“Methylene Bridge” to 5-HT3 Receptor Antagonists: Conformationally Constrained Phenylguanidines

2018 ◽  
Vol 10 (3) ◽  
pp. 1380-1389 ◽  
Author(s):  
Ahmed S. Abdelkhalek ◽  
Genevieve S. Alley ◽  
Osama I. Alwassil ◽  
Shailesh Khatri ◽  
Philip D. Mosier ◽  
...  
Keyword(s):  
Receptor Antagonists ◽  
Methylene Bridge ◽  
Conformationally Constrained

Synthesis of Benzobicyclo[2.2.1]heptylimidazoles as Conformationally Constrained Adrenergic Receptor Antagonists

Heterocycles ◽  
2005 ◽  
Vol 65 (11) ◽  
pp. 2783 ◽  
Author(s):  
Jari Yli-Kauhaluoma ◽  
Aki Laine ◽  
Jari Ratilainen ◽  
Arto Karjalainen
Keyword(s):  
Adrenergic Receptor ◽  
Receptor Antagonists ◽  
Conformationally Constrained

Design and synthesis of conformationally constrained N,N-disubstituted 1,4-diazepanes as potent orexin receptor antagonists

2010 ◽  
Vol 20 (7) ◽  
pp. 2311-2315 ◽  
Author(s):  
Paul J. Coleman ◽  
John D. Schreier ◽  
Georgia B. McGaughey ◽  
Michael J. Bogusky ◽  
Christopher D. Cox ◽  
...  
Keyword(s):  
Receptor Antagonists ◽  
Conformationally Constrained ◽  
Design And Synthesis

CCK2 receptor antagonists containing the conformationally constrained phenylalanine derivatives, including the new amino acid Xic

2002 ◽  
Vol 37 (5) ◽  
pp. 379-389 ◽  
Author(s):  
Susan E Gibson (née Thomas) ◽  
Nathalie Guillo ◽  
Jerome O Jones ◽  
Ildiko M Buck ◽  
S.Barret Kalindjian ◽  
...  
Keyword(s):  
Amino Acid ◽  
Receptor Antagonists ◽  
Conformationally Constrained ◽  
Cck2 Receptor

6-Substituted decahydroisoquinoline-3-carboxylic acids as potent and selective conformationally constrained NMDA receptor antagonists

1992 ◽  
Vol 35 (19) ◽  
pp. 3547-3560 ◽  
Author(s):  
Paul L. Ornstein ◽  
Darryle D. Schoepp ◽  
M. Brian Arnold ◽  
Nancy K. Augenstein ◽  
David Lodge ◽  
...  
Keyword(s):  
Nmda Receptor ◽  
Carboxylic Acids ◽  
Nmda Receptor Antagonists ◽  
Receptor Antagonists ◽  
Conformationally Constrained

Conformationally constrained N1-arylsulfonyltryptamine derivatives as 5-HT6 receptor antagonists

2005 ◽  
Vol 15 (21) ◽  
pp. 4780-4785 ◽  
Author(s):  
Derek C. Cole ◽  
William J. Lennox ◽  
Joseph R. Stock ◽  
John W. Ellingboe ◽  
Hossein Mazandarani ◽  
...  
Keyword(s):  
Receptor Antagonists ◽  
Conformationally Constrained

ChemInform Abstract: CCK2 Receptor Antagonists Containing the Conformationally Constrained Phenylalanine Derivatives, Including the New Amino Acid Xic.

ChemInform ◽  
2010 ◽  
Vol 33 (44) ◽  
pp. no-no
Author(s):  
Susan E. Gibson ◽  
Nathalie Guillo ◽  
Jerome O. Jones ◽  
Ildiko M. Buck ◽  
S. Barret Kalindjian ◽  
...  
Keyword(s):  
Amino Acid ◽  
Receptor Antagonists ◽  
Conformationally Constrained ◽  
Cck2 Receptor

Comparison of the central nervous system effects produced by six H1-receptor antagonists

1996 ◽  
Vol 26 (9) ◽  
pp. 1092-1097 ◽  
Author(s):  
F. E. R. SIMONS ◽  
T. G. FRASER ◽  
J. D. REGGIN ◽  
K. J. SIMONS
Keyword(s):  
Central Nervous System ◽  
Nervous System ◽  
H1 Receptor ◽  
Receptor Antagonists ◽  
The Central Nervous System
Sign in / Sign up

Export Citation Format

Share Document