Pharmacological characterization of high‐affinity σ
            1
            receptor ligands with spirocyclic thienopyran and thienofuran scaffold

Pharmacological Characterization of Novel High Affinity CGRP Receptor Antagonists that are Selective for Human CGRP Receptors

The FASEB Journal ◽

10.1096/fasebj.20.4.a665-a ◽

2006 ◽

Vol 20 (4) ◽

Author(s):

Chrsitopher K. Taylor ◽

D. David Smith ◽

Peter W. Abel

Keyword(s):

Cgrp Receptor ◽

Receptor Antagonists ◽

High Affinity ◽

Cgrp Receptor Antagonists

Pharmacological characterization of F-180: a selective human V1a vasopressin receptor agonist of high affinity

British Journal of Pharmacology ◽

10.1038/sj.bjp.0704634 ◽

2002 ◽

Vol 135 (7) ◽

pp. 1828-1836 ◽

Cited By ~ 21

Author(s):

Miriam Andrés ◽

Miguel Trueba ◽

Gilles Guillon

Keyword(s):

Receptor Agonist ◽

Vasopressin Receptor ◽

Pharmacological Characterization of Human κ / μ Opioid Receptor Chimeras that Retain High Affinity for Dynorphin A

Current Topics in Medicinal Chemistry ◽

10.2174/1568026053544542 ◽

2005 ◽

Vol 5 (3) ◽

pp. 303-313 ◽

Cited By ~ 8

Author(s):

Robert DeHaven ◽

Erik Mansson ◽

Jeffrey Daubert ◽

Joel Cassel

Keyword(s):

Opioid Receptor ◽

Dynorphin A ◽

High Affinity ◽

Receptor Chimeras

ChemInform Abstract: High-Affinity Leukotriene Receptor Antagonists. Synthesis and Pharmacological Characterization of 2-Hydroxy-3-((2-carboxyethyl)thio)-3-(2-(8- phenyloctyl)phenyl)propanoic Acid.

ChemInform ◽

10.1002/chin.198747167 ◽

1987 ◽

Vol 18 (47) ◽

Author(s):

J. G. GLEASON ◽

R. F. HALL ◽

C. D. PERCHONOCK ◽

K. F. ERHARD ◽

J. S. FRAZEE ◽

...

Keyword(s):

Propanoic Acid ◽

Receptor Antagonists ◽

High Affinity ◽

Leukotriene Receptor Antagonists ◽

Leukotriene Receptor

Synthesis and pharmacological characterization of [125I]MRS5127, a high affinity, selective agonist radioligand for the A3 adenosine receptor

Biochemical Pharmacology ◽

10.1016/j.bcp.2009.11.009 ◽

2010 ◽

Vol 79 (7) ◽

pp. 967-973 ◽

Cited By ~ 16

Author(s):

John A. Auchampach ◽

Elizabeth T. Gizewski ◽

Tina C. Wan ◽

Sonia de Castro ◽

Garth G. Brown ◽

...

Keyword(s):

Adenosine Receptor ◽

High Affinity ◽

Selective Agonist ◽

A3 Adenosine Receptor

Pharmacological Characterization of 2-Methyl-N-((2′-(pyrrolidin-1-ylsulfonyl)biphenyl-4-yl)methyl)propan-1-amine (PF-04455242), a High-Affinity Antagonist Selective for κ-Opioid Receptors

Journal of Pharmacology and Experimental Therapeutics ◽

10.1124/jpet.111.185108 ◽

2011 ◽

Vol 339 (2) ◽

pp. 555-566 ◽

Cited By ~ 37

Author(s):

S. Grimwood ◽

Y. Lu ◽

A. W. Schmidt ◽

M. A. Vanase-Frawley ◽

A. Sawant-Basak ◽

...

Keyword(s):

Opioid Receptors ◽

Pharmacological Characterization of Novel Opioid Receptor Ligands Aimed at Reducing the Development of Tolerance

10.33915/etd.616 ◽

2014 ◽

Author(s):

Jason Randall Healy

Keyword(s):

Opioid Receptor ◽

Receptor Ligands ◽

Opioid Receptor Ligands ◽

Development Of Tolerance

Pharmacological Characterization of 6-Bromo-3â²-nitroflavone, a Synthetic Flavonoid with High Affinity for the Benzodiazepine Receptors

Pharmacology Biochemistry and Behavior ◽

10.1016/s0091-3057(98)00088-4 ◽

1998 ◽

Vol 61 (3) ◽

pp. 239-246 ◽

Cited By ~ 14

Author(s):

C Wolfman

Keyword(s):

Benzodiazepine Receptors ◽

Pharmacological characterization of high affinity choline transporters in primary neuronal cultures in rat brain

Neuropharmacology ◽

10.1016/0028-3908(88)90100-1 ◽

1988 ◽

Vol 27 (8) ◽

pp. 837-842 ◽

Cited By ~ 7

Author(s):

M KELLEY ◽

M RAIZADA ◽

E MEYER

Keyword(s):

Rat Brain ◽

Neuronal Cultures ◽

Primary Neuronal Cultures ◽

Pharmacological characterization of benzodiazepine receptor ligands with intrinsic efficacies ranging from high to zero

Psychopharmacology ◽

10.1007/bf02253530 ◽

1993 ◽

Vol 111 (4) ◽

pp. 415-422 ◽

Cited By ~ 41

Author(s):

James R. Martin ◽

Peter Schoch ◽

François Jenck ◽

Jean-Luc Moreau ◽

Willy E. Haefely

Keyword(s):

Benzodiazepine Receptor ◽

Receptor Ligands ◽

Benzodiazepine Receptor Ligands