Identification of pathway-selective estrogen receptor ligands that inhibit NF- B transcriptional activity

Proceedings of the National Academy of Sciences ◽

10.1073/pnas.0405841102 ◽

2005 ◽

Vol 102 (7) ◽

pp. 2543-2548 ◽

Author(s):

C. C. Chadwick ◽

S. Chippari ◽

E. Matelan ◽

L. Borges-Marcucci ◽

A. M. Eckert ◽

...

Keyword(s):

Estrogen Receptor ◽

Transcriptional Activity ◽

Receptor Ligands ◽

Estrogen Receptor Ligands

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Transcriptional activity and biological effects of mammalian estrogen receptor ligands on three hepatic estrogen receptors in Mozambique tilapia

The Journal of Steroid Biochemistry and Molecular Biology ◽

10.1016/j.jsbmb.2010.05.009 ◽

2010 ◽

Vol 122 (4) ◽

pp. 272-278 ◽

Author(s):

L.K. Davis ◽

Y. Katsu ◽

T. Iguchi ◽

D.T. Lerner ◽

T. Hirano ◽

...

Keyword(s):

Estrogen Receptor ◽

Estrogen Receptors ◽

Transcriptional Activity ◽

Biological Effects ◽

Receptor Ligands ◽

Mozambique Tilapia ◽

Estrogen Receptor Ligands

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The utility of pathway selective estrogen receptor ligands that inhibit nuclear factor-κB transcriptional activity in models of rheumatoid arthritis

Arthritis Research & Therapy ◽

10.1186/ar1692 ◽

2005 ◽

Vol 7 (3) ◽

Author(s):

James C Keith ◽

Leo M Albert ◽

Yelena Leathurby ◽

Max Follettie ◽

Lili Wang ◽

...

Keyword(s):

Rheumatoid Arthritis ◽

Estrogen Receptor ◽

Transcriptional Activity ◽

Nuclear Factor Κb ◽

Nuclear Factor ◽

Receptor Ligands ◽

Estrogen Receptor Ligands

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Identification of estrogen receptor ligands leading to activation of non-genomic signaling pathways while exhibiting only weak transcriptional activity

The Journal of Steroid Biochemistry and Molecular Biology ◽

10.1016/j.jsbmb.2005.08.003 ◽

2006 ◽

Vol 98 (1) ◽

pp. 25-35 ◽

Author(s):

Silja Wessler ◽

Christiane Otto ◽

Nicola Wilck ◽

Verena Stangl ◽

Karl-Heinrich Fritzemeier

Keyword(s):

Estrogen Receptor ◽

Signaling Pathways ◽

Transcriptional Activity ◽

Receptor Ligands ◽

Estrogen Receptor Ligands

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Cyclopentadienyl Rhenium (Technetium) Tricarbonyl Complexes Integrated in Estrogen Receptor Ligands for ER+ Tumor Imaging

10.21236/ada456153 ◽

2005 ◽

Author(s):

Nathan C. Ackroyd ◽

John A. Katzenellenbogen

Keyword(s):

Estrogen Receptor ◽

Tumor Imaging ◽

Receptor Ligands ◽

Estrogen Receptor Ligands

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A Bipartite Recombinant Yeast System for the Identification of Subtype-Selective Estrogen Receptor Ligands

Molecular Biotechnology ◽

10.1007/s12033-008-9141-9 ◽

2009 ◽

Vol 41 (3) ◽

pp. 307-307

Author(s):

Kaiwei Liang ◽

Liuqing Yang ◽

Zhimin Xiao ◽

Jian Huang

Keyword(s):

Estrogen Receptor ◽

Recombinant Yeast ◽

Receptor Ligands ◽

Estrogen Receptor Ligands ◽

Subtype Selective

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Conformational Analysis of Bivalent Estrogen Receptor Ligands: From Intramolecular to Intermolecular Binding

ChemBioChem ◽

10.1002/cbic.201100529 ◽

2011 ◽

Vol 12 (17) ◽

pp. 2587-2598 ◽

Author(s):

Min Shan ◽

Alexander Bujotzek ◽

Frank Abendroth ◽

Anja Wellner ◽

Ronald Gust ◽

...

Keyword(s):

Estrogen Receptor ◽

Conformational Analysis ◽

Receptor Ligands ◽

Estrogen Receptor Ligands

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A Computationally Based Identification Algorithm for Estrogen Receptor Ligands: Part 2. Evaluation of a hERalpha Binding Affinity Model

Toxicological Sciences ◽

10.1093/toxsci/58.2.270 ◽

2000 ◽

Vol 58 (2) ◽

pp. 270-281 ◽

Author(s):

O. G. Mekenyan

Keyword(s):

Estrogen Receptor ◽

Binding Affinity ◽

Identification Algorithm ◽

Receptor Ligands ◽

Affinity Model ◽

Estrogen Receptor Ligands

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ChemInform Abstract: Binary Quantitative Structure-Activity Relationship (QSAR) Analysis of Estrogen Receptor Ligands.

10.1002/chin.199921263 ◽

2010 ◽

Vol 30 (21) ◽

pp. no-no

Author(s):

Hua Gao ◽

Chris Williams ◽

Paul Labute ◽

Juergen Bajorath

Keyword(s):

Estrogen Receptor ◽

Quantitative Structure Activity Relationship ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Quantitative Structure ◽

Receptor Ligands ◽

Qsar Analysis ◽

Structure Activity ◽

Estrogen Receptor Ligands

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Ketamine and ketamine metabolites as novel estrogen receptor ligands: Induction of cytochrome P450 and AMPA glutamate receptor gene expression

Biochemical Pharmacology ◽

10.1016/j.bcp.2018.03.032 ◽

2018 ◽

Vol 152 ◽

pp. 279-292 ◽

Author(s):

Ming-Fen Ho ◽

Cristina Correia ◽

James N. Ingle ◽

Rima Kaddurah-Daouk ◽

Liewei Wang ◽

...

Keyword(s):

Gene Expression ◽

Estrogen Receptor ◽

Cytochrome P450 ◽

Glutamate Receptor ◽

Receptor Gene ◽

Receptor Ligands ◽

Estrogen Receptor Ligands ◽

Receptor Gene Expression

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Exploiting Nongenomic Estrogen Receptor-Mediated Signaling for the Development of Pathway-Selective Estrogen Receptor Ligands

Tissue-Specific Estrogen Action - Ernst Schering Foundation Symposium Proceedings ◽

10.1007/2789_2006_022 ◽

2007 ◽

pp. 163-181 ◽

Author(s):

C. Otto ◽

S. Wessler ◽

K.-H. Fritzemeier

Keyword(s):

Estrogen Receptor ◽

Receptor Ligands ◽

Estrogen Receptor Ligands

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