Synthesis and Biological Evaluation of Water-Soluble 2-Boronoethylthio Compounds

Journal of Medicinal Chemistry ◽

10.1021/jm00335a016 ◽

1964 ◽

Vol 7 (5) ◽

pp. 640-643 ◽

Author(s):

D. S. Matteson ◽

A. H. Soloway ◽

D. W. Tomlinson ◽

J. D. Campbell ◽

G. A. Nixon

Keyword(s):

Biological Evaluation ◽

Water Soluble ◽

Synthesis And Biological Evaluation

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Abstract 284: Design, synthesis and biological evaluation of novel water-soluble salts of the antimitotic prodrugs 4-(3-alkyl-2-oxoimidazolidin-1-yl)-N-phenylbenzenesulfonamides selectively bioactivated by cytochrome p450 1A1 in breast cancer cells

10.1158/1538-7445.am2021-284 ◽

2021 ◽

Author(s):

Vincent Ouellette ◽

Atziri Corin Chavez Alvarez ◽

Sébastien Fortin

Keyword(s):

Breast Cancer ◽

Cytochrome P450 ◽

Cancer Cells ◽

Breast Cancer Cells ◽

Biological Evaluation ◽

Water Soluble ◽

Soluble Salts ◽

Cytochrome P450 1A1 ◽

Design Synthesis ◽

Synthesis And Biological Evaluation

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Design, synthesis and biological evaluation of water-soluble per-O-methylated cyclodextrin-C60 conjugates as anti-influenza virus agents

European Journal of Medicinal Chemistry ◽

10.1016/j.ejmech.2018.01.040 ◽

2018 ◽

Vol 146 ◽

pp. 194-205 ◽

Author(s):

Xiaolei Zhu ◽

Sulong Xiao ◽

Demin Zhou ◽

Matthieu Sollogoub ◽

Yongmin Zhang

Keyword(s):

Influenza Virus ◽

Biological Evaluation ◽

Water Soluble ◽

Design Synthesis ◽

Methylated Cyclodextrin ◽

Synthesis And Biological Evaluation

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Water Soluble Coumarin Quaternary Ammonium Chlorides: Synthesis and Biological Evaluation

Chemistry & Biodiversity ◽

10.1002/cbdv.202000258 ◽

2020 ◽

Author(s):

Mert O. Karataş ◽

Samir A. A. Noma ◽

Canbolat Gürses ◽

Sevgi Balcıoğlu ◽

Burhan Ateş ◽

...

Keyword(s):

Quaternary Ammonium ◽

Biological Evaluation ◽

Water Soluble ◽

Synthesis And Biological Evaluation

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Design, synthesis, and biological evaluation of novel water-soluble triptolide derivatives: Antineoplastic activity against imatinib-resistant CML cells bearing T315I mutant Bcr-Abl

Bioorganic & Medicinal Chemistry ◽

10.1016/j.bmc.2010.01.052 ◽

2010 ◽

Vol 18 (5) ◽

pp. 1806-1815 ◽

Author(s):

Fang Xu ◽

Xianping Shi ◽

Shichang Li ◽

Jieshun Cui ◽

Zhongzheng Lu ◽

...

Keyword(s):

Biological Evaluation ◽

Water Soluble ◽

Antineoplastic Activity ◽

Design Synthesis ◽

Imatinib Resistant ◽

Synthesis And Biological Evaluation

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Synthesis and biological evaluation of new water-soluble photoactive chlorin conjugate for targeted delivery

European Journal of Medicinal Chemistry ◽

10.1016/j.ejmech.2017.12.062 ◽

2018 ◽

Vol 144 ◽

pp. 740-750 ◽

Author(s):

Vasilii F. Otvagin ◽

Alexander V. Nyuchev ◽

Natalia S. Kuzmina ◽

Ivan D. Grishin ◽

Andrei E. Gavryushin ◽

...

Keyword(s):

Targeted Delivery ◽

Biological Evaluation ◽

Water Soluble ◽

Synthesis And Biological Evaluation

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Design, synthesis, and biological evaluation of water-soluble amino acid prodrug conjugates derived from combretastatin, dihydronaphthalene, and benzosuberene-based parent vascular disrupting agents

Bioorganic & Medicinal Chemistry ◽

10.1016/j.bmc.2016.01.007 ◽

2016 ◽

Vol 24 (5) ◽

pp. 938-956 ◽

Author(s):

Laxman Devkota ◽

Chen-Ming Lin ◽

Tracy E. Strecker ◽

Yifan Wang ◽

Justin K. Tidmore ◽

...

Keyword(s):

Biological Evaluation ◽

Water Soluble ◽

Vascular Disrupting Agents ◽

Design Synthesis ◽

Synthesis And Biological Evaluation ◽

Vascular Disrupting

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Lead structures for applications in photodynamic therapy. 5. Synthesis and biological evaluation of water soluble phosphorus(V) 5,10,15,20-tetraalkylporphyrins for PDT

Photodiagnosis and Photodynamic Therapy ◽

10.1016/j.pdpdt.2014.07.003 ◽

2014 ◽

Vol 11 (4) ◽

pp. 510-515 ◽

Author(s):

Aoife A. Ryan ◽

Mothi M. Ebrahim ◽

Rosine Petitdemange ◽

Gisela M. Vaz ◽

Edyta Paszko ◽

...

Keyword(s):

Photodynamic Therapy ◽

Biological Evaluation ◽

Water Soluble ◽

Soluble Phosphorus ◽

Synthesis And Biological Evaluation

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Development, synthesis, and biological evaluation of (-)-trans-(2S,5S)-2-[3-[(2-oxopropyl)sulfonyl]-4-n-propoxy-5-(3-hydroxypropoxy)-phenyl]-5-(3,4,5-trimethoxyphenyl)tetrahydrofuran, a potent orally active platelet-activating factor (PAF) antagonist and its water-soluble prodrug phosphate ester

Journal of Medicinal Chemistry ◽

10.1021/jm00097a005 ◽

1992 ◽

Vol 35 (19) ◽

pp. 3474-3482 ◽

Author(s):

N. N. Girotra ◽

T. Biftu ◽

M. M. Ponpipom ◽

J. J. Acton ◽

A. W. Alberts ◽

...

Keyword(s):

Platelet Activating Factor ◽

Biological Evaluation ◽

Water Soluble ◽

Phosphate Ester ◽

Orally Active ◽

Synthesis And Biological Evaluation

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Design, synthesis, and biological evaluation of novel water-soluble N-mustards as potential anticancer agents

Bioorganic & Medicinal Chemistry ◽

10.1016/j.bmc.2010.11.005 ◽

2011 ◽

Vol 19 (1) ◽

pp. 471-485 ◽

Author(s):

Naval Kapuriya ◽

Rajesh Kakadiya ◽

Huajin Dong ◽

Amit Kumar ◽

Pei-Chih Lee ◽

...

Keyword(s):

Anticancer Agents ◽

Biological Evaluation ◽

Water Soluble ◽

Design Synthesis ◽

Synthesis And Biological Evaluation

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Synthesis and biological evaluation of a water soluble phosphate prodrug of 3-aminopyridine-2-carboxaldehyde thiosemicarbazone (3-AP)

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/s0960-894x(98)00573-3 ◽

1998 ◽

Vol 8 (22) ◽

pp. 3159-3164 ◽

Author(s):

Jun Li ◽

Xiang Luo ◽

Qin Wang ◽

Li-mou Zheng ◽

I. King ◽

...

Keyword(s):

Biological Evaluation ◽

Water Soluble ◽

Soluble Phosphate ◽

Synthesis And Biological Evaluation

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