Design, synthesis, and structure–activity relationship studies of novel thienopyrrolidone derivatives with strong antifungal activity against Aspergillus fumigates

Activity Relationship ◽

Design Synthesis ◽

Structure Activity ◽

Aspergillus Fumigates

Design, synthesis, and structure-activity relationship studies of novel triazole agents with strong antifungal activity against Aspergillus fumigatus

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/j.bmcl.2020.126951 ◽

2020 ◽

Vol 30 (4) ◽

pp. 126951 ◽

Cited By ~ 1

Author(s):

Zichao Ding ◽

Tingjunhong Ni ◽

Fei Xie ◽

Yumeng Hao ◽

Shichong Yu ◽

...

Keyword(s):

Antifungal Activity ◽

Aspergillus Fumigatus ◽

Activity Relationship ◽

Design Synthesis ◽

Benzoic acid derivatives with improved antifungal activity: Design, synthesis, structure–activity relationship (SAR) and CYP53 docking studies

Bioorganic & Medicinal Chemistry ◽

10.1016/j.bmc.2015.06.042 ◽

2015 ◽

Vol 23 (15) ◽

pp. 4264-4276 ◽

Cited By ~ 6

Author(s):

Sabina Berne ◽

Lidija Kovačič ◽

Matej Sova ◽

Nada Kraševec ◽

Stanislav Gobec ◽

...

Keyword(s):

Antifungal Activity ◽

Benzoic Acid ◽

Docking Studies ◽

Activity Relationship ◽

Design Synthesis ◽

Benzoic Acid Derivatives ◽

Structure Activity ◽

Activity Design

Design, synthesis, antifungal activity, and structure–activity relationship studies of chalcones and hybrid dihydrochromane–chalcones

Molecular Diversity ◽

10.1007/s11030-019-09967-y ◽

2019 ◽

Vol 24 (3) ◽

pp. 603-615 ◽

Cited By ~ 3

Author(s):

Marco Mellado ◽

Luis Espinoza ◽

Alejandro Madrid ◽

Jaime Mella ◽

Eduardo Chávez-Weisser ◽

...

Keyword(s):

Antifungal Activity ◽

Activity Relationship ◽

Design Synthesis ◽

Design, Synthesis and Structure-Activity Relationship Studies of Novel 4 (1-adamantyl) Phenyl Analogues as HIF-1α Inhibitors

Medicinal Chemistry ◽

10.2174/1573406412666151109113007 ◽

2016 ◽

Vol 12 (4) ◽

pp. 338-346 ◽

Cited By ~ 2

Author(s):

Yan Xia ◽

Qiong Duan ◽

Bao-Hua Zhao ◽

Dong-Feng Li ◽

Rui-Bin Hou

Keyword(s):

Activity Relationship ◽

Design Synthesis ◽

Design, synthesis, biological evaluation and structure-activity relationship study of quinazolin-4(3H)-one derivatives as novel USP7 inhibitors

European Journal of Medicinal Chemistry ◽

10.1016/j.ejmech.2021.113291 ◽

2021 ◽

pp. 113291

Author(s):

Peng Li ◽

Ying Liu ◽

Hua Yang ◽

Hong-Min Liu

Keyword(s):

Biological Evaluation ◽

Activity Relationship ◽

Design Synthesis ◽

Structure Activity ◽

Relationship Study

New substituted pyrazolones and dipyrazolotriazines as promising tyrosyl-tRNA synthetase and peroxiredoxin-5 inhibitors: Design, synthesis, molecular docking and structure-activity relationship (SAR) analysis

Bioorganic Chemistry ◽

10.1016/j.bioorg.2021.104704 ◽

2021 ◽

Vol 109 ◽

pp. 104704

Author(s):

Ismail M.M. Othman ◽

Mohamed A.M. Gad-Elkareem ◽

El Hassane Anouar ◽

Kaïss Aouadi ◽

Mejdi Snoussi ◽

...

Keyword(s):

Molecular Docking ◽

Trna Synthetase ◽

Activity Relationship ◽

Design Synthesis ◽

Structure Activity ◽

Sar Analysis

Antileishmanial Chalcones: Statistical Design, Synthesis, and Three-Dimensional Quantitative Structure−Activity Relationship Analysis

Journal of Medicinal Chemistry ◽

10.1021/jm980410m ◽

1998 ◽

Vol 41 (24) ◽

pp. 4819-4832 ◽

Cited By ~ 183

Author(s):

Simon Feldbæk Nielsen ◽

Søren Brøgger Christensen ◽

Gabriele Cruciani ◽

Arsalan Kharazmi ◽

Tommy Liljefors

Keyword(s):

Three Dimensional ◽

Statistical Design ◽

Quantitative Structure Activity Relationship ◽

Activity Relationship ◽

Quantitative Structure ◽

Design Synthesis ◽

Relationship Analysis ◽

Novel Pyrazole-4-acetohydrazide Derivatives Potentially Targeting Fungal Succinate Dehydrogenase: Design, Synthesis, Three-Dimensional Quantitative Structure–Activity Relationship, and Molecular Docking

Journal of Agricultural and Food Chemistry ◽

10.1021/acs.jafc.1c03399 ◽

2021 ◽

Author(s):

Xiaobin Wang ◽

Mengqi Wang ◽

Ling Han ◽

Fei Jin ◽

Jian Jiao ◽

...

Keyword(s):

Molecular Docking ◽

Succinate Dehydrogenase ◽

Three Dimensional ◽

Quantitative Structure Activity Relationship ◽

Activity Relationship ◽

Quantitative Structure ◽

Design Synthesis ◽

Design, synthesis and structure–activity relationship (SAR) studies of imidazo[4,5-b]pyridine derived purine isosteres and their potential as cytotoxic agents

European Journal of Medicinal Chemistry ◽

10.1016/j.ejmech.2014.10.037 ◽

2015 ◽

Vol 89 ◽

pp. 21-31 ◽

Cited By ~ 26

Author(s):

Ayyiliath M. Sajith ◽

K.K. Abdul Khader ◽

Nithin Joshi ◽

Manchala Nageswar Reddy ◽

M. Syed Ali Padusha ◽

...

Keyword(s):

Cytotoxic Agents ◽

Activity Relationship ◽

Design Synthesis ◽

Sar Studies ◽

New carboxamide derivatives bearing benzenesulphonamide as a selective COX-II inhibitor: Design, synthesis and structure-activity relationship

PLoS ONE ◽

10.1371/journal.pone.0183807 ◽

2017 ◽

Vol 12 (9) ◽

pp. e0183807 ◽

Cited By ~ 3

Author(s):

David Izuchukwu Ugwu ◽

Uchechukwu Chris Okoro ◽

Hilal Ahmad

Keyword(s):

Activity Relationship ◽

Inhibitor Design ◽

Design Synthesis ◽