Synthesis, Biological Activity and Structure-Activity Relationship of Novel Diphenylurea Derivatives Containing Tetrahydroquinoline as Carbonic Anhydrase I and II Inhibitors

2018 ◽  
Vol 3 (2) ◽  
pp. 529-534 ◽  
Author(s):  
Alparslan Atahan ◽  
Nahit Gencer ◽  
Cigdem Bilen ◽  
Emre Yavuz ◽  
Hayriye Genc ◽  
...  
Keyword(s):  
Biological Activity ◽  
Carbonic Anhydrase ◽  
Structure Activity Relationship ◽  
Activity Relationship ◽  
Structure Activity ◽  
Carbonic Anhydrase I ◽  
Relationship Of

Synthesis of Hippospongic Acid A Analogues Designed for Investigating the Structure-Activity Relationship of its Biological Activity

2000 ◽  
Vol 53 (12) ◽  
pp. 909 ◽  
Author(s):  
Yoshikazu Hiraga ◽  
Mariko Ago ◽  
Munetaka Tokumasu ◽  
Ken Kaku ◽  
Katsuo Ohkata
Keyword(s):  
Biological Activity ◽  
Carboxylic Acid ◽  
Sea Urchin ◽  
Essential Feature ◽  
Structure Activity Relationship ◽  
Activity Relationship ◽  
Acid Moiety ◽  
Sea Urchin Embryos ◽  
Structure Activity ◽  
Relationship Of

Analogues of hippospongic acid A, which inhibit the gastrulation of sea urchin embryos, were synthesized. From a study on structure—activity relationships, the conjugated carboxylic acid moiety was found to be an essential feature for biological activity.

Synthesis, biological activity and structure–activity relationship of endomorphin-1/substance P derivatives

2012 ◽  
Vol 20 (21) ◽  
pp. 6335-6343 ◽  
Author(s):  
Pegah Varamini ◽  
Waleed M. Hussein ◽  
Friederike M. Mansfeld ◽  
Istvan Toth
Keyword(s):  
Biological Activity ◽  
Substance P ◽  
Structure Activity Relationship ◽  
Activity Relationship ◽  
Structure Activity ◽  
Relationship Of

Antiplasmodial activity of hydroxyethylamine analogs: Synthesis, biological activity and structure activity relationship of plasmepsin inhibitors

2018 ◽  
Vol 26 (13) ◽  
pp. 3837-3844 ◽  
Author(s):  
Amit Kumar Singh ◽  
Vinoth Rajendran ◽  
Snigdha Singh ◽  
Prashant Kumar ◽  
Yogesh Kumar ◽  
...  
Keyword(s):  
Biological Activity ◽  
Structure Activity Relationship ◽  
Antiplasmodial Activity ◽  
Activity Relationship ◽  
Structure Activity ◽  
Relationship Of

Expanding the structure-activity relationship of sulfoxaflor: the synthesis and biological activity ofN-heterocyclic sulfoximines

2014 ◽  
Vol 71 (7) ◽  
pp. 928-936 ◽  
Author(s):  
Benjamin M Nugent ◽  
Ann M Buysse ◽  
Michael R Loso ◽  
Jon M Babcock ◽  
Timothy C Johnson ◽  
...  
Keyword(s):  
Biological Activity ◽  
Structure Activity Relationship ◽  
Activity Relationship ◽  
Structure Activity ◽  
Relationship Of
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