Synthesis, reactions and structure–activity relationships of 1-hydroxyspiro[2.5]cyclooct-4-en-3-ones: Illudin analogs with in vitro cytotoxic activity

Structure Activity ◽

Synthesis Reactions

In Vitro Cytotoxic Activity and Structure Activity Relationships of Iridoid Glucosides Derived from Veronica species

Phytotherapy Research ◽

10.1002/ptr.3546 ◽

2011 ◽

Vol 26 (1) ◽

pp. 148-152 ◽

Cited By ~ 17

Author(s):

Iclal Saracoglu ◽

U. Sebnem Harput

Keyword(s):

Cytotoxic Activity ◽

Structure Activity ◽

Iridoid Glucosides

In vitro cytotoxic activity of 1-alkylpiperidine N-oxides and quantitative structure-activity relationships

Anti-Cancer Drugs ◽

10.1097/00001813-199306000-00012 ◽

1993 ◽

Vol 4 (3) ◽

pp. 355-364 ◽

Cited By ~ 3

Author(s):

Milan Miko ◽

Ferdinand Devinsky

Keyword(s):

Cytotoxic Activity ◽

Quantitative Structure ◽

Quantitative Structure Activity Relationships

Structure Activity ◽

New bioactive 5-arylcarboximidamidopyrazolo[3,4-c]pyridines: Synthesis, cytotoxic activity, mechanistic investigation and structure-activity relationships

European Journal of Medicinal Chemistry ◽

10.1016/j.ejmech.2021.113387 ◽

2021 ◽

pp. 113387

Author(s):

Athanasios Papastathopoulos ◽

Nikolaos Lougiakis ◽

Ioannis K. Kostakis ◽

Panagiotis Marakos ◽

Nicole Pouli ◽

...

Keyword(s):

Cytotoxic Activity ◽

Structure Activity ◽

Mechanistic Investigation

Synthesis and structure-activity relationships of pyrimidine derivatives as potent and orally active FGFR3 inhibitors with both increased systemic exposure and enhanced in vitro potency

Bioorganic & Medicinal Chemistry ◽

10.1016/j.bmc.2021.116019 ◽

2021 ◽

Vol 33 ◽

pp. 116019

Author(s):

Ikumi Kuriwaki ◽

Minoru Kameda ◽

Kazuhiko Iikubo ◽

Hiroyuki Hisamichi ◽

Yuichiro Kawamoto ◽

...

Keyword(s):

Systemic Exposure ◽

Pyrimidine Derivatives ◽

Structure Activity ◽

Orally Active

Aqua mediated synthesis of 2-amino-6-benzothiazol-2-ylsulfanyl-chromenes and its in vitro study, explanation of the structure–activity relationships (SARs) as antibacterial agent

European Journal of Medicinal Chemistry ◽

10.1016/j.ejmech.2010.08.010 ◽

2010 ◽

Vol 45 (11) ◽

pp. 5031-5038 ◽

Cited By ~ 21

Author(s):

Mazaahir Kidwai ◽

Roona Poddar ◽

Saurav Bhardwaj ◽

Satendra Singh ◽

Pratibha Mehta Luthra

Keyword(s):

Antibacterial Agent ◽

In Vitro Study ◽

Vitro Study ◽

Structure-activity relationships of steroids in inducing germinal vesicle breakdown of Atlantic croaker oocytes in vitro

General and Comparative Endocrinology ◽

10.1016/0016-6480(88)90259-6 ◽

1988 ◽

Vol 71 (2) ◽

pp. 307-317 ◽

Cited By ~ 72

Author(s):

John M. Trant ◽

Peter Thomas

Keyword(s):

Germinal Vesicle ◽

Atlantic Croaker ◽

Germinal Vesicle Breakdown ◽

Structure-activity relationships and inhibitory effects of various purine derivatives on the in vitro growth of Plasmodium falciparum11Abbreviations: CDK, cyclin-dependent kinase; CDK1, cyclin-dependent kinase 1; and PfPK, Plasmodium falciparum protein kinase.

Biochemical Pharmacology ◽

10.1016/s0006-2952(01)00644-x ◽

2001 ◽

Vol 62 (3) ◽

pp. 341-348 ◽

Cited By ~ 37

Author(s):

Leonie Harmse ◽

Robyn van Zyl ◽

Nathanael Gray ◽

Peter Schultz ◽

Sophie Leclerc ◽

...

Keyword(s):

Plasmodium Falciparum ◽

Protein Kinase ◽

In Vitro Growth ◽

Cyclin Dependent Kinase ◽

Purine Derivatives ◽

Inhibitory Effects ◽

Structure Activity ◽

Falciparum Protein

Advances in Experimental Medicine and Biology - Biological Reactive Intermediates IV ◽

Structure-Activity Relationships of Acrylate Esters: Reactivity Towards Glutathione and Hydrolysis by Carboxylesterase in Vitro

10.1007/978-1-4684-5877-0_42 ◽

1991 ◽

pp. 333-335 ◽

Cited By ~ 5

Author(s):

T. J. McCarthy ◽

G. Witz

Keyword(s):

Structure Activity ◽

Acrylate Esters

Structure-activity relationships of cysteine esters and their effects on thiol levels in rat lung in vitro

Biochemical Pharmacology ◽

10.1016/0006-2952(93)90301-c ◽

1993 ◽

Vol 45 (8) ◽

pp. 1605-1612 ◽

Cited By ~ 17

Author(s):

M.J. Hobbs ◽

M. Butterworth ◽

G.M. Cohen ◽

D.G. Upshall

Keyword(s):

Rat Lung ◽

Structure-activity relationships of tetramethylpiperidine-substituted phenazines against Mycobacterium leprae in vitro.

Antimicrobial Agents and Chemotherapy ◽

10.1128/aac.33.11.2004 ◽

1989 ◽

Vol 33 (11) ◽

pp. 2004-2005 ◽

Cited By ~ 15

Author(s):

S G Franzblau ◽

K E White ◽

J F O'Sullivan

Keyword(s):

Mycobacterium Leprae ◽