Interaction potential of the endothelin-A receptor antagonist atrasentan with drug transporters and drug-metabolising enzymes assessed in vitro

2011 ◽  
Vol 68 (4) ◽  
pp. 1093-1098 ◽  
Author(s):  
Johanna Weiss ◽  
Walter Emil Haefeli
Keyword(s):  
Receptor Antagonist ◽  
Interaction Potential ◽  
Drug Transporters ◽  
Endothelin A Receptor ◽  
Endothelin A ◽  
Drug Metabolising Enzymes

Specific endothelin-A-receptor antagonist ZD4054 inhibits breast cancer growth in vitro and in vivo

2008 ◽  
Vol 68 (S 01) ◽  
Author(s):  
M Smollich ◽  
M Götte ◽  
J Fischgräbe ◽  
I Radke ◽  
L Macedo ◽  
...  
Keyword(s):  
Breast Cancer ◽  
Receptor Antagonist ◽  
Cancer Growth ◽  
Endothelin A Receptor ◽  
Endothelin A ◽  
Breast Cancer Growth

The Selective Endothelin-A-Receptor Antagonist LU 135.252 Inhibits the Direct Arrhythmogenic Action of Endothelin-1

2000 ◽  
Vol 36 ◽  
pp. S314-S316 ◽  
Author(s):  
Béla Merkely ◽  
Tamás Szabó ◽  
László Gellér ◽  
Orsolya Kiss ◽  
Ferenc Horkay ◽  
...  
Keyword(s):  
Receptor Antagonist ◽  
Endothelin 1 ◽  
Endothelin A Receptor ◽  
Endothelin A

scholarly journals Antifibrotic effects of ambrisentan, an endothelin-A receptor antagonist, in a non-alcoholic steatohepatitis mouse model

2016 ◽  
Vol 8 (22) ◽  
pp. 933 ◽  
Author(s):  
Toshiaki Okamoto ◽  
Masahiko Koda ◽  
Kennichi Miyoshi ◽  
Takumi Onoyama ◽  
Manabu Kishina ◽  
...  
Keyword(s):  
Mouse Model ◽  
Receptor Antagonist ◽  
Alcoholic Steatohepatitis ◽  
Endothelin A Receptor ◽  
Endothelin A

Metabolism and transporter-mediated drug–drug interactions of the endothelin-A receptor antagonist CI-1034

2006 ◽  
Vol 159 (2) ◽  
pp. 156-168 ◽  
Author(s):  
Jasminder Sahi ◽  
Michael W. Sinz ◽  
Scott Campbell ◽  
Rouchelle Mireles ◽  
Xianxian Zheng ◽  
...  
Keyword(s):  
Drug Interactions ◽  
Receptor Antagonist ◽  
Endothelin A Receptor ◽  
Endothelin A
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