Pharmacokinetics of synthadotin (ILX651), a novel tubulin polymerization inhibitor, in patients with solid tumors

Journal of Clinical Oncology ◽

10.1200/jco.2004.22.14_suppl.2082 ◽

2004 ◽

Vol 22 (14_suppl) ◽

pp. 2082-2082

Author(s):

P. Bonate ◽

S. Ebbinghaus ◽

J. P. Eder ◽

A. Mita ◽

E. Rubin ◽

...

Keyword(s):

Solid Tumors ◽

Tubulin Polymerization ◽

Polymerization Inhibitor ◽

Tubulin Polymerization Inhibitor

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Tisotumab vedotin. Antibody-drug conjugate directed to tissue factor, Tubulin polymerization inhibitor, Treatment of solid tumors

Drugs of the Future ◽

10.1358/dof.2020.45.10.3168441 ◽

2020 ◽

Vol 45 (10) ◽

pp. 717

Author(s):

G. D'Alessandro ◽

F. Barra ◽

A. Boutros ◽

G. Evangelisti ◽

L. Ferro Desideri ◽

...

Keyword(s):

Tissue Factor ◽

Solid Tumors ◽

Tubulin Polymerization ◽

Antibody Drug Conjugate ◽

Drug Conjugate ◽

Polymerization Inhibitor ◽

Tubulin Polymerization Inhibitor ◽

Inhibitor Treatment ◽

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Pharmacokinetics of synthadotin (ILX651), a novel tubulin polymerization inhibitor, in patients with solid tumors

Journal of Clinical Oncology ◽

10.1200/jco.2004.22.90140.2082 ◽

2004 ◽

Vol 22 (14_suppl) ◽

pp. 2082-2082

Author(s):

P. Bonate ◽

S. Ebbinghaus ◽

J. P. Eder ◽

A. Mita ◽

E. Rubin ◽

...

Keyword(s):

Solid Tumors ◽

Tubulin Polymerization ◽

Polymerization Inhibitor ◽

Tubulin Polymerization Inhibitor

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Identification of CKD-516: A Potent Tubulin Polymerization Inhibitor with Marked Antitumor Activity against Murine and Human Solid Tumors

Journal of Medicinal Chemistry ◽

10.1021/jm1002414 ◽

2010 ◽

Vol 53 (17) ◽

pp. 6337-6354 ◽

Author(s):

Jaekwang Lee ◽

Soo Jin Kim ◽

Hojin Choi ◽

Young Hoon Kim ◽

In Taek Lim ◽

...

Keyword(s):

Antitumor Activity ◽

Solid Tumors ◽

Tubulin Polymerization ◽

Polymerization Inhibitor ◽

Human Solid Tumors ◽

Tubulin Polymerization Inhibitor

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Discovery of oxyepiberberine as a novel tubulin polymerization inhibitor and an anti-colon cancer agent against LS-1034 cells

Investigational New Drugs ◽

10.1007/s10637-020-01006-0 ◽

2020 ◽

Author(s):

Hanbing Ning ◽

Wenquan Lu ◽

Qiaoyu Jia ◽

Jingyun Wang ◽

Tingting Yao ◽

...

Keyword(s):

Colon Cancer ◽

Tubulin Polymerization ◽

Polymerization Inhibitor ◽

Cancer Agent ◽

Tubulin Polymerization Inhibitor

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Redox‐responsive glycosylated combretastatin A‐4 derivative as novel tubulin polymerization inhibitor for glioma and drug delivery

Drug Development Research ◽

10.1002/ddr.21889 ◽

2021 ◽

Author(s):

Yi Zhao ◽

Ze Zhao ◽

Yamin Cui ◽

Xing Chen ◽

Changqing Chen ◽

...

Keyword(s):

Drug Delivery ◽

Tubulin Polymerization ◽

Polymerization Inhibitor ◽

Redox Responsive ◽

Tubulin Polymerization Inhibitor

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Abstract 2498: BNC105 is a tubulin polymerization inhibitor that exhibits vascular disruptive activity in renal cancer and causes upregulation in HIF1alpha, HIF2alpha and mTOR

10.1158/1538-7445.am10-2498 ◽

2010 ◽

Author(s):

Annabell F. Leske ◽

Donna M. Beaumont ◽

Tina C. Lavranos ◽

Jelena Gasic ◽

Carolyn J. Coles ◽

...

Keyword(s):

Renal Cancer ◽

Tubulin Polymerization ◽

Polymerization Inhibitor ◽

Tubulin Polymerization Inhibitor

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Abstract 4425: Oral efficacy and preclinical ADME evaluation of CKD-516, a novel tubulin polymerization inhibitor

10.1158/1538-7445.am10-4425 ◽

2010 ◽

Author(s):

Soo Jin Kim ◽

Se-Mi Kim ◽

Jae-Hoon Choi ◽

Do Hyung Lee ◽

Dong Wook Lee ◽

...

Keyword(s):

Tubulin Polymerization ◽

Polymerization Inhibitor ◽

Tubulin Polymerization Inhibitor

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Polymorphs, co-crystal structure and pharmacodynamics study of MBRI-001, a deuterium-substituted plinabulin derivative as a tubulin polymerization inhibitor

Bioorganic & Medicinal Chemistry ◽

10.1016/j.bmc.2019.03.035 ◽

2019 ◽

Vol 27 (9) ◽

pp. 1836-1844 ◽

Author(s):

Mingxu Ma ◽

Zhongpeng Ding ◽

Shixiao Wang ◽

Lingling Ma ◽

Yuxi Wang ◽

...

Keyword(s):

Crystal Structure ◽

Tubulin Polymerization ◽

Polymerization Inhibitor ◽

Tubulin Polymerization Inhibitor

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A new tubulin polymerization inhibitor, auristatin PE, induces tumor regression in a human Waldenstrom's macroglobulinemia xenograft model.

International Journal of Oncology ◽

10.3892/ijo.15.2.367 ◽

1999 ◽

Author(s):

R M Mohammad ◽

C Limvarapuss ◽

N R Wall ◽

N Hamdy ◽

F W Beck ◽

...

Keyword(s):

Tumor Regression ◽

Xenograft Model ◽

Tubulin Polymerization ◽

Waldenström’S Macroglobulinemia ◽

Polymerization Inhibitor ◽

Waldenstrom's Macroglobulinemia ◽

Waldenstrom’S Macroglobulinemia ◽

Tubulin Polymerization Inhibitor ◽

Waldenström's Macroglobulinemia

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Tubulin Polymerization Inhibitor VERU-111

10.32388/ghdryw ◽

2020 ◽

Author(s):

Keyword(s):

Tubulin Polymerization ◽

Polymerization Inhibitor ◽

Tubulin Polymerization Inhibitor

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