scholarly journals Brassinosteroid phytohormones: structure, bioactivity and applications

2002 ◽  
Vol 14 (3) ◽  
pp. 143-181 ◽  
Author(s):  
Marco António Teixeira Zullo ◽  
Günter Adam
Keyword(s):  
Biological Activity ◽  
Plant Growth ◽  
Plant Hormones ◽  
Natural Occurrence ◽  
Regulatory Activity ◽  
Structure Activity Relationships ◽  
New Class ◽  
Structure Activity ◽  
Activity Structure ◽  
Steroid Structure

Brassinosteroids are a new class of plant hormones with a polyoxygenated steroid structure showing pronounced plant growth regulatory activity. This review covers their natural occurrence, biological and chromatographic methods for their detection, biosynthesis and metabolism, biological activity, structure-activity relationships and prospective agricultural uses.

scholarly journals Recent development of lipoxygenase inhibitors as anti-inflammatory agents

MedChemComm ◽  
2018 ◽  
Vol 9 (2) ◽  
pp. 212-225 ◽  
Author(s):  
Chaoyu Hu ◽  
Shutao Ma
Keyword(s):  
Biological Activity ◽  
Molecular Docking ◽  
Docking Studies ◽  
Lipoxygenase Inhibitors ◽  
Molecular Docking Studies ◽  
Structure Activity Relationships ◽  
Structure Activity ◽  
Activity Structure ◽  
Recent Developments ◽  
Lox Inhibitors

This review summarizes recent developments of LOX inhibitors. It also contains an introduction to their structures, biological activity, structure–activity relationships and molecular docking studies.

scholarly journals Re-Engineering of Yohimbine’s Biological Activity through Ring Distortion: Identification and Structure–Activity Relationships of a New Class of Antiplasmodial Agents

2020 ◽  
Vol 6 (2) ◽  
pp. 159-167 ◽  
Author(s):  
Nicholas G. Paciaroni ◽  
David L. Perry ◽  
Verrill M. Norwood ◽  
Claribel Murillo-Solano ◽  
Jennifer Collins ◽  
...  
Keyword(s):  
Biological Activity ◽  
Structure Activity Relationships ◽  
New Class ◽  
Structure Activity ◽  
Ring Distortion

Design, synthesis and biological activities of pyrrole-3-carboxamide derivatives as EZH2 (enhancer of zeste homologue 2) inhibitors and anticancer agents

2020 ◽  
Vol 44 (6) ◽  
pp. 2247-2255
Author(s):  
Qifan Zhou ◽  
Lina Jia ◽  
Fangyu Du ◽  
Xiaoyu Dong ◽  
Wanyu Sun ◽  
...  
Keyword(s):  
Biological Activity ◽  
Anticancer Agents ◽  
Biological Activities ◽  
Activity Assay ◽  
Design Synthesis ◽  
Structure Activity Relationships ◽  
Structure Activity ◽  
Enhancer Of Zeste

A novel series of pyrrole-3-carboxamides targeting EZH2 have been designed and synthesized. The structure–activity relationships were summarized by combining with in vitro biological activity assay and docking results.

Bis(phenazine-1-carboxamides):  Structure−Activity Relationships for a New Class of Dual Topoisomerase I/II-Directed Anticancer Drugs

2000 ◽  
Vol 43 (7) ◽  
pp. 1350-1358 ◽  
Author(s):  
Julie A. Spicer ◽  
Swarna A. Gamage ◽  
Gordon W. Rewcastle ◽  
Graeme J. Finlay ◽  
David J. A. Bridewell ◽  
...  
Keyword(s):  
Anticancer Drugs ◽  
Topoisomerase I ◽  
Structure Activity Relationships ◽  
New Class ◽  
Structure Activity
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