Design, synthesis and biological evaluation of novel flavone Mannich base derivatives as potential antibacterial agents

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Hao Liu ◽  
Zi-Li Ren ◽  
Wei Wang ◽  
Feng Tang ◽  
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Diana K. Hunt ◽  
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Caprazamycin analogues, which were designed and synthesized via an aza-Prins–Ritter reaction, exhibit a good MraY and antibacterial activity without cytotoxicity against human cells.


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