Synthesis and structure–activity relationship of a novel, achiral series of TNF-α converting enzyme inhibitors

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/j.bmcl.2006.02.015 ◽

2006 ◽

Vol 16 (10) ◽

pp. 2699-2704 ◽

Author(s):

John L. Gilmore ◽

Bryan W. King ◽

Cathy Harris ◽

Thomas Maduskuie ◽

Stephen E. Mercer ◽

...

Keyword(s):

Enzyme Inhibitors ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Converting Enzyme ◽

Converting Enzyme Inhibitors ◽

Structure Activity ◽

Tnf Α ◽

Relationship Of

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Synthesis and Structure—Activity Relationship of a Novel, Achiral Series of TNF-α Converting Enzyme Inhibitors.

10.1002/chin.200633145 ◽

2006 ◽

Vol 37 (33) ◽

Author(s):

John L. Gilmore ◽

et al. et al.

Keyword(s):

Enzyme Inhibitors ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Converting Enzyme ◽

Converting Enzyme Inhibitors ◽

Structure Activity ◽

Tnf Α ◽

Relationship Of

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Synthesis and structure–activity relationship of a novel, non-hydroxamate series of TNF-α converting enzyme inhibitors

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/j.bmcl.2007.05.100 ◽

2007 ◽

Vol 17 (16) ◽

pp. 4678-4682 ◽

Author(s):

John L. Gilmore ◽

Bryan W. King ◽

Naoyuki Asakawa ◽

Kimberly Harrison ◽

Andrew Tebben ◽

...

Keyword(s):

Enzyme Inhibitors ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Converting Enzyme ◽

Converting Enzyme Inhibitors ◽

Structure Activity ◽

Tnf Α ◽

Relationship Of

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Synthesis and structure–activity relationship of a novel sulfone series of TNF-α converting enzyme inhibitors

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/j.bmcl.2004.06.049 ◽

2004 ◽

Vol 14 (17) ◽

pp. 4453-4459 ◽

Author(s):

Chu-Biao Xue ◽

Xiao-Tao Chen ◽

Xiaohua He ◽

John Roderick ◽

Ronald L. Corbett ◽

...

Keyword(s):

Enzyme Inhibitors ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Converting Enzyme ◽

Converting Enzyme Inhibitors ◽

Structure Activity ◽

Tnf Α ◽

Relationship Of

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Synthesis and Structure—Activity Relationship of a Novel Sulfone Series of TNF-α Converting Enzyme Inhibitors.

10.1002/chin.200452094 ◽

2004 ◽

Vol 35 (52) ◽

Author(s):

Chu-Biao Xue ◽

Xiao-Tao Chen ◽

et al. et al.

Keyword(s):

Enzyme Inhibitors ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Converting Enzyme ◽

Converting Enzyme Inhibitors ◽

Structure Activity ◽

Tnf Α ◽

Relationship Of

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Structure–activity relationship study between Ornithyl-Proline and Lysyl-Proline based tripeptidomimics as angiotensin-converting enzyme inhibitors

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/j.bmcl.2006.01.061 ◽

2006 ◽

Vol 16 (8) ◽

pp. 2117-2121 ◽

Author(s):

Mahesh Chand Pavar ◽

Kashif Hanif ◽

Amir Azam ◽

Sneh lata ◽

M.A. Qadar Pasha ◽

...

Keyword(s):

Angiotensin Converting Enzyme ◽

Enzyme Inhibitors ◽

Angiotensin Converting Enzyme Inhibitors ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Converting Enzyme ◽

Converting Enzyme Inhibitors ◽

Structure Activity ◽

Relationship Study

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Discovery and structure–activity relationship of coumarin derivatives as TNF-α inhibitors

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/j.bmcl.2004.03.022 ◽

2004 ◽

Vol 14 (10) ◽

pp. 2411-2415 ◽

Author(s):

Jie-Fei Cheng ◽

Mi Chen ◽

David Wallace ◽

Sovouthy Tith ◽

Thomas Arrhenius ◽

...

Keyword(s):

Structure Activity Relationship ◽

Activity Relationship ◽

Coumarin Derivatives ◽

Structure Activity ◽

Tnf Α ◽

Relationship Of

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Rational Design, Synthesis and Structure—Activity Relationships of a Cyclic Succinate Series of TNF-α Converting Enzyme Inhibitors. Part 1. Lead Identification.

10.1002/chin.200414160 ◽

2004 ◽

Vol 35 (14) ◽

Author(s):

Chu-Biao Xue ◽

et al. et al.

Keyword(s):

Rational Design ◽

Enzyme Inhibitors ◽

Converting Enzyme ◽

Converting Enzyme Inhibitors ◽

Design Synthesis ◽

Structure Activity Relationships ◽

Structure Activity ◽

Tnf Α ◽

Lead Identification

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Structure–Activity Relationship of Plesiomonas shigelloides Lipid A to the Production of TNF-α, IL-1β, and IL-6 by Human and Murine Macrophages

Frontiers in Immunology ◽

10.3389/fimmu.2017.01741 ◽

2017 ◽

Vol 8 ◽

Author(s):

Marta Kaszowska ◽

Marta Wojcik ◽

Jakub Siednienko ◽

Czeslaw Lugowski ◽

Jolanta Lukasiewicz

Keyword(s):

Lipid A ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Plesiomonas Shigelloides ◽

Murine Macrophages ◽

Structure Activity ◽

Tnf Α ◽

Relationship Of

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Rational Design, Synthesis and Structure—Activity Relationships of a Cyclic Succinate Series of TNF-α Converting Enzyme Inhibitors. Part 2. Lead Optimization.

10.1002/chin.200414161 ◽

2004 ◽

Vol 35 (14) ◽

Author(s):

Chu-Biao Xue ◽

et al. et al.

Keyword(s):

Rational Design ◽

Enzyme Inhibitors ◽

Lead Optimization ◽

Converting Enzyme ◽

Converting Enzyme Inhibitors ◽

Design Synthesis ◽

Structure Activity Relationships ◽

Structure Activity ◽

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Advancement and prospects of production, transport, functional activity and structure-activity relationship of food-derived angiotensin converting enzyme (ACE) inhibitory peptides

Critical Reviews in Food Science and Nutrition ◽

10.1080/10408398.2021.1964433 ◽

2021 ◽

pp. 1-27

Author(s):

Lu Xiang ◽

Zhichang Qiu ◽

Renjie Zhao ◽

Zhenjia Zheng ◽

Xuguang Qiao

Keyword(s):

Angiotensin Converting Enzyme ◽

Functional Activity ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Converting Enzyme ◽

Inhibitory Peptides ◽

Structure Activity ◽

Ace Inhibitory Peptides ◽

Relationship Of ◽

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