ChemInform Abstract: Multicomponent Synthesis of Cyclic Depsipeptide Mimics by Ugi Reaction Including Cyclic Hemiacetals Derived from Asymmetric Organocatalysis.

ChemInform ◽  
2016 ◽  
Vol 47 (25) ◽  
Author(s):  
Alexander F. de la Torre ◽  
Daniel G. Rivera ◽  
Odette Concepcion ◽  
Radell Echemendia ◽  
Arlene G. Correa ◽  
...  
Keyword(s):  
Ugi Reaction ◽  
Multicomponent Synthesis ◽  
Cyclic Depsipeptide ◽  
Asymmetric Organocatalysis

Multicomponent Synthesis of Cyclic Depsipeptide Mimics by Ugi Reaction Including Cyclic Hemiacetals Derived from Asymmetric Organocatalysis

2016 ◽  
Vol 81 (3) ◽  
pp. 803-809 ◽  
Author(s):  
Alexander F. de la Torre ◽  
Daniel G. Rivera ◽  
Odette Concepción ◽  
Radell Echemendia ◽  
Arlene G. Correa ◽  
...  
Keyword(s):  
Ugi Reaction ◽  
Multicomponent Synthesis ◽  
Cyclic Depsipeptide ◽  
Asymmetric Organocatalysis

scholarly journals Ugi reaction-derived prolyl peptide catalysts grafted on the renewable polymer polyfurfuryl alcohol for applications in heterogeneous enamine catalysis

2019 ◽  
Vol 15 ◽  
pp. 1210-1216 ◽  
Author(s):  
Alexander F de la Torre ◽  
Gabriel S Scatena ◽  
Oscar Valdés ◽  
Daniel G Rivera ◽  
Márcio W Paixão
Keyword(s):  
Multicomponent Reactions ◽  
Supported Catalysts ◽  
Ugi Reaction ◽  
Multicomponent Synthesis ◽  
Polyfurfuryl Alcohol ◽  
Peptide Catalysts ◽  
Asymmetric Michael Addition ◽  
Enamine Catalysis ◽  
Work Supports ◽  
Peptide Catalyst

The multicomponent synthesis of prolyl pseudo-peptide catalysts using the Ugi reaction with furfurylamines or isocyanides is described. The incorporation of such a polymerizable furan handle enabled the subsequent polymerization of the peptide catalyst with furfuryl alcohol, thus rendering polyfurfuryl alcohol-supported catalysts for applications in heterogeneous enamine catalysis. The utilization of the polymer-supported catalysts in both batch and continuous-flow organocatalytic procedures proved moderate catalytic efficacy and enantioselectivity, but excellent diastereoselectivity in the asymmetric Michael addition of n-butanal to β-nitrostyrene that was used as a model reaction. This work supports the potential of multicomponent reactions towards the assembly of catalysts and their simultaneous functionalization for immobilization.

Imides: forgotten players in the Ugi reaction. One-pot multicomponent synthesis of quinazolinones

2011 ◽  
Vol 47 (24) ◽  
pp. 6966 ◽  
Author(s):  
Riccardo Mossetti ◽  
Tracey Pirali ◽  
Dèsirèe Saggiorato ◽  
Gian Cesare Tron
Keyword(s):  
Ugi Reaction ◽  
Multicomponent Synthesis ◽  
One Pot

ChemInform Abstract: Imides: Forgotten Players in the Ugi Reaction. One-Pot Multicomponent Synthesis of Quinazolinones.

ChemInform ◽  
2011 ◽  
Vol 42 (43) ◽  
pp. no-no
Author(s):  
Riccardo Mossetti ◽  
Tracey Pirali ◽  
Desiree Saggiorato ◽  
Gian Cesare Tron
Keyword(s):  
Ugi Reaction ◽  
Multicomponent Synthesis ◽  
One Pot

scholarly journals Multicomponent synthesis of artificial nucleases and their RNase and DNase activity

2011 ◽  
Vol 7 ◽  
pp. 1135-1140 ◽  
Author(s):  
Anton V Gulevich ◽  
Lyudmila S Koroleva ◽  
Olga V Morozova ◽  
Valentina N Bakhvalova ◽  
Vladimir N Silnikov ◽  
...  
Keyword(s):  
Amino Acid ◽  
Nuclease Activity ◽  
Ugi Reaction ◽  
Amino Acid Residues ◽  
Multicomponent Synthesis ◽  
Artificial Ribonucleases ◽  
Circular Dna ◽  
Artificial Nucleases ◽  
Target Molecules ◽  
New Compounds

The synthesis of new, artificial ribonucleases containing two amino acid residues connected by an aliphatic linker has been developed. Target molecules were synthesized via a catalytic three-component Ugi reaction from aliphatic diisocyanides. Preliminary investigations proved unspecific nuclease activity of the new compounds towards single-stranded RNA and double-stranded circular DNA.

New Antimycobacterial Leads from Multicomponent Hydrazino-Ugi Reaction

2015 ◽  
Vol 11 (999) ◽  
pp. 1-1
Author(s):  
Ekaterina Lakontseva ◽  
Ruben Karapetian ◽  
Mikhail Krasavin
Keyword(s):  
Ugi Reaction
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