Identification and Characterization of a Small Molecule Antagonist of Human VPAC2 Receptor

Molecular Pharmacology ◽

10.1124/mol.109.060137 ◽

2009 ◽

Vol 77 (1) ◽

pp. 95-101 ◽

Author(s):

Alan Chu ◽

Jeremy S. Caldwell ◽

Yu Alice Chen

Keyword(s):

Small Molecule ◽

Small Molecule Antagonist ◽

Identification And Characterization

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Identification and Characterization of INCB9471, an Allosteric Noncompetitive Small-Molecule Antagonist of C-C Chemokine Receptor 5 with Potent Inhibitory Activity against Monocyte Migration and HIV-1 Infection

Journal of Pharmacology and Experimental Therapeutics ◽

10.1124/jpet.111.179531 ◽

2011 ◽

Vol 338 (1) ◽

pp. 228-239 ◽

Author(s):

Niu Shin ◽

Kim Solomon ◽

Naiming Zhou ◽

Kathy He Wang ◽

Vasudha Garlapati ◽

...

Keyword(s):

Small Molecule ◽

Chemokine Receptor ◽

Inhibitory Activity ◽

Small Molecule Antagonist ◽

Monocyte Migration ◽

Identification And Characterization ◽

Hiv 1 ◽

Potent Inhibitory Activity ◽

Chemokine Receptor 5

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Faculty Opinions recommendation of Identification and characterization of a small molecule AMPK activator that treats key components of type 2 diabetes and the metabolic syndrome.

Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature ◽

10.3410/f.1001210.377705 ◽

2006 ◽

Author(s):

Steve Rattigan

Keyword(s):

Type 2 Diabetes ◽

Metabolic Syndrome ◽

Small Molecule ◽

The Metabolic Syndrome ◽

Identification And Characterization

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Faculty Opinions recommendation of Identification and characterization of a small molecule AMPK activator that treats key components of type 2 diabetes and the metabolic syndrome.

Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature ◽

10.3410/f.1001210.374806 ◽

2006 ◽

Author(s):

Bruce Kemp

Keyword(s):

Type 2 Diabetes ◽

Metabolic Syndrome ◽

Small Molecule ◽

The Metabolic Syndrome ◽

Identification And Characterization

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Faculty Opinions recommendation of Identification and characterization of a small molecule inhibitor of formin-mediated actin assembly.

Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature ◽

10.3410/f.1283961.751061 ◽

2009 ◽

Author(s):

Marie-France Carlier

Keyword(s):

Small Molecule ◽

Small Molecule Inhibitor ◽

Actin Assembly ◽

Molecule Inhibitor ◽

Identification And Characterization

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Identification and characterization of a novel small molecule agonist of lipoprotein lipase by random screening (654.12)

The FASEB Journal ◽

10.1096/fasebj.28.1_supplement.654.12 ◽

2014 ◽

Vol 28 (S1) ◽

Author(s):

Prabodh Sadana ◽

Danielle Aring ◽

Jamie Burke ◽

Werner Geldenhuys

Keyword(s):

Lipoprotein Lipase ◽

Small Molecule ◽

Identification And Characterization ◽

Random Screening

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Identification and characterization of benzo[d]oxazol-2(3H)-one derivatives as the first potent and selective small-molecule inhibitors of chromodomain protein CDYL

European Journal of Medicinal Chemistry ◽

10.1016/j.ejmech.2019.111656 ◽

2019 ◽

Vol 182 ◽

pp. 111656 ◽

Author(s):

Lixin Yang ◽

Yongqing Liu ◽

Minghua Fan ◽

Guiwang Zhu ◽

Hongwei Jin ◽

...

Keyword(s):

Small Molecule ◽

Small Molecule Inhibitors ◽

Identification And Characterization

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Identification and Characterization of JAK2 Pseudokinase Domain Small Molecule Binders

ACS Medicinal Chemistry Letters ◽

10.1021/acsmedchemlett.7b00153 ◽

2017 ◽

Vol 8 (6) ◽

pp. 618-621 ◽

Author(s):

David E. Puleo ◽

Kaury Kucera ◽

Henrik M. Hammarén ◽

Daniela Ungureanu ◽

Ana S. Newton ◽

...

Keyword(s):

Small Molecule ◽

Identification And Characterization

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Identification and Characterization of Small-Molecule Inhibitors of Lysine Acetyltransferases

Methods in Molecular Biology - Cancer Epigenetics ◽

10.1007/978-1-4939-1804-1_28 ◽

2014 ◽

pp. 539-548

Author(s):

Daiqing Liao

Keyword(s):

Small Molecule ◽

Small Molecule Inhibitors ◽

Identification And Characterization

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Abstract 1378: Identification and characterization of small molecule inhibitors targeting Eya phosphatase activity for anti-breast cancer therapy

10.1158/1538-7445.am2011-1378 ◽

2011 ◽

Author(s):

Aaron Krueger ◽

Seameen Dehdashti ◽

Noel Southhall ◽

Samarjit Patnaik ◽

Juan Marugan ◽

...

Keyword(s):

Breast Cancer ◽

Cancer Therapy ◽

Phosphatase Activity ◽

Small Molecule ◽

Small Molecule Inhibitors ◽

Breast Cancer Therapy ◽

Identification And Characterization

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Abstract 1377: Identification and characterization of small molecule inhibitors of the activator protein-1 pathway

10.1158/1538-7445.am2011-1377 ◽

2011 ◽

Author(s):

Nicole R. Miller ◽

Ruili Huang ◽

Menghang Xia

Keyword(s):

Small Molecule ◽

Small Molecule Inhibitors ◽

Activator Protein 1 ◽

Activator Protein ◽

Identification And Characterization

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