Opiate Aromatic Pharmacophore Structure−Activity Relationships in CTAP Analogues Determined by Topographical Bias, Two-Dimensional NMR, and Biological Activity Assays

2000 ◽  
Vol 43 (4) ◽  
pp. 569-580 ◽  
Author(s):  
G. Gregg Bonner ◽  
Peg Davis ◽  
Dagmar Stropova ◽  
Sidney Edsall ◽  
Henry I. Yamamura ◽  
...  
Keyword(s):  
Biological Activity ◽  
Two Dimensional ◽  
Structure Activity Relationships ◽  
Structure Activity

Design, synthesis and biological activities of pyrrole-3-carboxamide derivatives as EZH2 (enhancer of zeste homologue 2) inhibitors and anticancer agents

2020 ◽  
Vol 44 (6) ◽  
pp. 2247-2255
Author(s):  
Qifan Zhou ◽  
Lina Jia ◽  
Fangyu Du ◽  
Xiaoyu Dong ◽  
Wanyu Sun ◽  
...  
Keyword(s):  
Biological Activity ◽  
Anticancer Agents ◽  
Biological Activities ◽  
Activity Assay ◽  
Design Synthesis ◽  
Structure Activity Relationships ◽  
Structure Activity ◽  
Enhancer Of Zeste

A novel series of pyrrole-3-carboxamides targeting EZH2 have been designed and synthesized. The structure–activity relationships were summarized by combining with in vitro biological activity assay and docking results.

scholarly journals Brassinosteroid phytohormones: structure, bioactivity and applications

2002 ◽  
Vol 14 (3) ◽  
pp. 143-181 ◽  
Author(s):  
Marco António Teixeira Zullo ◽  
Günter Adam
Keyword(s):  
Biological Activity ◽  
Plant Growth ◽  
Plant Hormones ◽  
Natural Occurrence ◽  
Regulatory Activity ◽  
Structure Activity Relationships ◽  
New Class ◽  
Structure Activity ◽  
Activity Structure ◽  
Steroid Structure

Brassinosteroids are a new class of plant hormones with a polyoxygenated steroid structure showing pronounced plant growth regulatory activity. This review covers their natural occurrence, biological and chromatographic methods for their detection, biosynthesis and metabolism, biological activity, structure-activity relationships and prospective agricultural uses.

Adenosine receptors: synthesis, structure-activity relationships and biological activity of new 6-amino purine derivatives

1998 ◽  
Vol 33 (6) ◽  
pp. 501-508 ◽  
Author(s):  
Giovannella Strappaghetti ◽  
Stefano Corsano ◽  
Roberta Barbaro ◽  
Antonio Lucacchini ◽  
Gino Giannaccini ◽  
...  
Keyword(s):  
Biological Activity ◽  
Adenosine Receptors ◽  
Purine Derivatives ◽  
Structure Activity Relationships ◽  
Structure Activity

ChemInform Abstract: Adenosine Receptors: Synthesis, Structure-Activity Relationships and Biological Activity of New 6-Amino Purine Derivatives.

ChemInform ◽  
2010 ◽  
Vol 30 (3) ◽  
pp. no-no
Author(s):  
G. STRAPPAGHETTI ◽  
S. CORSANO ◽  
R. BARBARO ◽  
A. LUCACCHINI ◽  
G. GIANNACCINI ◽  
...  
Keyword(s):  
Biological Activity ◽  
Adenosine Receptors ◽  
Purine Derivatives ◽  
Structure Activity Relationships ◽  
Structure Activity

scholarly journals Bis-pyrazolylpyridine Complexes of Some Transition Metal Ions: Structure-Activity Relationships and Biological Activity

2020 ◽  
Vol 13 (3) ◽  
pp. 201-209
Author(s):  
Ana Rilak Simović ◽  
Jovana Bogojeski ◽  
Biljana Petrović ◽  
Snežana Jovanović-Stević
Keyword(s):  
Biological Activity ◽  
Transition Metal ◽  
Metal Ions ◽  
Transition Metal Ions ◽  
Structure Activity Relationships ◽  
Structure Activity
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