Discovery and Bioevaluation of Novel Pyrazolopyrimidine Analogs as Competitive Hsp90 Inhibitors Through Shape-Based Similarity Screening

2014 ◽  
Vol 33 (4) ◽  
pp. 293-306 ◽  
Author(s):  
Xiao-Li Xu ◽  
Hao-Peng Sun ◽  
Fang Liu ◽  
Jian-Min Jia ◽  
Xiao-Ke Guo ◽  
...  
Keyword(s):  
Hsp90 Inhibitors

C-terminal Hsp90-inhibitors restore glucocorticoid sensitivity in Cushing's disease

2013 ◽  
Vol 121 (10) ◽  
Author(s):  
M Riebold ◽  
M Theodoropoulou ◽  
C Kozany ◽  
F Hausch ◽  
GK Stalla ◽  
...  
Keyword(s):  
Cushing’S Disease ◽  
Cushing's Disease ◽  
Hsp90 Inhibitors ◽  
Glucocorticoid Sensitivity

Discovery and Development of Pyrazole-Scaffold Hsp90 Inhibitors

2006 ◽  
Vol 6 (11) ◽  
pp. 1193-1203 ◽  
Author(s):  
Edward McDonald ◽  
Keith Jones ◽  
Paul Brough ◽  
Martin Drysdale ◽  
Paul Workman
Keyword(s):  
Hsp90 Inhibitors

Development and application of Hsp90 inhibitors

2008 ◽  
Vol 13 (1-2) ◽  
pp. 38-43 ◽  
Author(s):  
D SOLIT
Keyword(s):  
Hsp90 Inhibitors

scholarly journals The Anticancer Drug AUY922 Generates a Proteomics Fingerprint That Is Highly Conserved among Structurally Diverse Hsp90 Inhibitors

2013 ◽  
Vol 12 (8) ◽  
pp. 3697-3706 ◽  
Author(s):  
Sudhakar Voruganti ◽  
Jeff C. LaCroix ◽  
Chelsea N. Rogers ◽  
Janet Rogers ◽  
Robert L. Matts ◽  
...  
Keyword(s):  
Anticancer Drug ◽  
Hsp90 Inhibitors

Hsp90 inhibitors deplete key anti-apoptotic proteins in pediatric solid tumor cells and demonstrate synergistic anticancer activity with cisplatin

2004 ◽  
Vol 113 (2) ◽  
pp. 179-188 ◽  
Author(s):  
Rochelle Bagatell ◽  
Jason Beliakoff ◽  
Cynthia L. David ◽  
Marilyn T. Marron ◽  
Luke Whitesell
Keyword(s):  
Anticancer Activity ◽  
Tumor Cells ◽  
Solid Tumor ◽  
Hsp90 Inhibitors ◽  
Pediatric Solid Tumor ◽  
Apoptotic Proteins

scholarly journals Update on Hsp90 Inhibitors in Clinical Trial

2009 ◽  
Vol 9 (15) ◽  
pp. 1479-1492 ◽  
Author(s):  
Y. Kim ◽  
S. Alarcon ◽  
S. Lee ◽  
M.-J. Lee ◽  
G. Giaccone ◽  
...  
Keyword(s):  
Clinical Trial ◽  
Hsp90 Inhibitors
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