Clean and efficient microwave-solvent-free conversion of homochiral amines, α-amino alcohols and α-amino acids to their chiral 2-substituted pyrrole derivatives

Tetrahedron ◽  
2005 ◽  
Vol 61 (12) ◽  
pp. 3019-3023 ◽  
Author(s):  
Feray Aydogan ◽  
Ayhan S. Demir
Keyword(s):  
Amino Acids ◽  
Amino Alcohols ◽  
Solvent Free ◽  
Pyrrole Derivatives

ChemInform Abstract: Conversion of Homochiral Amines, β-Amino Alcohols and α-Amino Acids to Their Chiral 2-Substituted Pyrrole Derivatives.

ChemInform ◽  
2010 ◽  
Vol 32 (50) ◽  
pp. no-no
Author(s):  
Ayhan S. Demir ◽  
Idris M. Akhmedov ◽  
Oezge Sesenoglu ◽  
Onur Alptuerk ◽  
Sinem Apaydin ◽  
...  
Keyword(s):  
Amino Acids ◽  
Amino Alcohols ◽  
Pyrrole Derivatives

Conversion of homochiral amines, β-amino alcohols and α-amino acids to their chiral 2-substituted pyrrole derivatives

2001 ◽  
pp. 1162-1167 ◽  
Author(s):  
Ayhan S. Demir ◽  
Idris M. Akhmedov ◽  
Özge Şeşenoglu ◽  
Onur Alptürk ◽  
Sinem Apaydın ◽  
...  
Keyword(s):  
Amino Acids ◽  
Amino Alcohols ◽  
Pyrrole Derivatives

scholarly journals Rapid Organocatalytic Chirality Analysis of Amines, Amino Acids, Alcohols, Amino Alcohols and Diols with Achiral Iso(thio)cyanate Probes

2021 ◽  
Author(s):  
Eryn Nelson ◽  
Jeffrey S. S. K. Formen ◽  
Christian Wolf
Keyword(s):  
Amino Acids ◽  
Absolute Configuration ◽  
Rapid Determination ◽  
Amino Alcohols ◽  
Enantioselective Synthesis ◽  
Widespread Occurrence ◽  
Chiral Compounds ◽  
New Methods ◽  
The Absolute

The widespread occurrence and significance of chiral compounds does not only require new methods for their enantioselective synthesis but also efficient tools that allow rapid determination of the absolute configuration,...

Chirality Sensing of Amines, Diamines, Amino Acids, Amino Alcohols, and α-Hydroxy Acids with a Single Probe

2013 ◽  
Vol 135 (48) ◽  
pp. 18052-18055 ◽  
Author(s):  
Keith W. Bentley ◽  
Yea G. Nam ◽  
Jaslynn M. Murphy ◽  
Christian Wolf
Keyword(s):  
Amino Acids ◽  
Amino Alcohols ◽  
Hydroxy Acids ◽  
Single Probe

N-Substituted α-trifluoromethyl β-nitro amines in the synthesis of fluorine-containing 1,2-diamines, amino alcohols, and β-amino acids

2009 ◽  
Vol 58 (9) ◽  
pp. 1886-1898 ◽  
Author(s):  
V. Yu. Korotaev ◽  
A. Yu. Barkov ◽  
M. I. Kodess ◽  
I. B. Kutyashev ◽  
P. A. Slepukhin ◽  
...  
Keyword(s):  
Amino Acids ◽  
Amino Alcohols

ChemInform Abstract: Trifluoromethyl syn- or anti-γ-Amino Alcohols by One-Pot Solvent-Free Mannich-Type Reactions under Temperature Control.

ChemInform ◽  
2015 ◽  
Vol 46 (34) ◽  
pp. no-no
Author(s):  
Stefania Fioravanti ◽  
Luca Parise ◽  
Alessia Pelagalli ◽  
Lucio Pellacani ◽  
Laura Trulli
Keyword(s):  
Temperature Control ◽  
Amino Alcohols ◽  
Solvent Free ◽  
One Pot

Coupling of Steroid O-(Carboxymethyl)oxime Derivatives with Amino Alcohols

1996 ◽  
Vol 61 (2) ◽  
pp. 288-297 ◽  
Author(s):  
Vladimír Pouzar ◽  
Ivan Černý
Keyword(s):  
Amino Acids ◽  
Hydroxy Group ◽  
Building Blocks ◽  
Amino Alcohols ◽  
New Approach ◽  
Alternative Synthesis ◽  
Oxime Derivatives ◽  
A Chain ◽  
Derivatives Of

New approach to the preparation of steroids with connecting bridge, based on an O-carboxymethyloxime (CMO) structure, and with terminal hydroxy group, is presented. 17-CMO derivatives of 3β-acetoxy- and 3β-methoxymethoxyandrost-5-en-17-one were condensed with α,ω-amino alcohols to give derivatives with a chain of seven to nine atoms. After THP-protection, these compounds were converted to 3-keto-4-ene derivatives. An alternative synthesis consisted in transformation of 17-CMO derivatives with bonded amino acids by reduction of the terminal carboxyl. The resulting compounds were designed as building blocks for the preparation of bis-haptens for sandwich immunoassays.

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