Design, synthesis, and bioactivity investigation of novel benzimidazole derivatives as potent urease inhibitors

2021 ◽  
pp. 1-11
Author(s):  
Ebrahim Saeedian Moghadam ◽  
Abdullah Mohammed Al-Saadi ◽  
Meysam Talebi ◽  
Massoud Amanlou ◽  
Mohsen Amini ◽  
...  
Keyword(s):  
Benzimidazole Derivatives ◽  
Urease Inhibitors ◽  
Design Synthesis

Novel thiobarbiturates as potent urease inhibitors with potential antibacterial activity: Design, synthesis, radiolabeling and biodistribution study

2020 ◽  
Vol 28 (23) ◽  
pp. 115759
Author(s):  
Hanan Gaber Abdulwahab ◽  
Marwa F. Harras ◽  
Nagwan Galal El Menofy ◽  
Amany M. Hegab ◽  
Basma M. Essa ◽  
...  
Keyword(s):  
Antibacterial Activity ◽  
Biodistribution Study ◽  
Urease Inhibitors ◽  
Design Synthesis ◽  
Activity Design

scholarly journals Design, synthesis, biological assessment and in silico ADME prediction of new 2-(4-(methylsulfonyl) phenyl) benzimidazoles as selective cyclooxygenase-2 inhibitors

RSC Advances ◽  
2021 ◽  
Vol 11 (44) ◽  
pp. 27659-27673
Author(s):  
Mohamed A. S. Badawy ◽  
Eman K. A. Abdelall ◽  
EL-Shaymaa EL-Nahass ◽  
Khaled R. A. Abdellatif ◽  
Hamdy M. Abdel-Rahman
Keyword(s):  
In Silico ◽  
Cyclooxygenase 2 ◽  
Biological Assessment ◽  
Benzimidazole Derivatives ◽  
Design Synthesis ◽  
Adme Prediction ◽  
In Silico Adme Prediction ◽  
Cyclooxygenase 2 Inhibitors

A novel series of benzimidazole derivatives wherein 4-(methylsulfonyl) phenyl pharmacophore attached via its C-2 position was designed and synthesized.

Design, synthesis and docking studies of benzimidazole derivatives as potential EGFR inhibitors

2019 ◽  
Vol 173 ◽  
pp. 240-249 ◽  
Author(s):  
İsmail Celik ◽  
Gülgün Ayhan-Kılcıgil ◽  
Berna Guven ◽  
Zümra Kara ◽  
A. Selen Gurkan-Alp ◽  
...  
Keyword(s):  
Docking Studies ◽  
Egfr Inhibitors ◽  
Benzimidazole Derivatives ◽  
Design Synthesis

Design, synthesis and biological evaluation of some novel benzimidazole derivatives for their potential anticonvulsant activity

2010 ◽  
Vol 33 (7) ◽  
pp. 971-980 ◽  
Author(s):  
Priyal Jain ◽  
Prakash Kumar Sharma ◽  
Harish Rajak ◽  
Rajesh Singh Pawar ◽  
Umesh Kumar Patil ◽  
...  
Keyword(s):  
Anticonvulsant Activity ◽  
Biological Evaluation ◽  
Benzimidazole Derivatives ◽  
Design Synthesis ◽  
Synthesis And Biological Evaluation

Design, synthesis, mechanistic studies and in silico ADME predictions of benzimidazole derivatives as novel antifungal agents

2020 ◽  
Vol 101 ◽  
pp. 103956 ◽  
Author(s):  
Martha M. Morcoss ◽  
El Shimaa M.N. Abdelhafez ◽  
Reham A. Ibrahem ◽  
Hamdy M. Abdel-Rahman ◽  
Mohamed Abdel-Aziz ◽  
...  
Keyword(s):  
In Silico ◽  
Antifungal Agents ◽  
Benzimidazole Derivatives ◽  
Mechanistic Studies ◽  
Design Synthesis

Design, synthesis, and characterization of some new benzimidazole derivatives and biological evaluation

2020 ◽  
Vol 57 (5) ◽  
pp. 2234-2242
Author(s):  
Hakan Bektaş ◽  
Bahar B. Sökmen ◽  
Sinem Aydın ◽  
Emre Menteşe ◽  
Adile Bektaş ◽  
...  
Keyword(s):  
Biological Evaluation ◽  
Synthesis And Characterization ◽  
Benzimidazole Derivatives ◽  
Design Synthesis
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