Design of Novel Cyclic Hexapeptide Somatostatin Analogs from a Model of the Bioactive Conformation

ACS Symposium Series - Conformationally Directed Drug Design ◽

10.1021/bk-1984-0251.ch008 ◽

1984 ◽

pp. 169-187 ◽

Author(s):

ROGER M. FREIDINGER ◽

DANIEL F. VEBER

Keyword(s):

Somatostatin Analogs ◽

Bioactive Conformation ◽

Cyclic Hexapeptide

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Conformational modifications of cyclic hexapeptide somatostatin analogs

International journal of peptide & protein research ◽

10.1111/j.1399-3011.1984.tb02704.x ◽

2009 ◽

Vol 23 (2) ◽

pp. 142-150 ◽

Author(s):

Roger M. Freidinger ◽

Debra Schwenk Perlow ◽

William C. Randall ◽

Richard Saperstein ◽

Byron H. Arison ◽

...

Keyword(s):

Somatostatin Analogs ◽

Cyclic Hexapeptide

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4486415 Cyclic hexapeptide somatostatin analogs

Biotechnology Advances ◽

10.1016/0734-9750(85)90147-8 ◽

1985 ◽

Vol 3 (1) ◽

pp. 118

Keyword(s):

Somatostatin Analogs ◽

Cyclic Hexapeptide

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4522813 Cyclic hexapeptide somatostatin analogs

Biotechnology Advances ◽

10.1016/0734-9750(85)90395-7 ◽

1985 ◽

Vol 3 (2) ◽

pp. 263-264

Keyword(s):

Somatostatin Analogs ◽

Cyclic Hexapeptide

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Evidence for the bioactive conformation in a cyclic hexapeptide analogue of somatostatin containing a cis-peptide bond mimic

Biochemical and Biophysical Research Communications ◽

10.1016/0006-291x(88)90170-2 ◽

1988 ◽

Vol 154 (2) ◽

pp. 515-521 ◽

Author(s):

M. Elseviers ◽

L. Van Der Auwera ◽

H. Pepermans ◽

D. Tourwé ◽

G. Van Binst

Keyword(s):

Peptide Bond ◽

Bioactive Conformation ◽

Cyclic Hexapeptide

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Presurgical treatment with somatostatin analogs in patients with acromegaly: effects on the remission and complication rates

Yearbook of Neurology and Neurosurgery ◽

10.1016/s0513-5117(08)70205-9 ◽

2007 ◽

Vol 2007 ◽

pp. 297-298

Author(s):

K. Erkmen

Keyword(s):

Somatostatin Analogs ◽

Complication Rates

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Characterization and sub-cellular localization of somatostatin receptors in DU-145 and PC-3 human androgen-independent prostate cancer cells: effect of mono- and bi-specific somatostatin analogs on cell growth

Endocrine Abstracts ◽

10.1530/endoabs.32.p514 ◽

2013 ◽

Author(s):

Massimiliano Ruscica ◽

Marica Arvigo ◽

Liliana Steffani ◽

Federico Gatto ◽

Manuela Albertelli ◽

...

Keyword(s):

Prostate Cancer ◽

Cell Growth ◽

Cancer Cells ◽

Cellular Localization ◽

Somatostatin Receptors ◽

Somatostatin Analogs ◽

Prostate Cancer Cells ◽

Androgen Independent

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T2-weighted MRI signal and response to somatostatin analogs in acromegaly

Endocrine Abstracts ◽

10.1530/endoabs.49.ep1062 ◽

2017 ◽

Author(s):

Luis Cerqueira ◽

Ana Palha ◽

Luisa Cortez ◽

Amets Sagarribay ◽

Fernando Fonseca ◽

...

Keyword(s):

Somatostatin Analogs

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Efficacy and safety of telotristat ethyl in patients with carcinoid syndrome inadequately controlled by somatostatin analogs: Analysis of the completed TELESTAR extension period

Endocrine Abstracts ◽

10.1530/endoabs.52.p14 ◽

2017 ◽

Author(s):

D Horsch ◽

MH Kulke ◽

M Caplin ◽

L Anthony ◽

E Bergsland ◽

...

Keyword(s):

Carcinoid Syndrome ◽

Somatostatin Analogs ◽

Efficacy And Safety ◽

Extension Period

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Faculty Opinions recommendation of Preliminary data on biochemical remission of acromegaly after somatostatin analogs withdrawal.

Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature ◽

10.3410/f.1136911.623608 ◽

2009 ◽

Author(s):

Marcello Bronstein

Keyword(s):

Preliminary Data ◽

Somatostatin Analogs ◽

Biochemical Remission

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Faculty Opinions recommendation of Partial surgical removal of growth hormone-secreting pituitary tumors enhances the response to somatostatin analogs in acromegaly.

Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature ◽

10.3410/f.723735015.793511706 ◽

2015 ◽

Author(s):

Niki Karavitaki ◽

Georgia Ntali

Keyword(s):

Growth Hormone ◽

Somatostatin Analogs ◽

Pituitary Tumors ◽

Surgical Removal

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