scholarly journals Computational analysis of novel drugs designed for use as acetylcholinesterase inhibitors and histamine H3 receptor antagonists for Alzheimer's disease by docking, scoring and de novo evolution

2012 ◽  
Vol 5 (4) ◽  
pp. 1043-1048 ◽  
Author(s):  
PO-YUAN CHEN ◽  
CHING-TSAN TSAI ◽  
CHE-YEN OU ◽  
WEI-TSE HSU ◽  
MIEN-DE JHUO ◽  
...  
Keyword(s):  
Alzheimer’S Disease ◽  
Alzheimer's Disease ◽  
Computational Analysis ◽  
De Novo ◽  
Acetylcholinesterase Inhibitors ◽  
Receptor Antagonists ◽  
Histamine H3 Receptor ◽  
H3 Receptor ◽  
Novel Drugs ◽  
Histamine H3

Rational design of new multitarget histamine H3 receptor ligands as potential candidates for treatment of Alzheimer’s disease

2020 ◽  
Vol 207 ◽  
pp. 112743
Author(s):  
Dorota Łażewska ◽  
Marek Bajda ◽  
Maria Kaleta ◽  
Paula Zaręba ◽  
Agata Doroz-Płonka ◽  
...  
Keyword(s):  
Alzheimer’S Disease ◽  
Alzheimer's Disease ◽  
Rational Design ◽  
Receptor Ligands ◽  
Histamine H3 Receptor ◽  
H3 Receptor ◽  
Histamine H3

Search for new multi-target compounds against Alzheimer’s disease among histamine H3 receptor ligands

2020 ◽  
Vol 185 ◽  
pp. 111785 ◽  
Author(s):  
Marek Bajda ◽  
Dorota Łażewska ◽  
Justyna Godyń ◽  
Paula Zaręba ◽  
Kamil Kuder ◽  
...  
Keyword(s):  
Alzheimer’S Disease ◽  
Alzheimer's Disease ◽  
Receptor Ligands ◽  
Histamine H3 Receptor ◽  
H3 Receptor ◽  
Histamine H3

Lead identification of acetylcholinesterase inhibitors–histamine H3 receptor antagonists from molecular modeling

2008 ◽  
Vol 16 (6) ◽  
pp. 2968-2973 ◽  
Author(s):  
Scott D. Bembenek ◽  
John M. Keith ◽  
Michael A. Letavic ◽  
Richard Apodaca ◽  
Ann J. Barbier ◽  
...  
Keyword(s):  
Molecular Modeling ◽  
Acetylcholinesterase Inhibitors ◽  
Receptor Antagonists ◽  
Histamine H3 Receptor ◽  
H3 Receptor ◽  
Lead Identification ◽  
Histamine H3

ChemInform Abstract: 4-Chlorobenzyl Sulfonamide and Sulfamide Derivatives of Histamine Homologues: The Design of Potent Histamine H3 Receptor Antagonists.

ChemInform ◽  
2010 ◽  
Vol 31 (8) ◽  
pp. no-no
Author(s):  
Matthew J. Tozer ◽  
Ildiko M. Buck ◽  
Tracey Cooke ◽  
S. Barret Kalindjian ◽  
Iain M. McDonald ◽  
...  
Keyword(s):  
Receptor Antagonists ◽  
Histamine H3 Receptor ◽  
H3 Receptor ◽  
Derivatives Of ◽  
Histamine H3

ChemInform Abstract: Substituted N-Phenylcarbamates as Histamine H3 Receptor Antagonists with Improved in vivo Potency.

ChemInform ◽  
2010 ◽  
Vol 31 (24) ◽  
pp. no-no
Author(s):  
S. Reidemeister ◽  
H. Stark ◽  
X. Ligneau ◽  
C. R. Ganellin ◽  
J.-C. Schwartz ◽  
...  
Keyword(s):  
Receptor Antagonists ◽  
Histamine H3 Receptor ◽  
H3 Receptor ◽  
Histamine H3
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