Rational Design, Synthesis and Evaluation of Coumarin Derivatives as Protein-protein Interaction Inhibitors

2016 ◽  
Vol 35 (8-9) ◽  
pp. 460-473 ◽  
Author(s):  
Laura De Luca ◽  
Fatima E. Agharbaoui ◽  
Rosaria Gitto ◽  
Maria Rosa Buemi ◽  
Frauke Christ ◽  
...  
Keyword(s):  
Protein Interaction ◽  
Rational Design ◽  
Coumarin Derivatives ◽  
Design Synthesis ◽  
Protein Protein Interaction

scholarly journals Correction: Rational design of a stapled JAZ9 peptide inhibiting protein–protein interaction of a plant transcription factor

2021 ◽  
Author(s):  
Kaho Suzuki ◽  
Yousuke Takaoka ◽  
Minoru Ueda
Keyword(s):  
Transcription Factor ◽  
Protein Interaction ◽  
Rational Design ◽  
Protein Protein Interaction ◽  
Inhibiting Protein

Correction for ‘Rational design of a stapled JAZ9 peptide inhibiting protein–protein interaction of a plant transcription factor’ by Kaho Suzuki et al., RSC Chem. Biol., 2021, DOI: 10.1039/d0cb00204f.

scholarly journals Rational design of a stapled JAZ9 peptide inhibiting protein–protein interaction of a plant transcription factor

2021 ◽  
Author(s):  
Kaho Suzuki ◽  
Yousuke Takaoka ◽  
Minoru Ueda
Keyword(s):  
Arabidopsis Thaliana ◽  
Transcription Factor ◽  
Protein Interaction ◽  
Rational Design ◽  
Master Regulators ◽  
Jasmonate Signaling ◽  
Protein Protein Interaction ◽  
Inhibiting Protein

A rationally designed stapled JAZ peptide selectively inhibited MYCs, master-regulators of the jasmonate signaling in Arabidopsis thaliana. It is proposed as a novel chemical tool for the analysis of MYC related jasmonate signaling.

Design, synthesis and bioevaluation of inhibitors targeting HSP90-CDC37 protein-protein interaction based on a hydrophobic core

2021 ◽  
Vol 210 ◽  
pp. 112959
Author(s):  
Qiuyue Zhang ◽  
Xuexuan Wu ◽  
Jianrui Zhou ◽  
Lixiao Zhang ◽  
Xiaoli Xu ◽  
...  
Keyword(s):  
Protein Interaction ◽  
Hydrophobic Core ◽  
Design Synthesis ◽  
Protein Protein Interaction

In Silico Approaches Assisting the Rational Design of Low Molecular Weight Protein–Protein Interaction Modulators

2015 ◽  
pp. 441-482
Author(s):  
Bruno Villoutreix ◽  
Melaine Kuenemann ◽  
David Lagorce ◽  
Olivier Sperandio ◽  
Maria Miteva
Keyword(s):  
Molecular Weight ◽  
Protein Interaction ◽  
In Silico ◽  
Rational Design ◽  
Low Molecular Weight ◽  
Molecular Weight Protein ◽  
Protein Protein Interaction ◽  
Weight Protein ◽  
Low Molecular Weight Protein

scholarly journals Design, Synthesis, and Pharmacological Evaluation of Analogues Derived from the PLEV Tetrapeptide as Protein–Protein Interaction Modulators of Voltage-Gated Sodium Channel 1.6

2020 ◽  
Vol 63 (20) ◽  
pp. 11522-11547
Author(s):  
Pingyuan Wang ◽  
Paul A. Wadsworth ◽  
Nolan M. Dvorak ◽  
Aditya K. Singh ◽  
Haiying Chen ◽  
...  
Keyword(s):  
Sodium Channel ◽  
Protein Interaction ◽  
Voltage Gated Sodium Channel ◽  
Design Synthesis ◽  
Voltage Gated ◽  
Protein Protein Interaction ◽  
Pharmacological Evaluation

scholarly journals Design, synthesis, and biological evaluation of novel FAK scaffold inhibitors targeting the FAK–VEGFR3 protein–protein interaction

2014 ◽  
Vol 80 ◽  
pp. 154-166 ◽  
Author(s):  
Priyanka N. Gogate ◽  
Manivannan Ethirajan ◽  
Elena V. Kurenova ◽  
Andrew T. Magis ◽  
Ravindra K. Pandey ◽  
...  
Keyword(s):  
Protein Interaction ◽  
Biological Evaluation ◽  
Design Synthesis ◽  
Protein Protein Interaction ◽  
Synthesis And Biological Evaluation

Abstract 828: Design, synthesis and biological evaluation of peptide inhibitors of the Keap1-Nrf2 protein-protein interaction

2011 ◽  
Author(s):  
Rowena Hancock ◽  
Helene Bertrand ◽  
Shama Naz ◽  
Tadayuki Tsujita ◽  
John Hayes ◽  
...  
Keyword(s):  
Protein Interaction ◽  
Biological Evaluation ◽  
Peptide Inhibitors ◽  
Design Synthesis ◽  
Protein Protein Interaction ◽  
Synthesis And Biological Evaluation ◽  
Nrf2 Protein

Rational Design, Synthesis, Biological Evaluation, Homology and Docking Studies of Coumarin Derivatives as α1-Adrenoceptor Antagonists

2011 ◽  
Vol 8 (6) ◽  
pp. 1052-1064 ◽  
Author(s):  
Xiang Zhou ◽  
Ya-Dong Chen ◽  
Tao Wang ◽  
Xiao-Bing Wang ◽  
Ling-Yi Kong
Keyword(s):  
Rational Design ◽  
Docking Studies ◽  
Biological Evaluation ◽  
Coumarin Derivatives ◽  
Design Synthesis
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