Dietary flavonoids fisetin and myricetin: Dual inhibitors of Plasmodium falciparum falcipain-2 and plasmepsin II

Fitoterapia ◽  
2014 ◽  
Vol 94 ◽  
pp. 55-61 ◽  
Author(s):  
Huangtao Jin ◽  
Zhongyu Xu ◽  
Kunqiang Cui ◽  
Tianshu Zhang ◽  
Weiqiang Lu ◽  
...  
Keyword(s):  
Plasmodium Falciparum ◽  
Dual Inhibitors ◽  
Plasmepsin Ii ◽  
Dietary Flavonoids

In Vitro Antimalarial Evaluation of Piperidine- and Piperazine-Based Chalcones: Inhibition of Falcipain-2 and Plasmepsin II Hemoglobinases Activities from Plasmodium falciparum

2017 ◽  
Vol 2 (25) ◽  
pp. 7684-7690 ◽  
Author(s):  
Hemandra Kumar Tiwari ◽  
Prashant Kumar ◽  
Nidhi Jatana ◽  
Krishan Kumar ◽  
Sandeep Garg ◽  
...  
Keyword(s):  
Plasmodium Falciparum ◽  
Plasmepsin Ii

scholarly journals Discovery of oxybisbenzoylamides as a new class of antimalarial agents

MedChemComm ◽  
2015 ◽  
Vol 6 (6) ◽  
pp. 1173-1177 ◽  
Author(s):  
A. Pancotti ◽  
S. Parapini ◽  
M. Dell'Agli ◽  
L. Gambini ◽  
C. Galli ◽  
...  
Keyword(s):  
Plasmodium Falciparum ◽  
New Class ◽  
Antimalarial Agents ◽  
Dual Inhibitors

A new antimalarial pharmacophore has been obtained starting from previously described dual inhibitors of Plasmodium falciparum.

Selective inhibitors of plasmepsin II of Plasmodium falciparum on the basis of pepstatin

2008 ◽  
Vol 34 (6) ◽  
pp. 660-667
Author(s):  
L. D. Rumsh ◽  
A. G. Mikhailova ◽  
I. V. Mikhura ◽  
I. A. Prudchenko ◽  
L. D. Chikin ◽  
...  
Keyword(s):  
Plasmodium Falciparum ◽  
Selective Inhibitors ◽  
Plasmepsin Ii

Spermine alkaloids from Albizia adinocephala with activity against Plasmodium falciparum plasmepsin II

2002 ◽  
Vol 60 (2) ◽  
pp. 175-177 ◽  
Author(s):  
Simon P.B Ovenden ◽  
Shugeng Cao ◽  
Chungyan Leong ◽  
Horst Flotow ◽  
Mahabir P Gupta ◽  
...  
Keyword(s):  
Plasmodium Falciparum ◽  
Plasmepsin Ii

scholarly journals Overexpression of plasmepsin II and plasmepsin III does not directly cause reduction in Plasmodium falciparum sensitivity to artesunate, chloroquine and piperaquine

2019 ◽  
Vol 9 ◽  
pp. 16-22 ◽  
Author(s):  
Duangkamon Loesbanluechai ◽  
Namfon Kotanan ◽  
Cristina de Cozar ◽  
Theerarat Kochakarn ◽  
Megan R. Ansbro ◽  
...  
Keyword(s):  
Plasmodium Falciparum ◽  
Plasmepsin Ii

Identification of potent inhibitors of Plasmodium falciparum plasmepsin II from an encoded statine combinatorial library

1998 ◽  
Vol 8 (17) ◽  
pp. 2315-2320 ◽  
Author(s):  
Carolyn DiIanni Carroll ◽  
Hitesh Patel ◽  
Theodore O. Johnson ◽  
Tao Guo ◽  
Marc Orlowski ◽  
...  
Keyword(s):  
Plasmodium Falciparum ◽  
Combinatorial Library ◽  
Plasmepsin Ii

scholarly journals Potent dual inhibitors of Plasmodium falciparum M1 and M17 aminopeptidases through optimization of S1 pocket interactions

2016 ◽  
Vol 110 ◽  
pp. 43-64 ◽  
Author(s):  
Nyssa Drinkwater ◽  
Natalie B. Vinh ◽  
Shailesh N. Mistry ◽  
Rebecca S. Bamert ◽  
Chiara Ruggeri ◽  
...  
Keyword(s):  
Plasmodium Falciparum ◽  
Dual Inhibitors
Sign in / Sign up

Export Citation Format

Share Document