Occupancy of α7 Nicotinic Acetylcholine Receptors in the Brain by Tropisetron: A Positron Emission Tomography Study Using [11C]CHIBA-1001 in Healthy Human Subjects

Acetylcholine Receptors ◽

Human Subjects ◽

Emission Tomography ◽

Healthy Human ◽

Nicotinic Acetylcholine ◽

Positron Emission ◽

Healthy Human Subjects ◽

Synthesis and evaluation of new radioligands [11C]A-833834 and [11C]A-752274 for positron-emission tomography of α7-nicotinic acetylcholine receptors

Nuclear Medicine and Biology ◽

10.1016/j.nucmedbio.2012.11.013 ◽

2013 ◽

Vol 40 (3) ◽

pp. 395-402 ◽

Cited By ~ 13

Author(s):

Andrew G. Horti ◽

Hayden T. Ravert ◽

Yongjun Gao ◽

Daniel P. Holt ◽

William H. Bunnelle ◽

...

Keyword(s):

Α7 Nicotinic Acetylcholine Receptors

Acetylcholine Receptors ◽

Emission Tomography ◽

Nicotinic Acetylcholine ◽

Positron Emission ◽

Derivatives of Dibenzothiophene for Positron Emission Tomography Imaging of α7-Nicotinic Acetylcholine Receptors

Journal of Medicinal Chemistry ◽

10.1021/jm401184f ◽

2013 ◽

Vol 56 (19) ◽

pp. 7574-7589 ◽

Cited By ~ 36

Author(s):

Yongjun Gao ◽

Kenneth J. Kellar ◽

Robert P. Yasuda ◽

Thao Tran ◽

Yingxian Xiao ◽

...

Keyword(s):

Acetylcholine Receptors ◽

Positron Emission Tomography Imaging ◽

Emission Tomography ◽

Nicotinic Acetylcholine ◽

Tomography Imaging ◽

Positron Emission ◽

Derivatives Of

Synthesis and biological evaluation of novel carbon-11 labeled pyridyl ethers: candidate ligands for in vivo imaging of α4β2 nicotinic acetylcholine receptors (α4β2-nAChRs) in the brain with positron emission tomography

Bioorganic & Medicinal Chemistry ◽

10.1016/j.bmc.2009.05.021 ◽

2009 ◽

Vol 17 (13) ◽

pp. 4367-4377 ◽

Cited By ~ 6

Author(s):

Yongjun Gao ◽

Hayden T. Ravert ◽

Hiroto Kuwabara ◽

Yingxian Xiao ◽

Christopher J. Endres ◽

...

Keyword(s):

In Vivo Imaging ◽

Acetylcholine Receptors ◽

Biological Evaluation ◽

Emission Tomography ◽

Nicotinic Acetylcholine ◽

Positron Emission ◽

Synthesis And Biological Evaluation ◽

LC-MS Supported Studies on the in Vitro Metabolism of both Enantiomers of Flubatine and the in Vivo Metabolism of (+)-[18F]Flubatine—A Positron Emission Tomography Radioligand for Imaging α4β2 Nicotinic Acetylcholine Receptors

Molecules ◽

10.3390/molecules21091200 ◽

2016 ◽

Vol 21 (9) ◽

pp. 1200 ◽

Cited By ~ 7

Author(s):

Friedrich-Alexander Ludwig ◽

René Smits ◽

Steffen Fischer ◽

Cornelius Donat ◽

Alexander Hoepping ◽

...

Keyword(s):

Acetylcholine Receptors ◽

In Vitro Metabolism ◽

Emission Tomography ◽

In Vivo Metabolism ◽

Nicotinic Acetylcholine ◽

Positron Emission

Synthesis and Evaluation of a Novel Series of 2-Chloro-5-((1-methyl-2-(S)-pyrrolidinyl)methoxy)-3-(2-(4-pyridinyl)vinyl)pyridine Analogues as Potential Positron Emission Tomography Imaging Agents for Nicotinic Acetylcholine Receptors

Journal of Medicinal Chemistry ◽

10.1021/jm010550n ◽

2002 ◽

Vol 45 (13) ◽

pp. 2841-2849 ◽

Cited By ~ 18

Author(s):

LaVerne L. Brown ◽

Santosh Kulkarni ◽

Olga A. Pavlova ◽

Andrei O. Koren ◽

Alexey G. Mukhin ◽

...

Keyword(s):

Acetylcholine Receptors ◽

Positron Emission Tomography Imaging ◽

Emission Tomography ◽

Imaging Agents ◽

Nicotinic Acetylcholine ◽

Tomography Imaging ◽

Positron Emission ◽

Vinyl Pyridine

Positron emission tomography imaging of D2/3agonist binding in healthy human subjects with the radiotracer [11C]-N-propyl-norapomorphine: Preliminary evaluation and reproducibility studies

Synapse ◽

10.1002/syn.20633 ◽

2009 ◽

Vol 63 (7) ◽

pp. 574-584 ◽

Cited By ~ 18

Author(s):

Rajesh Narendran ◽

W. Gordon Frankle ◽

N. Scott Mason ◽

Charles M. Laymon ◽

Brian J. Lopresti ◽

...

Keyword(s):

Human Subjects ◽

Positron Emission Tomography Imaging ◽

Emission Tomography ◽

Preliminary Evaluation ◽

Healthy Human ◽

Tomography Imaging ◽

Positron Emission ◽

Healthy Human Subjects

Cerebral nicotinic acetylcholine receptors in patients with Alzheimer's disease or vascular dementia - evaluation with 2-[18F]F-A85380 and positron emission tomography (PET)

Journal of Cerebral Blood Flow & Metabolism ◽

10.1038/sj.jcbfm.9591524.0580 ◽

2005 ◽

Vol 25 (1_suppl) ◽

pp. S580-S580

Author(s):

Kai Kendziorra ◽

Philipp Meyer ◽

Henryk Barthel ◽

Georg Becker ◽

Dietlind Sorger ◽

...

Keyword(s):

Alzheimer’S Disease ◽

Alzheimer's Disease ◽

Vascular Dementia ◽

Acetylcholine Receptors ◽

Emission Tomography ◽

Nicotinic Acetylcholine ◽

Positron Emission

A Promising PET Tracer for Imaging of α7 Nicotinic Acetylcholine Receptors in the Brain: Design, Synthesis, and in Vivo Evaluation of a Dibenzothiophene-Based Radioligand

Molecules ◽

10.3390/molecules201018387 ◽

2015 ◽

Vol 20 (10) ◽

pp. 18387-18421 ◽

Cited By ~ 11

Author(s):

Rodrigo Teodoro ◽

Matthias Scheunemann ◽

Winnie Deuther-Conrad ◽

Barbara Wenzel ◽

Francesca Fasoli ◽

...

Keyword(s):

Acetylcholine Receptors ◽

In Vivo Evaluation ◽

Nicotinic Acetylcholine ◽

Design Synthesis ◽

Pet Tracer ◽

Kynurenic acid as an antagonist of α7 nicotinic acetylcholine receptors in the brain: Facts and challenges

Biochemical Pharmacology ◽

10.1016/j.bcp.2012.12.014 ◽

2013 ◽

Vol 85 (8) ◽

pp. 1027-1032 ◽

Cited By ~ 71

Author(s):

Edson X. Albuquerque ◽

Robert Schwarcz

Keyword(s):

Acetylcholine Receptors ◽

Kynurenic Acid ◽

Nicotinic Acetylcholine ◽

Radiosynthesis and evaluation of 5-(2-(4-pyridinyl)vinyl)-6-chloro-3-(1-[11CH3]methyl-2-(S)-pyrrolidinylmethoxy)pyridine and its analogs, high affinity ligands for studying nicotinic acetylcholine receptors by positron emission tomography

Journal of Labelled Compounds and Radiopharmaceuticals ◽

10.1002/jlcr.2580440104 ◽

2001 ◽

Vol 44 (S1) ◽

pp. S9-S11

Author(s):

L. L. Brown ◽

A. G. Mukhin ◽

S. I. Chefer ◽

O. Pavlova ◽

A. O. Koren ◽

...

Keyword(s):

Acetylcholine Receptors ◽

Emission Tomography ◽

Nicotinic Acetylcholine ◽

Affinity Ligands ◽

High Affinity ◽

Positron Emission