Structural modifications in the distal, regulatory region of histamine H3 receptor antagonists leading to the identification of a potent anti-obesity agent

2020 ◽  
pp. 113041
Author(s):  
Katarzyna Szczepańska ◽  
Steffen Pockes ◽  
Sabina Podlewska ◽  
Carina Höring ◽  
Kamil Mika ◽  
...  
Keyword(s):  
Regulatory Region ◽  
Receptor Antagonists ◽  
Histamine H3 Receptor ◽  
Structural Modifications ◽  
H3 Receptor ◽  
Distal Regulatory Region ◽  
Histamine H3

ChemInform Abstract: 4-Chlorobenzyl Sulfonamide and Sulfamide Derivatives of Histamine Homologues: The Design of Potent Histamine H3 Receptor Antagonists.

ChemInform ◽  
2010 ◽  
Vol 31 (8) ◽  
pp. no-no
Author(s):  
Matthew J. Tozer ◽  
Ildiko M. Buck ◽  
Tracey Cooke ◽  
S. Barret Kalindjian ◽  
Iain M. McDonald ◽  
...  
Keyword(s):  
Receptor Antagonists ◽  
Histamine H3 Receptor ◽  
H3 Receptor ◽  
Derivatives Of ◽  
Histamine H3

ChemInform Abstract: Substituted N-Phenylcarbamates as Histamine H3 Receptor Antagonists with Improved in vivo Potency.

ChemInform ◽  
2010 ◽  
Vol 31 (24) ◽  
pp. no-no
Author(s):  
S. Reidemeister ◽  
H. Stark ◽  
X. Ligneau ◽  
C. R. Ganellin ◽  
J.-C. Schwartz ◽  
...  
Keyword(s):  
Receptor Antagonists ◽  
Histamine H3 Receptor ◽  
H3 Receptor ◽  
Histamine H3

Piperidine-Containing Histamine H3 Receptor Antagonists of the Carbamate Series: The Influence of the Additional Ether Functionality

ChemInform ◽  
2003 ◽  
Vol 34 (16) ◽  
Author(s):  
D. Lazewska ◽  
K. Kiec-Kononowicz ◽  
H. H. Pertz ◽  
S. Elz ◽  
H. Stark ◽  
...  
Keyword(s):  
Receptor Antagonists ◽  
Histamine H3 Receptor ◽  
H3 Receptor ◽  
Histamine H3

Keynote review: Histamine H3 receptor antagonists reach out for the clinic

2005 ◽  
Vol 10 (23-24) ◽  
pp. 1613-1627 ◽  
Author(s):  
Sylvain Celanire ◽  
Maikel Wijtmans ◽  
Patrice Talaga ◽  
Rob Leurs ◽  
Iwan J.P. de Esch
Keyword(s):  
Receptor Antagonists ◽  
Histamine H3 Receptor ◽  
H3 Receptor ◽  
Histamine H3

Non-imidazole heterocyclic histamine H3 receptor antagonists

2003 ◽  
Vol 13 (10) ◽  
pp. 1767-1770 ◽  
Author(s):  
Wenying Chai ◽  
J.Guy Breitenbucher ◽  
Annette Kwok ◽  
Xiaobing Li ◽  
Victoria Wong ◽  
...  
Keyword(s):  
Receptor Antagonists ◽  
Histamine H3 Receptor ◽  
H3 Receptor ◽  
Histamine H3
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