Design, synthesis, biological evaluation, and computational studies of novel thiazolo-pyrazole hybrids as promising selective COX-2 inhibitors: Implementation of apoptotic genes expression for ulcerogenic liability assessment

2021 ◽  
Vol 111 ◽  
pp. 104883
Author(s):  
Adel A. Marzouk ◽  
Ehab S. Taher ◽  
Montaser Sh. A. Shaykoon ◽  
Ping Lan ◽  
Walaa Hamada Abd-Allah ◽  
...  
Keyword(s):  
Biological Evaluation ◽  
Computational Studies ◽  
Design Synthesis ◽  
Genes Expression ◽  
Cox 2 ◽  
Apoptotic Genes ◽  
Cox 2 Inhibitors

scholarly journals Design, Synthesis, Molecular Docking and Biological Evaluation of Novel Coumarin-Oxime Ether Derivatives as COX-2 Inhibitors

2017 ◽  
Vol 29 (11) ◽  
pp. 2559-2564
Author(s):  
M. Vijaya Bhargavi ◽  
P. Shashikala ◽  
M. Sumakanth ◽  
Shravan Kumar Gunda
Keyword(s):  
Molecular Docking ◽  
Biological Evaluation ◽  
Oxime Ether ◽  
Design Synthesis ◽  
Cox 2 ◽  
Cox 2 Inhibitors

Design, synthesis, and biological evaluation of substituted 3-alkylthio-4,5-diaryl-4H-1,2,4-triazoles as selective COX-2 inhibitors

2006 ◽  
Vol 14 (8) ◽  
pp. 2507-2517 ◽  
Author(s):  
Latifeh Navidpour ◽  
Hamed Shafaroodi ◽  
Khosrou Abdi ◽  
Mohsen Amini ◽  
Mohammad H. Ghahremani ◽  
...  
Keyword(s):  
Biological Evaluation ◽  
Design Synthesis ◽  
Cox 2 ◽  
Cox 2 Inhibitors ◽  
Synthesis And Biological Evaluation

Design, Synthesis and Biological Evaluation of New 1,3-diphenyl-3- (phenylamino)propan-1-ones as Selective Cyclooxygenase (COX-2) Inhibitors

2018 ◽  
Vol 14 (7) ◽  
pp. 652-659 ◽  
Author(s):  
Shabnam Farzaneh ◽  
Soraya Shahhosseini ◽  
Hadi Arefi ◽  
Bahram Daraei ◽  
Marjan Esfahanizadeh ◽  
...  
Keyword(s):  
Biological Evaluation ◽  
Design Synthesis ◽  
Cox 2 ◽  
Cox 2 Inhibitors ◽  
Synthesis And Biological Evaluation

Design, Synthesis, and Biological Evaluation of New Peptide Analogues as Selective COX-2 Inhibitors

2017 ◽  
Vol 350 (10) ◽  
pp. 1700158 ◽  
Author(s):  
Mohammad A. Ahmaditaba ◽  
Soraya Shahosseini ◽  
Bahram Daraei ◽  
Afshin Zarghi ◽  
Mohammad H. Houshdar Tehrani
Keyword(s):  
Biological Evaluation ◽  
Design Synthesis ◽  
Cox 2 ◽  
Cox 2 Inhibitors ◽  
Synthesis And Biological Evaluation ◽  
Peptide Analogues

Design, synthesis, biological evaluation and molecular modeling of dihydropyrazole sulfonamide derivatives as potential COX-1/COX-2 inhibitors

2015 ◽  
Vol 25 (9) ◽  
pp. 1947-1951 ◽  
Author(s):  
Zhong Chen ◽  
Zhong-Chang Wang ◽  
Xiao-Qiang Yan ◽  
Peng-Fei Wang ◽  
Xiao-Yuan Lu ◽  
...  
Keyword(s):  
Molecular Modeling ◽  
Biological Evaluation ◽  
Design Synthesis ◽  
Cox 2 ◽  
Cox 2 Inhibitors ◽  
Cox 1

Molecular design, synthesis and biological evaluation of cyclic imides bearing benzenesulfonamide fragment as potential COX-2 inhibitors. Part 2

2013 ◽  
Vol 23 (9) ◽  
pp. 2601-2605 ◽  
Author(s):  
Ibrahim A. Al-Suwaidan ◽  
Amer M. Alanazi ◽  
Adel S. El-Azab ◽  
Abdulrahman M. Al-Obaid ◽  
Kamal E.H. ElTahir ◽  
...  
Keyword(s):  
Molecular Design ◽  
Biological Evaluation ◽  
Design Synthesis ◽  
Cyclic Imides ◽  
Cox 2 ◽  
Cox 2 Inhibitors ◽  
Synthesis And Biological Evaluation
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