Fragment-based lead discovery of indazole-based compounds as AXL kinase inhibitors

2021 ◽  
Vol 49 ◽  
pp. 116437
Author(s):  
Pearly Shuyi Ng ◽  
Klement Foo ◽  
Sandra Sim ◽  
Gang Wang ◽  
Chuhui Huang ◽  
...  
Keyword(s):  
Kinase Inhibitors ◽  
Lead Discovery

scholarly journals Identification of “Preferred” Human Kinase Inhibitors for Sleeping Sickness Lead Discovery. Are Some Kinases Better than Others for Inhibitor Repurposing?

2016 ◽  
Vol 2 (3) ◽  
pp. 180-186 ◽  
Author(s):  
Emanuele Amata ◽  
Hualin Xi ◽  
Gonzalo Colmenarejo ◽  
Rosario Gonzalez-Diaz ◽  
Carlos Cordon-Obras ◽  
...  
Keyword(s):  
Kinase Inhibitors ◽  
Sleeping Sickness ◽  
Lead Discovery ◽  
Human Kinase ◽  
Better Than

scholarly journals First Cdc7 Kinase Inhibitors: Pyrrolopyridinones as Potent and Orally Active Antitumor Agents. 2. Lead Discovery

2009 ◽  
Vol 52 (4) ◽  
pp. 1230-1230
Author(s):  
Maria Menichincheri ◽  
Alberto Bargiotti ◽  
Jens Berthelsen ◽  
Jay A. Bertrand ◽  
Roberto Bossi ◽  
...  
Keyword(s):  
Kinase Inhibitors ◽  
Antitumor Agents ◽  
Lead Discovery ◽  
Cdc7 Kinase ◽  
Orally Active

First Cdc7 Kinase Inhibitors: Pyrrolopyridinones as Potent and Orally Active Antitumor Agents. 2. Lead Discovery†

2009 ◽  
Vol 52 (2) ◽  
pp. 293-307 ◽  
Author(s):  
Maria Menichincheri ◽  
Alberto Bargiotti ◽  
Jens Berthelsen ◽  
Jay A. Bertrand ◽  
Roberto Bossi ◽  
...  
Keyword(s):  
Kinase Inhibitors ◽  
Antitumor Agents ◽  
Lead Discovery ◽  
Cdc7 Kinase ◽  
Orally Active

Lessons learned from the optimization of natural product based kinase inhibitors through molecular calculations

Planta Medica ◽  
2008 ◽  
Vol 74 (09) ◽  
Author(s):  
V Myrianthopoulos ◽  
P Magiatis ◽  
AL Skaltsounis ◽  
L Meijer ◽  
E Mikros
Keyword(s):  
Natural Product ◽  
Kinase Inhibitors ◽  
Lessons Learned ◽  
Molecular Calculations

Signal transduction therapy of colon tumors with multiple target kinase inhibitors

2009 ◽  
Vol 47 (05) ◽  
Author(s):  
G Kéri ◽  
L Őrfi ◽  
Z Greff ◽  
Z Varga ◽  
B Szokol ◽  
...  
Keyword(s):  
Signal Transduction ◽  
Kinase Inhibitors ◽  
Multiple Target ◽  
Colon Tumors ◽  
Signal Transduction Therapy

Effects of multi-kinase inhibitors on pulmonary vascular and right ventricular remodelling

Pneumologie ◽  
2011 ◽  
Vol 65 (S 01) ◽  
Author(s):  
B Kojonazarov ◽  
A Sydykov ◽  
H Luitel ◽  
D Kosanovic ◽  
S Pullamsetti ◽  
...  
Keyword(s):  
Right Ventricular ◽  
Kinase Inhibitors ◽  
Ventricular Remodelling

Side effects of tyrosine kinase inhibitors (TKIs) on bone remodelling

2012 ◽  
Vol 224 (03) ◽  
Author(s):  
JT Tauer ◽  
A Ulmer ◽  
LC Hofbauer ◽  
M Suttorp
Keyword(s):  
Side Effects ◽  
Tyrosine Kinase ◽  
Tyrosine Kinase Inhibitors ◽  
Kinase Inhibitors ◽  
Bone Remodelling
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