Pyrrolobenzoxazepinone Derivatives as Non-Nucleoside HIV-1 RT Inhibitors:  Further Structure−Activity Relationship Studies and Identification of More Potent Broad-Spectrum HIV-1 RT Inhibitors with Antiviral Activity

1999 ◽  
Vol 42 (21) ◽  
pp. 4462-4470 ◽  
Author(s):  
Giuseppe Campiani ◽  
Elena Morelli ◽  
Monica Fabbrini ◽  
Vito Nacci ◽  
Giovanni Greco ◽  
...  
Keyword(s):  
Antiviral Activity ◽  
Broad Spectrum ◽  
Structure Activity Relationship ◽  
Activity Relationship ◽  
Structure Activity ◽  
Rt Inhibitors ◽  
Hiv 1

scholarly journals Synthesis, Antiviral Activity, and Structure–Activity Relationship of 1,3‐Benzodioxolyl Pyrrole‐Based Entry Inhibitors Targeting the Phe43 Cavity in HIV‐1 gp120

ChemMedChem ◽  
2018 ◽  
Vol 13 (21) ◽  
pp. 2332-2348 ◽  
Author(s):  
Francesca Curreli ◽  
Dmitry S. Belov ◽  
Shahad Ahmed ◽  
Ranjith R. Ramesh ◽  
Alexander V. Kurkin ◽  
...  
Keyword(s):  
Antiviral Activity ◽  
Structure Activity Relationship ◽  
Activity Relationship ◽  
Entry Inhibitors ◽  
Structure Activity ◽  
Relationship Of ◽  
Hiv 1

Structure–activity relationship of neomycin, paromomycin, and neamine–arginine conjugates, targeting HIV-1 gp120–CXCR4 binding step

2003 ◽  
Vol 60 (3) ◽  
pp. 181-192 ◽  
Author(s):  
Gadi Borkow ◽  
Veerappan Vijayabaskar ◽  
Humberto Herman Lara ◽  
Alexander Kalinkovich ◽  
Aviva Lapidot
Keyword(s):  
Structure Activity Relationship ◽  
Activity Relationship ◽  
Structure Activity ◽  
Relationship Of ◽  
Hiv 1

scholarly journals Isothiazolo[4,3-b]pyridines as inhibitors of cyclin G associated kinase: synthesis, structure–activity relationship studies and antiviral activity

MedChemComm ◽  
2015 ◽  
Vol 6 (9) ◽  
pp. 1666-1672 ◽  
Author(s):  
Jiahong Li ◽  
Sona Kovackova ◽  
Szuyuan Pu ◽  
Jef Rozenski ◽  
Steven De Jonghe ◽  
...  
Keyword(s):  
Antiviral Activity ◽  
Structure Activity Relationship ◽  
Activity Relationship ◽  
Structure Activity ◽  
Cyclin G

Starting from a known isothiazolo[4,3-b]pyridine scaffold, different series of novel, potent GAK ligands were synthesized.

scholarly journals Structure–Activity Relationship Studies of HIV-1 Integrase Oligonucleotide Inhibitors

2011 ◽  
Vol 2 (7) ◽  
pp. 532-537 ◽  
Author(s):  
Julia Agapkina ◽  
Timofei Zatsepin ◽  
Ekaterina Knyazhanskaya ◽  
Jean-Francois Mouscadet ◽  
Marina Gottikh
Keyword(s):  
Structure Activity Relationship ◽  
Activity Relationship ◽  
Structure Activity ◽  
Hiv 1

Anti-HIV-1 activity of thiadiazole derivatives: structure-activity relationship, reverse transcriptase inhibition, and lipophilicity

1996 ◽  
Vol 31 (1-2) ◽  
pp. 87-94 ◽  
Author(s):  
Katsushi Ijichi ◽  
Masatoshi Fujiwara ◽  
Hideki Nagano ◽  
Yukiharu Matsumoto ◽  
Yasuaki Hanasaki ◽  
...  
Keyword(s):  
Reverse Transcriptase ◽  
Structure Activity Relationship ◽  
Activity Relationship ◽  
Structure Activity ◽  
Thiadiazole Derivatives ◽  
Anti Hiv ◽  
Hiv 1
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