Itching-like behavior: A common effect of the kappa opioid receptor antagonist 5'-guanidinonaltrindole and the biased kappa opioid receptor agonist 6'-guanidinonaltrindole in mice

Common Effect ◽

Nalbuphine, a kappa opioid receptor agonist and mu opioid receptor antagonist attenuates pruritus, decreases IL-31, and increases IL-10 in mice with contact dermatitis

European Journal of Pharmacology ◽

10.1016/j.ejphar.2019.172702 ◽

2019 ◽

Vol 864 ◽

pp. 172702 ◽

Cited By ~ 8

Author(s):

Saadet Inan ◽

Alvaro Torres-Huerta ◽

Liselotte E. Jensen ◽

Nae J. Dun ◽

Alan Cowan

Keyword(s):

Contact Dermatitis ◽

Receptor Antagonist ◽

Opioid Receptor ◽

Receptor Agonist ◽

Mu Opioid Receptor ◽

Kappa Opioid Receptor ◽

Kappa Opioid ◽

Mu Opioid ◽

244 Efficacy of kappa-opioid receptor agonist and mu-opioid receptor antagonist to treat itch in imiquimod-induced psoriasis-like dermatitis model

Journal of Investigative Dermatology ◽

10.1016/j.jid.2016.06.264 ◽

2016 ◽

Vol 136 (9) ◽

pp. S203

Author(s):

N. Takahashi ◽

M. Tominaga ◽

Y. Kamata ◽

Y. Umehara ◽

H. Matsuda ◽

...

Keyword(s):

Receptor Antagonist ◽

Opioid Receptor ◽

Receptor Agonist ◽

Mu Opioid Receptor ◽

Kappa Opioid Receptor ◽

Kappa Opioid ◽

Mu Opioid ◽

The G protein-biased kappa opioid receptor agonist 6′-GNTI blocks hippocampal paroxysmal discharges without inducing aversion

Intrinsic Activity ◽

10.25006/ia.3.s2-a2.14 ◽

2015 ◽

Vol 3 (Suppl. 2) ◽

pp. A2.14

Author(s):

Luca Zangrandi

Keyword(s):

G Protein ◽

Opioid Receptor ◽

Receptor Agonist ◽

Kappa Opioid Receptor ◽

Kappa Opioid ◽

Faculty Opinions recommendation of Chronic peripheral administration of kappa-opioid receptor antagonist advances puberty onset associated with acceleration of pulsatile luteinizing hormone secretion in female rats.

Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature ◽

10.3410/f.718110987.793483835 ◽

2013 ◽

Author(s):

Pamela Mellon ◽

Alexander Kauffman

Keyword(s):

Luteinizing Hormone ◽

Receptor Antagonist ◽

Opioid Receptor ◽

Hormone Secretion ◽

Kappa Opioid Receptor ◽

Female Rats ◽

Luteinizing Hormone Secretion ◽

Kappa Opioid ◽

Puberty Onset

Effect of Difelikefalin, a Selective Kappa Opioid Receptor Agonist, on Respiratory Depression: A Randomized, Double‐Blind, Placebo‐Controlled Trial

Clinical and Translational Science ◽

10.1111/cts.13042 ◽

2021 ◽

Author(s):

Eugene R. Viscusi ◽

Marc C. Torjman ◽

Catherine L. Munera ◽

Joseph W. Stauffer ◽

Beatrice S. Setnik ◽

...

Keyword(s):

Respiratory Depression ◽

Opioid Receptor ◽

Receptor Agonist ◽

Controlled Trial ◽

Kappa Opioid Receptor ◽

Kappa Opioid ◽

Double Blind ◽

Double Blind Placebo ◽

Blockade of ethanol reward by the kappa opioid receptor agonist U50,488H

Alcohol ◽

10.1016/j.alcohol.2009.05.001 ◽

2009 ◽

Vol 43 (5) ◽

pp. 359-365 ◽

Cited By ~ 53

Author(s):

Marian L. Logrip ◽

Patricia H. Janak ◽

Dorit Ron

Keyword(s):

Opioid Receptor ◽

Receptor Agonist ◽

Kappa Opioid Receptor ◽

Kappa Opioid ◽

A unique binding epitope for salvinorin A, a non-nitrogenous kappa opioid receptor agonist

FEBS Journal ◽

10.1111/j.1742-4658.2006.05212.x ◽

2006 ◽

Vol 273 (9) ◽

pp. 1966-1974 ◽

Cited By ~ 27

Author(s):

Brian E. Kane ◽

Marcelo J. Nieto ◽

Christopher R. McCurdy ◽

David M. Ferguson

Keyword(s):

Opioid Receptor ◽

Receptor Agonist ◽

Kappa Opioid Receptor ◽

Salvinorin A ◽

Kappa Opioid ◽

Opioid Receptor Agonist ◽

Binding Epitope

The Kappa-Opioid Receptor Agonist MR-2034 Stimulates the Rat Hypothalamic-Pituitary-Adrenal Axis: Studiesin vivoandin vitro

Journal of Neuroendocrinology ◽

10.1111/j.1365-2826.1996.tb00691.x ◽

1996 ◽

Vol 8 (8) ◽

pp. 579-585 ◽

Cited By ~ 31

Author(s):

A. E. Calogero ◽

S. Scaccianoce ◽

N. Burrello ◽

R. Nicolai ◽

L. A. A. Muscolo ◽

...

Keyword(s):

Opioid Receptor ◽

Receptor Agonist ◽

Kappa Opioid Receptor ◽

Hypothalamic Pituitary Adrenal Axis ◽

Kappa Opioid ◽

Hypothalamic Pituitary Adrenal ◽

Adrenal Axis ◽

Opioid Receptor Agonist ◽

Pituitary Adrenal Axis

Effects of the Kappa-opioid Receptor Agonist, U69593, on the Development of Sensitization and on the Maintenance of Cocaine Self-administration

Neuropsychopharmacology ◽

10.1016/s0893-133x(00)00190-1 ◽

2001 ◽

Vol 24 (4) ◽

pp. 441-450 ◽

Cited By ~ 17

Author(s):

S Schenk

Keyword(s):

Opioid Receptor ◽

Receptor Agonist ◽

Kappa Opioid Receptor ◽

Self Administration ◽

Kappa Opioid ◽

Synthesis and Structure–Activity Relationships of 5′-Aryl-14-alkoxypyridomorphinans: Identification of a μ Opioid Receptor Agonist/δ Opioid Receptor Antagonist Ligand with Systemic Antinociceptive Activity and Diminished Opioid Side Effects

Journal of Medicinal Chemistry ◽

10.1021/acs.jmedchem.0c00503 ◽

2020 ◽

Vol 63 (14) ◽

pp. 7663-7694 ◽

Cited By ~ 2

Author(s):

Rakesh H. Vekariya ◽

Wei Lei ◽

Abhisek Ray ◽

Surendra K. Saini ◽

Sixue Zhang ◽

...

Keyword(s):

Side Effects ◽

Receptor Antagonist ◽

Opioid Receptor ◽

Receptor Agonist ◽

Antinociceptive Activity ◽

Structure Activity ◽

Opioid Receptor Agonist ◽

Μ Opioid Receptor ◽

Δ Opioid Receptor