Design, synthesis and biological evaluation of α-substituted isonipecotic acid benzothiazole analogues as potent bacterial type II topoisomerase inhibitors

2013 ◽  
Vol 23 (24) ◽  
pp. 6598-6603 ◽  
Author(s):  
Lorraine C. Axford ◽  
Piyush K. Agarwal ◽  
Kelly H. Anderson ◽  
Laura N. Andrau ◽  
John Atherall ◽  
...  
Keyword(s):  
Biological Evaluation ◽  
Type Ii ◽  
Topoisomerase Inhibitors ◽  
Design Synthesis ◽  
Isonipecotic Acid ◽  
Synthesis And Biological Evaluation ◽  
Bacterial Type

Design, synthesis and biological evaluation of type-II VEGFR-2 inhibitors based on quinoxaline scaffold

2014 ◽  
Vol 56 ◽  
pp. 16-26 ◽  
Author(s):  
Mai I. Shahin ◽  
Dalal A. Abou El Ella ◽  
Nasser S.M. Ismail ◽  
Khaled A.M. Abouzid
Keyword(s):  
Biological Evaluation ◽  
Type Ii ◽  
Design Synthesis ◽  
Synthesis And Biological Evaluation

Design, synthesis and biological evaluation of new oligopyrrole carboxamides linked with tricyclic DNA-intercalators as potential DNA ligands or topoisomerase inhibitors

2007 ◽  
Vol 42 (6) ◽  
pp. 752-771 ◽  
Author(s):  
Marie-Hélène David-Cordonnier ◽  
Marie-Paule Hildebrand ◽  
Brigitte Baldeyrou ◽  
Amelie Lansiaux ◽  
Christoph Keuser ◽  
...  
Keyword(s):  
Biological Evaluation ◽  
Topoisomerase Inhibitors ◽  
Design Synthesis ◽  
Dna Intercalators ◽  
Synthesis And Biological Evaluation

Design, Synthesis and Biological Evaluation of New 5‐(2‐Nitrophenyl)‐1‐aryl‐1 H ‐pyrazoles as Topoisomerase Inhibitors

2021 ◽  
Vol 6 (26) ◽  
pp. 6644-6651
Author(s):  
Manpreet Kaur ◽  
Vikrant Mehta ◽  
Sahil Arora ◽  
Anjana Munshi ◽  
Sandeep Singh ◽  
...  
Keyword(s):  
Biological Evaluation ◽  
Topoisomerase Inhibitors ◽  
Design Synthesis ◽  
Synthesis And Biological Evaluation

scholarly journals Rational Design, Synthesis and Biological Evaluation of Pyrimidine-4,6-diamine derivatives as Type-II inhibitors of FLT3 Selective Against c-KIT

2018 ◽  
Vol 8 (1) ◽  
Author(s):  
Jaideep B. Bharate ◽  
Nicholas McConnell ◽  
Gunaganti Naresh ◽  
Lingtian Zhang ◽  
Naga Rajiv Lakkaniga ◽  
...  
Keyword(s):  
Rational Design ◽  
Biological Evaluation ◽  
Type Ii ◽  
Design Synthesis ◽  
Synthesis And Biological Evaluation

Design, Synthesis and Biological Evaluation of Hybrid Molecules Containing Conjugated Styryl Ketone and α-Bromoacryloyl Moieties

2012 ◽  
Vol 9 (2) ◽  
pp. 140-152 ◽  
Author(s):  
Romeo Romagnoli ◽  
Pier Giovanni Baraldi ◽  
Olga Cruz-Lopez ◽  
Maria Kimatrai Salvador ◽  
Delia Preti ◽  
...  
Keyword(s):  
Biological Evaluation ◽  
Design Synthesis ◽  
Hybrid Molecules ◽  
Synthesis And Biological Evaluation
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