Design, synthesis and biological activity of a novel ethylenediamine derivatives as H1 receptor antagonists

2019 ◽  
Vol 27 (24) ◽  
pp. 115127
Author(s):  
Shiyang Zhou ◽  
Gangliang Huang ◽  
Guangying Chen
Keyword(s):  
Biological Activity ◽  
H1 Receptor ◽  
Receptor Antagonists ◽  
Design Synthesis ◽  
Ethylenediamine Derivatives

Design, synthesis and biological activity evaluation of desloratadine analogues as H1 receptor antagonists

2013 ◽  
Vol 21 (14) ◽  
pp. 4178-4185 ◽  
Author(s):  
Yan Lin ◽  
Yue Wang ◽  
Li-Feng Sima ◽  
Dong-Hua Wang ◽  
Xiao-Hui Cao ◽  
...  
Keyword(s):  
Biological Activity ◽  
H1 Receptor ◽  
Receptor Antagonists ◽  
Design Synthesis ◽  
Activity Evaluation

Design, synthesis and biological activity of 4′-[(benzimidazol-1-yl)methyl]biphenyl-2-sulphonamides as dual angiotensin II and endothelin A receptor antagonists

MedChemComm ◽  
2015 ◽  
Vol 6 (4) ◽  
pp. 715-718 ◽  
Author(s):  
Li-Ping Hao ◽  
Wei-Zhe Xue ◽  
Xiao-Feng Han ◽  
Xing He ◽  
Jun Zhang ◽  
...  
Keyword(s):  
Biological Activity ◽  
Angiotensin Ii ◽  
Model Simulation ◽  
Molecular Model ◽  
Pharmacophore Model ◽  
Receptor Antagonists ◽  
Design Synthesis ◽  
3D Pharmacophore ◽  
Endothelin A Receptor ◽  
Endothelin A

A series of novel 4′-[(benzimidazol-1-yl)methyl]biphenyl-2-sulphonamides was designed, and their molecular model simulation fitting to a new HipHop 3D pharmacophore model was examined.

Non-peptide angiotensin II receptor antagonists. 1. Design, synthesis, and biological activity of N-substituted indoles and dihydroindoles

1993 ◽  
Vol 36 (26) ◽  
pp. 4230-4238 ◽  
Author(s):  
Daljit S. Dhanoa ◽  
Scott W. Bagley ◽  
Raymond S. L. Chang ◽  
Victor J. Lotti ◽  
Tsing Bau Chen ◽  
...  
Keyword(s):  
Biological Activity ◽  
Angiotensin Ii ◽  
Angiotensin Ii Receptor ◽  
Angiotensin Ii Receptor Antagonists ◽  
Receptor Antagonists ◽  
Design Synthesis

scholarly journals Design, Synthesis, and Biological Activity Studies of Istradefylline Derivatives Based on Adenine as A2A Receptor Antagonists

ACS Omega ◽  
2021 ◽  
Vol 6 (6) ◽  
pp. 4386-4394
Author(s):  
Yiyun Wang ◽  
Haojie Xu ◽  
Hongyi Wang ◽  
Zhonghui Zheng ◽  
Zihui Meng ◽  
...  
Keyword(s):  
Biological Activity ◽  
Receptor Antagonists ◽  
Design Synthesis ◽  
A2a Receptor

scholarly journals Design, Synthesis and Biological Activity of Rigid Cannabinoid CB1 Receptor Antagonists

2002 ◽  
Vol 50 (8) ◽  
pp. 1109-1113 ◽  
Author(s):  
Axel Reinhard Stoit ◽  
Jos Hubertus Maria Lange ◽  
Arnold Peter den Hartog ◽  
Eric Ronken ◽  
Koos Tipker ◽  
...  
Keyword(s):  
Biological Activity ◽  
Cb1 Receptor ◽  
Cannabinoid Cb1 Receptor ◽  
Receptor Antagonists ◽  
Design Synthesis ◽  
Cb1 Receptor Antagonists

Design, Synthesis and Biological Activity of Rigid Cannabinoid CB1 Receptor Antagonists.

ChemInform ◽  
2003 ◽  
Vol 34 (3) ◽  
Author(s):  
Axel Reinhard Stoit ◽  
Jos Hubertus Maria Lange ◽  
Arnold Peter den Hartog ◽  
Eric Ronken ◽  
Koos Tipker ◽  
...  
Keyword(s):  
Biological Activity ◽  
Cb1 Receptor ◽  
Cannabinoid Cb1 Receptor ◽  
Receptor Antagonists ◽  
Design Synthesis ◽  
Cb1 Receptor Antagonists
Sign in / Sign up

Export Citation Format

Share Document