Effect of the acyl groups on O→N acyl migration in the water-soluble prodrugs of HIV-1 protease inhibitor

2003 ◽  
Vol 13 (16) ◽  
pp. 2727-2730 ◽  
Author(s):  
Yoshio Hamada ◽  
Hikaru Matsumoto ◽  
Tooru Kimura ◽  
Yoshio Hayashi ◽  
Yoshiaki Kiso
Keyword(s):  
Protease Inhibitor ◽  
Acyl Migration ◽  
Water Soluble ◽  
Hiv 1

Coupling of an Acyl Migration Prodrug Strategy with Bio-activation To Improve Oral Delivery of the HIV-1 Protease Inhibitor Atazanavir

2018 ◽  
Vol 61 (9) ◽  
pp. 4176-4188 ◽  
Author(s):  
Murugaiah A. M. Subbaiah ◽  
Nicholas A. Meanwell ◽  
John F. Kadow ◽  
Lakshumanan Subramani ◽  
Mathiazhagan Annadurai ◽  
...  
Keyword(s):  
Protease Inhibitor ◽  
Oral Delivery ◽  
Acyl Migration ◽  
Hiv 1

O—N Intramolecular Acyl Migration Strategy in Water-Soluble Prodrugs of Taxoids.

ChemInform ◽  
2004 ◽  
Vol 35 (13) ◽  
Author(s):  
Mariusz Skwarczynski ◽  
Youhei Sohma ◽  
Maiko Kimura ◽  
Yoshio Hayashi ◽  
Tooru Kimura ◽  
...  
Keyword(s):  
Acyl Migration ◽  
Water Soluble ◽  
Migration Strategy

scholarly journals Simplification Therapy with Once‐Daily Emtricitabine, Didanosine, and Efavirenz in HIV‐1–Infected Adults with Viral Suppression Receiving a Protease Inhibitor–Based Regimen: A Randomized Trial

2005 ◽  
Vol 191 (6) ◽  
pp. 830-839 ◽  
Author(s):  
Jean‐Michel Molina ◽  
Valérie Journot ◽  
Laurence Morand‐Joubert ◽  
Patrick Yéni ◽  
Willy Rozenbaum ◽  
...  
Keyword(s):  
Protease Inhibitor ◽  
Randomized Trial ◽  
Viral Suppression ◽  
Once Daily ◽  
Hiv 1
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