Design, Synthesis, and Characterization of the Macrocyclic Tetrapeptide cyclo[Pro-Sar-Phe-d-Phe]: A Mixed Opioid Receptor Agonist–Antagonist Following Oral Administration

2020 ◽  
Vol 11 (9) ◽  
pp. 1324-1336 ◽  
Author(s):  
Michael J. Ferracane ◽  
Ariana C. Brice-Tutt ◽  
Jeremy S. Coleman ◽  
Grant G. Simpson ◽  
Lisa L. Wilson ◽  
...  
Keyword(s):  
Oral Administration ◽  
Opioid Receptor ◽  
Receptor Agonist ◽  
Synthesis And Characterization ◽  
Design Synthesis ◽  
Opioid Receptor Agonist

scholarly journals Synthesis and Characterization of a Dual Kappa-Delta Opioid Receptor Agonist Analgesic Blocking Cocaine Reward Behavior

2015 ◽  
Vol 6 (11) ◽  
pp. 1813-1824 ◽  
Author(s):  
András Váradi ◽  
Gina F. Marrone ◽  
Shainnel O. Eans ◽  
Michelle L. Ganno ◽  
Joan J. Subrath ◽  
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Keyword(s):  
Opioid Receptor ◽  
Receptor Agonist ◽  
Synthesis And Characterization ◽  
Delta Opioid Receptor ◽  
Opioid Receptor Agonist ◽  
Cocaine Reward

Design, synthesis, and characterization of 6β-naltrexol analogs, and their selectivity for in vitro opioid receptor subtypes

2009 ◽  
Vol 19 (10) ◽  
pp. 2811-2814 ◽  
Author(s):  
Andrea L. Pelotte ◽  
Ryan M. Smith ◽  
Mario Ayestas ◽  
Christina M. Dersch ◽  
Edward J. Bilsky ◽  
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Keyword(s):  
Opioid Receptor ◽  
Synthesis And Characterization ◽  
Receptor Subtypes ◽  
Design Synthesis ◽  
Opioid Receptor Subtypes

Characterization of the complex morphinan derivative BU72 as a high efficacy, long-lasting mu-opioid receptor agonist

2004 ◽  
Vol 499 (1-2) ◽  
pp. 107-116 ◽  
Author(s):  
Claire L. Neilan ◽  
Stephen M. Husbands ◽  
Simon Breeden ◽  
M.C. (Holden) Ko ◽  
Mario D. Aceto ◽  
...  
Keyword(s):  
Opioid Receptor ◽  
Receptor Agonist ◽  
Mu Opioid Receptor ◽  
High Efficacy ◽  
Mu Opioid ◽  
Opioid Receptor Agonist

scholarly journals Characterization of methadone as a β-arrestin-biased μ-opioid receptor agonist

2016 ◽  
Vol 12 ◽  
pp. 174480691665414 ◽  
Author(s):  
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Tomohisa Mori ◽  
Naoki Uzawa ◽  
Takamichi Arima ◽  
Tomoyuki Takahashi ◽  
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Keyword(s):  
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Receptor Agonist ◽  
Opioid Receptor Agonist ◽  
Μ Opioid Receptor
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