ChemInform Abstract: Synthesis of Prolyl Endopeptidase Inhibitors and Evaluation of Their Structure-Activity Relationships: in vitro Inhibition of Prolyl Endopeptidase from Canine Brain.

H. ARAI; H. NISHIOKA; S. NIWA; T. YAMANAKA; Y. TANAKA; K. YOSHINAGA; N. KOBAYASHI; N. MIURA; Y. IKEDA

doi:10.1002/chin.199421142

ChemInform Abstract: Synthesis of Prolyl Endopeptidase Inhibitors and Evaluation of Their Structure-Activity Relationships: in vitro Inhibition of Prolyl Endopeptidase from Canine Brain.

ChemInform ◽

10.1002/chin.199421142 ◽

2010 ◽

Vol 25 (21) ◽

pp. no-no

Author(s):

H. ARAI ◽

H. NISHIOKA ◽

S. NIWA ◽

T. YAMANAKA ◽

Y. TANAKA ◽

...

Keyword(s):

Prolyl Endopeptidase ◽

Structure Activity Relationships ◽

Structure Activity ◽

Canine Brain ◽

In Vitro Inhibition

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Synthesis of Prolyl Endopeptidase Inhibitors and Evaluation of Their Structure-Activity Relationships: In Vitro Inhibition of Prolyl Endopeptidase from Canine Brain.

Chemical and Pharmaceutical Bulletin ◽

10.1248/cpb.41.1583 ◽

1993 ◽

Vol 41 (9) ◽

pp. 1583-1588 ◽

Cited By ~ 17

Author(s):

Heihachiro ARAI ◽

Hiroyasu NISHIOKA ◽

Seiichi NIWA ◽

Takeshi YAMANAKA ◽

Yoshiaki TANAKA ◽

...

Keyword(s):

Prolyl Endopeptidase ◽

Structure Activity Relationships ◽

Structure Activity ◽

Canine Brain ◽

In Vitro Inhibition

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In vitro inhibition effects on erythrocyte carbonic anhydrase I and II and structure–activity relationships of cumarylthiazole derivatives

Биоорганическая химия ◽

10.7868/s0132342316050043 ◽

2016 ◽

Vol 42 (5) ◽

pp. 561-566

Author(s):

Belma Z. Kurt ◽

Fatih Sonmez ◽

Basak Gokce ◽

Adem Ergun ◽

Nahit Gencer ◽

...

Keyword(s):

Carbonic Anhydrase ◽

Structure Activity Relationships ◽

Structure Activity ◽

Carbonic Anhydrase I ◽

In Vitro Inhibition ◽

Erythrocyte Carbonic Anhydrase

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In vitro inhibition effect and structure–activity relationships of some saccharin derivatives on erythrocyte carbonic anhydrase I and II

Journal of Enzyme Inhibition and Medicinal Chemistry ◽

10.3109/14756366.2012.757222 ◽

2013 ◽

Vol 29 (1) ◽

pp. 118-123 ◽

Cited By ~ 13

Author(s):

Fatih Sonmez ◽

Cigdem Bilen ◽

Sinem Sumersan ◽

Nahit Gencer ◽

Semra Isik ◽

...

Keyword(s):

Carbonic Anhydrase ◽

Inhibition Effect ◽

Structure Activity Relationships ◽

Structure Activity ◽

Carbonic Anhydrase I ◽

In Vitro Inhibition ◽

Erythrocyte Carbonic Anhydrase

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In vitro inhibition effects on erythrocyte carbonic anhydrase I and II and structure-activity relationships of cumarylthiazole derivatives

Russian Journal of Bioorganic Chemistry ◽

10.1134/s1068162016050046 ◽

2016 ◽

Vol 42 (5) ◽

pp. 506-511 ◽

Cited By ~ 7

Author(s):

Belma Z. Kurt ◽

Fatih Sonmez ◽

Basak Gokce ◽

Adem Ergun ◽

Nahit Gencer ◽

...

Keyword(s):

Carbonic Anhydrase ◽

Structure Activity Relationships ◽

Structure Activity ◽

Carbonic Anhydrase I ◽

In Vitro Inhibition ◽

Erythrocyte Carbonic Anhydrase

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Tyrosine Kinase Inhibitors. 4. Structure-Activity Relationships among N- and 3-Substituted 2,2'-Dithiobis(1H-indoles) for in vitro Inhibition of Receptor and Nonreceptor Protein Tyrosine Kinases

Journal of Medicinal Chemistry ◽

10.1021/jm00001a011 ◽

1995 ◽

Vol 38 (1) ◽

pp. 58-67 ◽

Cited By ~ 47

Author(s):

Brian D. Palmer ◽

Gordon W. Rewcastle ◽

Andrew M. Thompson ◽

Maruta Boyd ◽

H. D. Hollis Showalter ◽

...

Keyword(s):

Tyrosine Kinase ◽

Tyrosine Kinase Inhibitors ◽

Tyrosine Kinases ◽

Kinase Inhibitors ◽

Protein Tyrosine Kinases ◽

Structure Activity Relationships ◽

Structure Activity ◽

In Vitro Inhibition ◽

Nonreceptor Protein Tyrosine Kinases

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In vitro inhibition of liver forms of the rodent malaria parasite Plasmodium berghei by naphthylisoquinoline alkaloids - structure-activity relationships of dioncophyllines A and C and ancistrocladine

Parasitology Research ◽

10.1007/s004360050318 ◽

1997 ◽

Vol 83 (7) ◽

pp. 673-679 ◽

Cited By ~ 17

Author(s):

Guido François ◽

Georges Timperman ◽

Tania Steenackers ◽

Laurent Aké Assi ◽

Jörg Holenz ◽

...

Keyword(s):

Plasmodium Berghei ◽

Malaria Parasite ◽

Rodent Malaria Parasite ◽

Rodent Malaria ◽

Structure Activity Relationships ◽

Structure Activity ◽

Naphthylisoquinoline Alkaloids ◽

Parasite Plasmodium ◽

In Vitro Inhibition

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In vitro inhibition of mouse epidermal cell lipoxygenase by flavonoids: structure—activity relationships

Carcinogenesis ◽

10.1093/carcin/7.1.33 ◽

1986 ◽

Vol 7 (1) ◽

pp. 33-36 ◽

Cited By ~ 19

Author(s):

Edward L. Wheeler ◽

David L. Berry

Keyword(s):

Epidermal Cell ◽

Structure Activity Relationships ◽

Structure Activity ◽

In Vitro Inhibition ◽

Mouse Epidermal Cell

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Synthesis and structure-activity relationships of pyrimidine derivatives as potent and orally active FGFR3 inhibitors with both increased systemic exposure and enhanced in vitro potency

Bioorganic & Medicinal Chemistry ◽

10.1016/j.bmc.2021.116019 ◽

2021 ◽

Vol 33 ◽

pp. 116019

Author(s):

Ikumi Kuriwaki ◽

Minoru Kameda ◽

Kazuhiko Iikubo ◽

Hiroyuki Hisamichi ◽

Yuichiro Kawamoto ◽

...

Keyword(s):

Systemic Exposure ◽

Pyrimidine Derivatives ◽

Structure Activity Relationships ◽

Structure Activity ◽

Orally Active

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Aqua mediated synthesis of 2-amino-6-benzothiazol-2-ylsulfanyl-chromenes and its in vitro study, explanation of the structure–activity relationships (SARs) as antibacterial agent

European Journal of Medicinal Chemistry ◽

10.1016/j.ejmech.2010.08.010 ◽

2010 ◽

Vol 45 (11) ◽

pp. 5031-5038 ◽

Cited By ~ 21

Author(s):

Mazaahir Kidwai ◽

Roona Poddar ◽

Saurav Bhardwaj ◽

Satendra Singh ◽

Pratibha Mehta Luthra

Keyword(s):

Antibacterial Agent ◽

In Vitro Study ◽

Vitro Study ◽

Structure Activity Relationships ◽

Structure Activity

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Structure-activity relationships of steroids in inducing germinal vesicle breakdown of Atlantic croaker oocytes in vitro

General and Comparative Endocrinology ◽

10.1016/0016-6480(88)90259-6 ◽

1988 ◽

Vol 71 (2) ◽

pp. 307-317 ◽

Cited By ~ 72

Author(s):

John M. Trant ◽

Peter Thomas

Keyword(s):

Germinal Vesicle ◽

Atlantic Croaker ◽

Germinal Vesicle Breakdown ◽

Structure Activity Relationships ◽

Structure Activity

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