The Discovery and Structure‐Activity Evaluation of (+)‐Floyocidin B and Synthetic Analogs

ChemMedChem ◽

10.1002/cmdc.202100644 ◽

2021 ◽

Author(s):

Yolanda Kleiner ◽

Christoph Pöverlein ◽

Jannike Klädtke ◽

Michael Kurz ◽

Henrik F. König ◽

...

Keyword(s):

Synthetic Analogs ◽

Activity Evaluation ◽

Structure Activity

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Isothiocyanate Synthetic Analogs: Biological Activities, Structure-Activity Relationships and Synthetic Strategies

Mini-Reviews in Medicinal Chemistry ◽

10.2174/1389557514666141106131909 ◽

2014 ◽

Vol 14 (12) ◽

pp. 963-977 ◽

Author(s):

Andrea Milelli ◽

Carmela Fimognari ◽

Nicole Ticchi ◽

Paolo Neviani ◽

Anna Minarini ◽

...

Keyword(s):

Biological Activities ◽

Synthetic Analogs ◽

Structure Activity Relationships ◽

Structure Activity

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ChemInform Abstract: DRUGS DERIVED FROM CANNABINOIDS. 7. TACHYCARDIA AND ANALGESIA STRUCTURE-ACTIVITY RELATIONSHIPS IN Δ9-TETRAHYDROCANNABINOL AND SOME SYNTHETIC ANALOGS

Chemischer Informationsdienst ◽

10.1002/chin.197851203 ◽

1978 ◽

Vol 9 (51) ◽

Author(s):

P. F. OSGOOD ◽

J. F. HOWES ◽

R. K. RAZDAM ◽

H. G. PARS

Keyword(s):

Synthetic Analogs ◽

Structure Activity Relationships ◽

Structure Activity

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Potent, Orally Active Heterocycle-Based Combretastatin A-4 Analogues: Synthesis, Structure−Activity Relationship, Pharmacokinetics, and In Vivo Antitumor Activity Evaluation

Journal of Medicinal Chemistry ◽

10.1021/jm010523x ◽

2002 ◽

Vol 45 (8) ◽

pp. 1697-1711 ◽

Author(s):

Le Wang ◽

Keith W. Woods ◽

Qun Li ◽

Kenneth J. Barr ◽

Richard W. McCroskey ◽

...

Keyword(s):

Antitumor Activity ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Activity Evaluation ◽

Structure Activity ◽

In Vivo Antitumor Activity ◽

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Structure-Activity Relationships of Synthetic Analogs of Jasmonic Acid and Coronatine on Induction of Benzophenanthridine Alkaloid Accumulation in Eschscholzia californica Cell Cultures

Biological Chemistry ◽

10.1515/bc.2000.094 ◽

2000 ◽

Vol 381 (8) ◽

Author(s):

G. Haider ◽

T. von Schrader ◽

M. Füßlein ◽

S. Blechert ◽

T.M. Kutchan

Keyword(s):

Jasmonic Acid ◽

Cell Cultures ◽

Synthetic Analogs ◽

Eschscholzia Californica ◽

Structure Activity Relationships ◽

Structure Activity ◽

Benzophenanthridine Alkaloid

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ChemInform Abstract: STRUCTURE-ACTIVITY RELATIONSHIP IN CINNAMAMIDES. 3. SYNTHESIS AND ANTICONVULSANT ACTIVITY EVALUATION OF SOME DERIVATIVES OF (E)- AND (Z)-M-(TRIFLUOROMETHYL)CINNAMAMIDE

Chemischer Informationsdienst ◽

10.1002/chin.198143145 ◽

1981 ◽

Vol 12 (43) ◽

Author(s):

A. BALSAMO ◽

P. CROTTI ◽

A. LAPUCCI ◽

B. MACCHIA ◽

F. MACCHIA ◽

...

Keyword(s):

Anticonvulsant Activity ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Activity Evaluation ◽

Structure Activity ◽

Abstract Structure ◽

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Screening of antimicrobial activity of diarylamines in the 2,3,5-trimethylbenzo[b]thiophene series: a structure–activity evaluation study

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/j.bmcl.2004.09.038 ◽

2004 ◽

Vol 14 (23) ◽

pp. 5831-5833 ◽

Author(s):

Isabel C.F.R. Ferreira ◽

Ricardo C. Calhelha ◽

Letícia M. Estevinho ◽

Maria-João R.P. Queiroz

Keyword(s):

Antimicrobial Activity ◽

Evaluation Study ◽

Activity Evaluation ◽

Structure Activity ◽

Thiophene Series

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Antimicrobial properties of amine- and guanidine-functionalized derivatives of betulinic, ursolic and oleanolic acids: Synthesis and structure/activity evaluation

Steroids ◽

10.1016/j.steroids.2019.108530 ◽

2020 ◽

Vol 154 ◽

pp. 108530 ◽

Author(s):

Anna Yu. Spivak ◽

Rezeda R. Khalitova ◽

Darya A. Nedopekina ◽

Rinat R. Gubaidullin

Keyword(s):

Antimicrobial Properties ◽

Activity Evaluation ◽

Structure Activity ◽

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Systematic Drug Structure-Activity Evaluation/Correlation

Chemical Structures ◽

10.1007/978-3-642-73975-0_24 ◽

1988 ◽

pp. 235-241 ◽

Author(s):

Ernst Meyer ◽

Ehrhard Sens

Keyword(s):

Activity Evaluation ◽

Structure Activity

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Biological activity evaluation and structure–activity relationships analysis of ferulic acid and caffeic acid derivatives for anticancer

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/j.bmcl.2012.08.038 ◽

2012 ◽

Vol 22 (19) ◽

pp. 6085-6088 ◽

Author(s):

Weixia Li ◽

Nianguang Li ◽

Yuping Tang ◽

Baoquan Li ◽

Li Liu ◽

...

Keyword(s):

Biological Activity ◽

Ferulic Acid ◽

Caffeic Acid ◽

Caffeic Acid Derivatives ◽

Structure Activity Relationships ◽

Activity Evaluation ◽

Structure Activity

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Synthesis, Structure Activity Relationships and Biological Activity Evaluation of Novel Spirocyclic Thiazolidin-4-ones as Potential Anti-Breast Cancer and Epidermal Growth Factor Receptor Inhibitors

Drug Research ◽

10.1055/s-0033-1351314 ◽

2013 ◽

Vol 64 (01) ◽

pp. 23-30

Author(s):

D. Fleita ◽

O. Sakka ◽

R. Mohareb

Keyword(s):

Breast Cancer ◽

Epidermal Growth Factor Receptor ◽

Biological Activity ◽

Growth Factor ◽

Epidermal Growth Factor ◽

Growth Factor Receptor ◽

Structure Activity Relationships ◽

Activity Evaluation ◽

Structure Activity ◽

Epidermal Growth

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