Synthesis of novel cycloheptylbenzothiazole-2-carboxamides and biological evaluation as human estrogen receptor modulators

Human Estrogen Receptor ◽

The Human Estrogen Receptor-α Is a Ubiquitinated Protein Whose Stability Is Affected Differentially by Agonists, Antagonists, and Selective Estrogen Receptor Modulators

Journal of Biological Chemistry ◽

10.1074/jbc.m101097200 ◽

2001 ◽

Vol 276 (38) ◽

pp. 35684-35692 ◽

Cited By ~ 278

Author(s):

Ashini L. Wijayaratne ◽

Donald P. McDonnell

Keyword(s):

Estrogen Receptor ◽

Estrogen Receptor Α ◽

Ubiquitinated Protein ◽

Human Estrogen Receptor ◽

Human estrogen receptor-α (ER-α) transactivation by selective estrogen receptor modulators (SERMs) on VIT regulatory region in ER-α-negative breast cancer cell line Evsa-T transiently transfected by ER-α

Breast Cancer Research ◽

10.1186/bcr372 ◽

2001 ◽

Vol 3 (S1) ◽

Author(s):

IP Nyamagana Butera ◽

S Hadiy ◽

G Leclercq

Keyword(s):

Breast Cancer ◽

Estrogen Receptor ◽

Cell Line ◽

Breast Cancer Cell Line ◽

Regulatory Region ◽

Cancer Cell Line ◽

Estrogen Receptor Α ◽

Human Estrogen Receptor ◽

Synthesis, biological evaluation, structural–activity relationship, and docking study for a series of benzoxepin-derived estrogen receptor modulators

Bioorganic & Medicinal Chemistry ◽

10.1016/j.bmc.2008.09.035 ◽

2008 ◽

Vol 16 (21) ◽

pp. 9554-9573 ◽

Cited By ~ 33

Author(s):

Irene Barrett ◽

Mary J. Meegan ◽

Rosario B. Hughes ◽

Miriam Carr ◽

Andrew J.S. Knox ◽

...

Keyword(s):

Estrogen Receptor ◽

Docking Study ◽

Biological Evaluation ◽

Activity Relationship ◽

Structural Activity Relationship ◽

3,5-Diphenylpyrazolylethanone Derivatives as Selective Estrogen Receptor Modulators: Design, Synthesis, Biological Evaluation and Docking Analysis

Indo Global Journal of Pharmaceutical Sciences ◽

10.35652/igjps.2020.10104 ◽

2020 ◽

Vol 10 (01) ◽

pp. 25-32

Author(s):

Pritam N. Dube ◽

Vivekanand A. Chatpalliwar

Keyword(s):

Estrogen Receptor ◽

Biological Evaluation ◽

Design Synthesis ◽

Docking Analysis ◽

Design, synthesis and biological evaluation of novel indole-xanthendione hybrids as selective estrogen receptor modulators

Bioorganic & Medicinal Chemistry ◽

10.1016/j.bmc.2017.11.040 ◽

2018 ◽

Vol 26 (1) ◽

pp. 266-277 ◽

Cited By ~ 8

Author(s):

Ramit Singla ◽

Kunj Bihari Gupta ◽

Shishir Upadhyay ◽

Monisha Dhiman ◽

Vikas Jaitak

Keyword(s):

Estrogen Receptor ◽

Biological Evaluation ◽

Design Synthesis ◽

Synthesis And Biological Evaluation

Receptor Modulators ◽

Design, synthesis and biological evaluation of novel 2-methoxyestradiol analogs as dual selective estrogen receptor modulators (SERMs) and antiangiogenic agents

European Journal of Medicinal Chemistry ◽

10.1016/j.ejmech.2017.08.016 ◽

2017 ◽

Vol 139 ◽

pp. 390-400 ◽

Cited By ~ 3

Author(s):

Kejing Lao ◽

Yejun Wang ◽

Mingqi Chen ◽

Jingjing Zhang ◽

Qidong You ◽

...

Keyword(s):

Estrogen Receptor ◽

Biological Evaluation ◽

Antiangiogenic Agents ◽

Design Synthesis ◽

Synthesis And Biological Evaluation

Receptor Modulators ◽

A review of selective estrogen receptor modulators in the treatment of breast and endometrial cancer

Seminars in Oncology ◽

10.1053/sonc.2002.34065 ◽

2002 ◽

Vol 29 (3 Suppl 11) ◽

pp. 129-133 ◽

Cited By ~ 27

Author(s):

Stephen Chan

Keyword(s):

Estrogen Receptor ◽

Endometrial Cancer ◽

Faculty Opinions recommendation of FDA-approved selective estrogen receptor modulators inhibit Ebola virus infection.

Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature ◽

10.3410/f.718030692.793484645 ◽

2013 ◽

Author(s):

Anne Moscona ◽

Laura M Palermo ◽

Matteo Porotto

Keyword(s):

Estrogen Receptor ◽

Virus Infection ◽

Ebola Virus ◽

Receptor Modulators ◽

Ebola Virus Infection

Definition of the Molecular Mechanisms Which Distinguish Between Selective Estrogen Receptor Modulators (SERMs) and Full Antiestrogens

10.21236/ada426883 ◽

2004 ◽

Author(s):

Huey-Jing Huang

Keyword(s):

Estrogen Receptor ◽

Molecular Mechanisms ◽

Definition Of ◽

Definition of the Molecular Mechanisms Which Distinguish Between Selective Estrogen Receptor Modulators (SERMs) and Full Antiestrogens

10.21236/ada436900 ◽

2005 ◽

Author(s):

Huey-Jing Huang

Keyword(s):

Estrogen Receptor ◽

Molecular Mechanisms ◽

Definition Of ◽