Neuroimaging of histamine H1
-receptor occupancy in human brain by positron emission tomography (PET): A comparative study of ebastine, a second-generation antihistamine, and (+)-chlorpheniramine, a classical antihistamine

Comparative Study ◽

Human Brain ◽

Second Generation ◽

Receptor Occupancy ◽

Emission Tomography ◽

H1 Receptor ◽

Histamine H1 Receptor ◽

Positron Emission ◽

Histamine H1 Receptor Occupancy in the Human Brain Measured by Positron Emission Tomography

Histamine Receptors ◽

10.1007/978-3-319-40308-3_13 ◽

2016 ◽

pp. 311-325

Author(s):

Kazuhiko Yanai ◽

Kotaro Hiraoka ◽

Anikó Kárpáti ◽

Fumito Naganuma ◽

Nobuyuki Okamura ◽

...

Keyword(s):

Human Brain ◽

Receptor Occupancy ◽

Emission Tomography ◽

H1 Receptor ◽

Histamine H1 Receptor ◽

Positron Emission ◽

Histamine H1 receptor occupancy by the new-generation antipsychotics olanzapine and quetiapine: a positron emission tomography study in healthy volunteers

Psychopharmacology ◽

10.1007/s00213-015-4002-2 ◽

2015 ◽

Vol 232 (19) ◽

pp. 3497-3505 ◽

Cited By ~ 13

Author(s):

Hirotoshi Sato ◽

Chihiro Ito ◽

Kotaro Hiraoka ◽

Manabu Tashiro ◽

Katsuhiko Shibuya ◽

...

Keyword(s):

Healthy Volunteers ◽

Receptor Occupancy ◽

Emission Tomography ◽

Positron Emission Tomography Study ◽

H1 Receptor ◽

Histamine H1 Receptor ◽

Positron Emission ◽

New Generation ◽

Histamine H1 receptor occupancy by the new-generation antidepressants fluvoxamine and mirtazapine: a positron emission tomography study in healthy volunteers

Psychopharmacology ◽

10.1007/s00213-013-3146-1 ◽

2013 ◽

Vol 230 (2) ◽

pp. 227-234 ◽

Cited By ~ 12

Author(s):

Hirotoshi Sato ◽

Chihiro Ito ◽

Manabu Tashiro ◽

Kotaro Hiraoka ◽

Katsuhiko Shibuya ◽

...

Keyword(s):

Healthy Volunteers ◽

Receptor Occupancy ◽

Emission Tomography ◽

Positron Emission Tomography Study ◽

H1 Receptor ◽

Histamine H1 Receptor ◽

Positron Emission ◽

New Generation ◽

Brain histamine H1 receptor occupancy of orally administered antihistamines measured by positron emission tomography with 11C-doxepin in a placebo-controlled crossover study design in healthy subjects: a comparison of olopatadine and ketotifen

British Journal of Clinical Pharmacology ◽

10.1111/j.1365-2125.2005.02514.x ◽

2006 ◽

Vol 61 (1) ◽

pp. 16-26 ◽

Cited By ~ 49

Author(s):

Manabu Tashiro ◽

Hideki Mochizuki ◽

Yumiko Sakurada ◽

Kenji Ishii ◽

Keiichi Oda ◽

...

Keyword(s):

Crossover Study ◽

Study Design ◽

Healthy Subjects ◽

Receptor Occupancy ◽

Emission Tomography ◽

H1 Receptor ◽

Brain Histamine ◽

Positron Emission ◽

Neuroimaging of histamine H1-receptor in the schizophrenic human brain by positron emission tomography

International Clinical Psychopharmacology ◽

10.1097/00004850-200305000-00016 ◽

2003 ◽

Vol 18 (3) ◽

pp. 180 ◽

Cited By ~ 2

Author(s):

Kentaro Iwabuchi ◽

Chihiro Ito ◽

Yasuhiko Kubota ◽

Manabu Tashiro ◽

Motohisa Kato ◽

...

Keyword(s):

Human Brain ◽

Emission Tomography ◽

H1 Receptor ◽

Histamine H1 Receptor ◽

Positron Emission

Central Effects of Fexofenadine and Cetirizine: Measurement of Psychomotor Performance, Subjective Sleepiness, and Brain Histamine H1-Receptor Occupancy Using11C-Doxepin Positron Emission Tomography

The Journal of Clinical Pharmacology ◽

10.1177/0091270004267590 ◽

2004 ◽

Vol 44 (8) ◽

pp. 890-900 ◽

Cited By ~ 89

Author(s):

Manabu Tashiro ◽

Yumiko Sakurada ◽

Kentaro Iwabuchi ◽

Hideki Mochizuki ◽

Motohisa Kato ◽

...

Keyword(s):

Psychomotor Performance ◽

Receptor Occupancy ◽

Emission Tomography ◽

H1 Receptor ◽

Brain Histamine ◽

Central Effects ◽

Positron Emission ◽

Subjective Sleepiness ◽

Histamine H1 receptor occupancy in human brains after single oral doses of histamine H1 antagonists measured by positron emission tomography

British Journal of Pharmacology ◽

10.1111/j.1476-5381.1995.tb16386.x ◽

1995 ◽

Vol 116 (1) ◽

pp. 1649-1655 ◽

Cited By ~ 78

Author(s):

Kazuhiko Yanai ◽

Jong Hoon Ryu ◽

Takehiko Watanabe ◽

Ren Iwata ◽

Tatsuo Ido ◽

...

Keyword(s):

Receptor Occupancy ◽

Emission Tomography ◽

H1 Receptor ◽

Positron Emission ◽

Human Brains ◽

Oral Doses ◽

H1 Antagonists ◽

Histamine H1 Antagonists ◽

No regional difference in dopamine D2 receptor occupancy by the second-generation antipsychotic drug risperidone in humans: a positron emission tomography study

The International Journal of Neuropsychopharmacology ◽

10.1017/s1461145708009577 ◽

2008 ◽

Vol 12 (05) ◽

pp. 667 ◽

Cited By ~ 18

Author(s):

Hiroshi Ito ◽

Ryosuke Arakawa ◽

Hidehiko Takahashi ◽

Harumasa Takano ◽

Masaki Okumura ◽

...

Keyword(s):

Antipsychotic Drug ◽

Regional Difference ◽

Second Generation ◽

Dopamine D2 Receptor ◽

D2 Receptor ◽

Receptor Occupancy ◽

Emission Tomography ◽

Positron Emission ◽

Second Generation Antipsychotic

Histamine H1 receptor occupancy in the human brain after single oral doses of antihistamines measured by PET.

The Japanese Journal of Pharmacology ◽

10.1016/s0021-5198(19)36339-5 ◽

1996 ◽

Vol 71 ◽

pp. 19

Author(s):

Kazuhiko Yanai ◽

Takehiko Watanabe

Keyword(s):

Human Brain ◽

Receptor Occupancy ◽

H1 Receptor ◽

Histamine H1 Receptor ◽

Oral Doses ◽

Central benzodiazepine receptor occupancy by zolpidem in the human brain as assessed by positron emission tomography

European Journal of Pharmacology ◽

10.1016/0014-2999(95)00633-8 ◽

1996 ◽

Vol 295 (1) ◽

pp. 35-44 ◽

Cited By ~ 38

Author(s):

Pascale Abadie ◽

Patrice Rioux ◽

Bernard Scatton ◽

Edouard Zarifian ◽

Louisa Barré ◽

...

Keyword(s):

Human Brain ◽

Receptor Occupancy ◽

Benzodiazepine Receptor ◽

Emission Tomography ◽

Positron Emission ◽

Central Benzodiazepine Receptor