The kappa-opioid receptor from human placenta: Hydrodynamic characteristics and evidence for its association with A G protein

Life Sciences ◽

10.1016/0024-3205(88)90159-2 ◽

1988 ◽

Vol 43 (6) ◽

pp. 559-567 ◽

Author(s):

G. Porthé ◽

B. Francés ◽

B. Vertier ◽

J. Cros ◽

J.-C. Meunier

Keyword(s):

G Protein ◽

Opioid Receptor ◽

Human Placenta ◽

Kappa Opioid Receptor ◽

Hydrodynamic Characteristics ◽

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The G protein-biased kappa opioid receptor agonist 6′-GNTI blocks hippocampal paroxysmal discharges without inducing aversion

Intrinsic Activity ◽

10.25006/ia.3.s2-a2.14 ◽

2015 ◽

Vol 3 (Suppl. 2) ◽

pp. A2.14

Author(s):

Luca Zangrandi

Keyword(s):

G Protein ◽

Opioid Receptor ◽

Receptor Agonist ◽

Kappa Opioid Receptor ◽

Kappa Opioid ◽

Opioid Receptor Agonist

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Faculty Opinions recommendation of Prolonged kappa opioid receptor phosphorylation mediated by G-protein receptor kinase underlies sustained analgesic tolerance.

Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature ◽

10.3410/f.1016246.200307 ◽

2003 ◽

Author(s):

Eric Nestler

Keyword(s):

G Protein ◽

Opioid Receptor ◽

Kappa Opioid Receptor ◽

Receptor Kinase ◽

Kappa Opioid ◽

Receptor Phosphorylation ◽

Analgesic Tolerance ◽

Protein Receptor

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Regulator of G Protein Signaling-12 (RGS12) in dopaminergic and kappa opioid receptor-dependent signaling and behavior

10.33915/etd.4060 ◽

2019 ◽

Author(s):

Joshua David Gross

Keyword(s):

G Protein ◽

Opioid Receptor ◽

Kappa Opioid Receptor ◽

G Protein Signaling ◽

Protein Signaling ◽

Kappa Opioid ◽

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Structure–Activity Relationship Studies of Functionally Selective Kappa Opioid Receptor Agonists that Modulate ERK 1/2 Phosphorylation While Preserving G Protein Over βArrestin2 Signaling Bias

ACS Chemical Neuroscience ◽

10.1021/acschemneuro.5b00092 ◽

2015 ◽

Vol 6 (8) ◽

pp. 1411-1419 ◽

Author(s):

Kimberly M. Lovell ◽

Kevin J. Frankowski ◽

Edward L. Stahl ◽

Stephen R. Slauson ◽

Euna Yoo ◽

...

Keyword(s):

G Protein ◽

Opioid Receptor ◽

Structure Activity Relationship ◽

Kappa Opioid Receptor ◽

Activity Relationship ◽

Kappa Opioid ◽

Receptor Agonists ◽

Structure Activity ◽

Opioid Receptor Agonists

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Activation of G-protein and c-Jun N-terminal kinase by kappa opioid receptor ligands

Drug and Alcohol Dependence ◽

10.1016/j.drugalcdep.2014.02.306 ◽

2014 ◽

Vol 140 ◽

pp. e106

Author(s):

B.I. Knapp ◽

Jean M. Bidlack

Keyword(s):

G Protein ◽

Opioid Receptor ◽

Kappa Opioid Receptor ◽

Receptor Ligands ◽

Kappa Opioid ◽

Opioid Receptor Ligands

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Characterization of the kappa opioid receptor‐mediated G protein signaling in mouse striatum using a [ 35 S]GTPγS binding assay (659.6)

The FASEB Journal ◽

10.1096/fasebj.28.1_supplement.659.6 ◽

2014 ◽

Vol 28 (S1) ◽

Author(s):

Lei Zhou ◽

Edward Stahl ◽

Kimberly Lovell ◽

Stephen Slauson ◽

Kevin Frankowski ◽

...

Keyword(s):

G Protein ◽

Opioid Receptor ◽

Binding Assay ◽

Kappa Opioid Receptor ◽

G Protein Signaling ◽

Protein Signaling ◽

Kappa Opioid ◽

Mouse Striatum ◽

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Prolonged Kappa Opioid Receptor Phosphorylation Mediated by G-protein Receptor Kinase Underlies Sustained Analgesic Tolerance

Journal of Biological Chemistry ◽

10.1074/jbc.m305796200 ◽

2003 ◽

Vol 279 (3) ◽

pp. 1810-1818 ◽

Author(s):

Jay P. McLaughlin ◽

Lisa C. Myers ◽

Paul E. Zarek ◽

Marc G. Caron ◽

Robert J. Lefkowitz ◽

...

Keyword(s):

G Protein ◽

Opioid Receptor ◽

Kappa Opioid Receptor ◽

Receptor Kinase ◽

Kappa Opioid ◽

Receptor Phosphorylation ◽

Analgesic Tolerance ◽

Protein Receptor

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Peripheral Kappa Opioid Receptor (KOR)‐Mediated Antinociception Requires G Protein‐Gated Inward Rectifying Potassium (GIRK) Channels

The FASEB Journal ◽

10.1096/fasebj.2019.33.1_supplement.808.18 ◽

2019 ◽

Vol 33 (S1) ◽

Author(s):

Miryam M. Pando ◽

Elaine M. Jennings ◽

William P. Clarke ◽

Kelly A. Berg

Keyword(s):

G Protein ◽

Opioid Receptor ◽

Kappa Opioid Receptor ◽

Kappa Opioid ◽

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G‐protein alpha subunits differentially alter the conformation of kappa opioid receptor

The FASEB Journal ◽

10.1096/fasebj.21.5.a429-c ◽

2007 ◽

Vol 21 (5) ◽

Author(s):

Feng Yan ◽

Bryan Roth

Keyword(s):

G Protein ◽

Opioid Receptor ◽

Kappa Opioid Receptor ◽

Kappa Opioid ◽

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Nalfurafine is a G-protein biased agonist having significantly greater bias at the human than rodent form of the kappa opioid receptor

Cellular Signalling ◽

10.1016/j.cellsig.2017.01.016 ◽

2017 ◽

Vol 32 ◽

pp. 59-65 ◽

Author(s):

Selena S. Schattauer ◽

Jamie R. Kuhar ◽

Allisa Song ◽

Charles Chavkin

Keyword(s):

G Protein ◽

Opioid Receptor ◽

Kappa Opioid Receptor ◽

Kappa Opioid ◽

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