽
Allosteric Modulators
◽
Α7 Nicotinic Acetylcholine Receptor
◽
Nicotinic Acetylcholine
◽
Positive Allosteric Modulators
Download Full-text
Antinociceptive effects of α7 nicotinic acetylcholine receptor positive allosteric modulators type I and II in models of acute and chronic pain in mice
The FASEB Journal
◽
10.1096/fasebj.27.1_supplement.886.14
◽
2013
◽
Vol 27
(S1)
◽
Author(s):
Kelen Freitas
◽
S Stevens Negus
◽
F Ivy Carroll
◽
M Imad Damaj
Keyword(s):
Chronic Pain
◽
Acetylcholine Receptor
◽
Nicotinic Acetylcholine Receptor
◽
Type I
◽
Allosteric Modulators
◽
Α7 Nicotinic Acetylcholine Receptor
◽
Nicotinic Acetylcholine
◽
Antinociceptive Effects
◽
Positive Allosteric Modulators
Download Full-text
Evaluation of α7 Nicotinic Acetylcholine Receptor Agonists and Positive Allosteric Modulators Using the Parallel Oocyte Electrophysiology Test Station
Assay and Drug Development Technologies
◽
10.1089/adt.2009.0194
◽
2009
◽
Vol 7
(4)
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pp. 374-390
◽
Cited By ~ 21
Author(s):
John Malysz
◽
Jens H. Grønlien
◽
Daniel B. Timmermann
◽
Monika Håkerud
◽
Kirsten Thorin-Hagene
◽
...
Keyword(s):
Acetylcholine Receptor
◽
Nicotinic Acetylcholine Receptor
◽
Allosteric Modulators
◽
Α7 Nicotinic Acetylcholine Receptor
◽
Nicotinic Acetylcholine
◽
Receptor Agonists
◽
Positive Allosteric Modulators
◽
Electrophysiology Test
Download Full-text
Diversity of Nicotinic Acetylcholine Receptor Positive Allosteric Modulators Revealed by Mutagenesis and a Revised Structural Model
Molecular Pharmacology
◽
10.1124/mol.117.110551
◽
2017
◽
Vol 93
(2)
◽
pp. 128-140
◽
Cited By ~ 23
Author(s):
Joseph Newcombe
◽
Anna Chatzidaki
◽
Tom D. Sheppard
◽
Maya Topf
◽
Neil S. Millar
Keyword(s):
Acetylcholine Receptor
◽
Nicotinic Acetylcholine Receptor
◽
Structural Model
◽
Allosteric Modulators
◽
Nicotinic Acetylcholine
◽
Positive Allosteric Modulators
Download Full-text
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