Synthesis and binding properties of the fluorinated substituted benzamide [3H]NCQ 115, a new selective dopamine D2 receptor ligand

1991 ◽  
Vol 201 (1) ◽  
pp. 1-10 ◽  
Author(s):  
Håkan Hall ◽  
Thomas Högberg ◽  
Christer Halldin ◽  
Stefan Bengtsson ◽  
Ilse Wedel
Keyword(s):  
Dopamine D2 Receptor ◽  
D2 Receptor ◽  
Binding Properties ◽  
Receptor Ligand ◽  
Dopamine D2 ◽  
Substituted Benzamide ◽  
Selective Dopamine

ChemInform Abstract: New 2-Thioether-Substituted Apomorphines as Potent and Selective Dopamine D2 Receptor Agonists.

ChemInform ◽  
2011 ◽  
Vol 42 (41) ◽  
pp. no-no
Author(s):  
Reet Reinart ◽  
Zsuzsanna Gyulai ◽  
Sandor Berenyi ◽  
Sandor Antus ◽  
Argo Vonk ◽  
...  
Keyword(s):  
Dopamine D2 Receptor ◽  
D2 Receptor ◽  
Receptor Agonists ◽  
Dopamine D2 ◽  
Selective Dopamine

Cerebral kinetics of the dopamine D2 receptor ligand [123I]IBZM in mice

2008 ◽  
Vol 35 (4) ◽  
pp. 467-473 ◽  
Author(s):  
Philipp T. Meyer ◽  
Dagmar Salber ◽  
Johannes Schiefer ◽  
Markus Cremer ◽  
Wolfgang M. Schaefer ◽  
...  
Keyword(s):  
Dopamine D2 Receptor ◽  
D2 Receptor ◽  
Receptor Ligand ◽  
Dopamine D2 ◽  
Kinetics Of

SSR181507, a dopamine D2 receptor and 5-HT1A receptor ligand: Evidence for mixed anxiolytic- and antidepressant-like activities

2011 ◽  
Vol 97 (3) ◽  
pp. 428-435 ◽  
Author(s):  
Denis Boulay ◽  
Ronan Depoortere ◽  
Caroline Louis ◽  
Martine Lacave ◽  
Marie Thérèse Lucas ◽  
...  
Keyword(s):  
Dopamine D2 Receptor ◽  
D2 Receptor ◽  
Receptor Ligand ◽  
Dopamine D2

An attempt at the hydrated imidazoline ring expansion (HIRE) of diarene-fused [1,4]diazepinones delivers selective dopamine D2 receptor ligands

Synthesis ◽  
2021 ◽  
Author(s):  
Sergey Grintsevich ◽  
Alexander V. Sapegin ◽  
Andrzej Bojarski ◽  
Beata Duszyńska ◽  
Mikhail Krasavin
Keyword(s):  
Dopamine D2 Receptor ◽  
D2 Receptor ◽  
Ring Expansion ◽  
Side Chain ◽  
Receptor Ligands ◽  
Structure Activity Relationships ◽  
Dopamine D2 ◽  
Structure Activity ◽  
Imidazoline Ring ◽  
Selective Dopamine

Attempts to extend the hydrated imidazoline ring expansion (HIRE) strategy to a series of diarene-fused [1,4]diazepinones (earlier applied successfully to bis-pyrido substrate nevirapine) resulted in no ring expansion but rather 2-aminoethyl side chain expulsion. This seeming setback (setting the limitations to the HIRE methodology substrate scope) led to the discovery of selective dopamine D2 ligands with elements of structure-activity relationships.

Remoxipride, a selective dopamine D2 receptor antagonist, in tardive dyskinesia

1988 ◽  
Vol 94 (2) ◽  
Author(s):  
Ulf Andersson ◽  
Jan-Erik H�ggstr�m ◽  
Maj-Inger Nilsson ◽  
Erik Widerl�v
Keyword(s):  
Tardive Dyskinesia ◽  
Receptor Antagonist ◽  
Dopamine D2 Receptor ◽  
D2 Receptor ◽  
Dopamine D2 ◽  
Selective Dopamine ◽  
Dopamine D2 Receptor Antagonist
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