One-pot, highly efficient, asymmetric synthesis of ring-fused piperidine derivatives bearing N,O- or N,N-acetal moieties
2016 ◽
Vol 14
(8)
◽
pp. 2444-2453
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Keyword(s):
One Pot
◽
Lactols or cyclic hemiaminals are directly used as nucleophiles in the asymmetric aza-Diels–Alder reaction to synthesize ring-fused piperidine derivatives.